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Found 47 with Last Name = 'nistri' and Initial = 'a'
TargetP2X purinoceptor 3(Mus musculus)
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535408(CHEMBL4462568)
Affinity DataIC50:  24nMAssay Description:Antagonist activity at P2X3R in mouse TG sensory neurons assessed as inhibition of P2X3R agonist alpha,beta-meATP-induced current at -65 mV holding p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Mus musculus)
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535414(CHEMBL4463334)
Affinity DataIC50:  81nMAssay Description:Antagonist activity at P2X3R in mouse TG sensory neurons assessed as inhibition of P2X3R agonist alpha,beta-meATP-induced current at -65 mV holding p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Mus musculus)
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535410(CHEMBL4525343)
Affinity DataIC50:  83nMAssay Description:Antagonist activity at P2X3R in mouse TG sensory neurons assessed as inhibition of P2X3R agonist alpha,beta-meATP-induced current at -65 mV holding p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Mus musculus)
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535415(CHEMBL4463578)
Affinity DataIC50:  127nMAssay Description:Antagonist activity at P2X3R in mouse TG sensory neurons assessed as inhibition of P2X3R agonist alpha,beta-meATP-induced current at -65 mV holding p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Mus musculus)
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535409(CHEMBL4456926)
Affinity DataIC50:  211nMAssay Description:Antagonist activity at P2X3R in mouse TG sensory neurons assessed as inhibition of P2X3R agonist alpha,beta-meATP-induced current at -65 mV holding p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535414(CHEMBL4463334)
Affinity DataIC50:  611nMAssay Description:Antagonist activity at human P2X3R transfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influxMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535410(CHEMBL4525343)
Affinity DataIC50:  883nMAssay Description:Antagonist activity at human P2X3R transfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influxMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Mus musculus)
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535413(CHEMBL4561510)
Affinity DataIC50: >1.00E+3nMAssay Description:Antagonist activity at P2X3R in mouse TG sensory neurons assessed as inhibition of P2X3R agonist alpha,beta-meATP-induced current at -65 mV holding p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50436790(CHEMBL2402580)
Affinity DataIC50:  1.74E+3nMAssay Description:Antagonist activity at rat recombinant P2X3 receptor expressed in HEK293T cells assessed as desensitization of alpha,beta-methyleneATP-induced curren...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50436788(CHEMBL2402587)
Affinity DataIC50:  2.23E+3nMAssay Description:Antagonist activity at rat recombinant P2X3 receptor expressed in HEK293T cells assessed as desensitization of alpha,beta-methyleneATP-induced curren...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535408(CHEMBL4462568)
Affinity DataIC50:  4.11E+3nMAssay Description:Antagonist activity at human P2X3R transfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influxMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535409(CHEMBL4456926)
Affinity DataIC50:  5.83E+3nMAssay Description:Antagonist activity at human P2X3R transfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influxMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 1(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535410(CHEMBL4525343)
Affinity DataIC50:  8.06E+3nMAssay Description:Antagonist activity at human P2X1R transfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influxMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535414(CHEMBL4463334)
Affinity DataIC50:  8.53E+3nMAssay Description:Antagonist activity at human P2X7R transfected in human 1321N1 cells assessed as inhibition of Bz-ATP-induced calcium influxMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 2(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535412(CHEMBL4570607)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human P2X2R transfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influxMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 1(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535412(CHEMBL4570607)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human P2X1R transfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influxMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535414(CHEMBL4463334)
Affinity DataIC50:  1.10E+4nMAssay Description:Antagonist activity at human P2X4R transfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influxMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535409(CHEMBL4456926)
Affinity DataIC50:  1.24E+4nMAssay Description:Antagonist activity at human P2X4R transfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influxMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535415(CHEMBL4463578)
Affinity DataIC50:  1.75E+4nMAssay Description:Antagonist activity at human P2X3R transfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influxMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50436789(CHEMBL2402586)
Affinity DataIC50:  1.86E+4nMAssay Description:Antagonist activity at rat recombinant P2X3 receptor expressed in HEK293T cells assessed as desensitization of alpha,beta-methyleneATP-induced curren...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535410(CHEMBL4525343)
Affinity DataIC50:  2.96E+4nMAssay Description:Antagonist activity at human P2X4R transfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influxMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535411(CHEMBL4440260)
Affinity DataIC50: >3.00E+4nMAssay Description:Antagonist activity at human P2X7R transfected in human 1321N1 cells assessed as inhibition of Bz-ATP-induced calcium influxMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535412(CHEMBL4570607)
Affinity DataIC50: >3.00E+4nMAssay Description:Antagonist activity at human P2X7R transfected in human 1321N1 cells assessed as inhibition of Bz-ATP-induced calcium influxMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535412(CHEMBL4570607)
Affinity DataIC50: >3.00E+4nMAssay Description:Antagonist activity at human P2X4R transfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influxMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 1(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535408(CHEMBL4462568)
Affinity DataIC50:  4.11E+4nMAssay Description:Antagonist activity at human P2X1R transfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influxMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535408(CHEMBL4462568)
Affinity DataIC50:  4.80E+4nMAssay Description:Antagonist activity at human P2X4R transfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influxMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 2(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535410(CHEMBL4525343)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human P2X2R transfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influxMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 2(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535415(CHEMBL4463578)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human P2X2R transfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influxMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535415(CHEMBL4463578)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human P2X7R transfected in human 1321N1 cells assessed as inhibition of Bz-ATP-induced calcium influxMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535410(CHEMBL4525343)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human P2X7R transfected in human 1321N1 cells assessed as inhibition of Bz-ATP-induced calcium influxMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535411(CHEMBL4440260)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human P2X4R transfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influxMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 1(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535415(CHEMBL4463578)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human P2X1R transfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influxMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 2(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535409(CHEMBL4456926)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human P2X2R transfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influxMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535413(CHEMBL4561510)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human P2X7R transfected in human 1321N1 cells assessed as inhibition of Bz-ATP-induced calcium influxMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535415(CHEMBL4463578)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human P2X4R transfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influxMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 4(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535413(CHEMBL4561510)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human P2X4R transfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influxMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535409(CHEMBL4456926)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human P2X7R transfected in human 1321N1 cells assessed as inhibition of Bz-ATP-induced calcium influxMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535413(CHEMBL4561510)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human P2X3R transfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influxMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 1(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535413(CHEMBL4561510)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human P2X1R transfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influxMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 1(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535411(CHEMBL4440260)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human P2X1R transfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influxMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 2(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535414(CHEMBL4463334)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human P2X2R transfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influxMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 2(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535413(CHEMBL4561510)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human P2X2R transfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influxMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 2(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535411(CHEMBL4440260)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human P2X2R transfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influxMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535408(CHEMBL4462568)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human P2X7R transfected in human 1321N1 cells assessed as inhibition of Bz-ATP-induced calcium influxMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 1(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535409(CHEMBL4456926)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human P2X1R transfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influxMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 2(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535408(CHEMBL4462568)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human P2X2R transfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influxMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50535411(CHEMBL4440260)
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human P2X3R transfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influxMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed