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Found 592 with Last Name = 'o''connell' and Initial = 'j'
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283704((R)-N*1*-[(S)-2-Cyclohexyl-1-(2-morpholin-4-yl-eth...)
Affinity DataKi:  0.0100nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283703((R)-N*1*-{(S)-2-Cyclohexyl-1-[2-(4-sulfamoyl-pheny...)
Affinity DataKi:  0.0100nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283701(3-{(S)-2-[(R)-5-(4-Chloro-phenyl)-2-hydroxycarbamo...)
Affinity DataKi:  0.0100nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283708(3-{(S)-2-[(R)-5-(4-Chloro-phenyl)-2-hydroxycarbamo...)
Affinity DataKi:  0.0100nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283705((R)-2-[3-(4-Chloro-phenyl)-propyl]-N*1*-{(S)-2-cyc...)
Affinity DataKi:  0.0100nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283715((R)-N*1*-{(S)-2-Cyclohexyl-1-[2-(morpholine-4-sulf...)
Affinity DataKi:  0.0100nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283711((R)-2-[3-(4-Chloro-phenyl)-propyl]-N*1*-[(S)-2-cyc...)
Affinity DataKi:  0.0200nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283710((R)-N*1*-[(S)-2-Cyclohexyl-1-(4-morpholin-4-yl-but...)
Affinity DataKi:  0.0200nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283713((R)-N*1*-[(S)-2-Cyclohexyl-1-(4-dimethylamino-buty...)
Affinity DataKi:  0.0200nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283707((R)-2-[3-(4-Chloro-phenyl)-propyl]-N*1*-[(S)-2-cyc...)
Affinity DataKi:  0.0300nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50101495((R)-2-[3-(4-Chloro-phenyl)-propyl]-N*1*-((S)-2-cyc...)
Affinity DataKi:  0.0300nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283702((R)-2-[3-(4-Chloro-phenyl)-propyl]-N*1*-{(S)-2-cyc...)
Affinity DataKi:  0.0300nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283714((R)-2-[3-(4-Chloro-phenyl)-propyl]-N*1*-[(S)-2-cyc...)
Affinity DataKi:  0.0500nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50101492((R)-N*1*-((S)-2-Cyclohexyl-1-phenethylcarbamoyl-et...)
Affinity DataKi:  0.0600nMAssay Description:Inhibition of the Gelatinase-A enzyme was determined from purified NSO cells.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50101526((R)-N*1*-((S)-2-Cyclohexyl-1-phenethylcarbamoyl-et...)
Affinity DataKi:  0.0600nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50101530((R)-N*1*-((S)-2-Cyclohexyl-1-phenethylcarbamoyl-et...)
Affinity DataKi:  0.0600nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50101492((R)-N*1*-((S)-2-Cyclohexyl-1-phenethylcarbamoyl-et...)
Affinity DataKi:  0.0620nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50101513((R)-N*1*-((S)-2-Cyclohexyl-1-phenethylcarbamoyl-et...)
Affinity DataKi:  0.0800nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50101494((R)-N*1*-((S)-2-Cyclohexyl-1-phenethylcarbamoyl-et...)
Affinity DataKi:  0.100nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50101528((R)-N*1*-((S)-2-Cyclohexyl-1-phenethylcarbamoyl-et...)
Affinity DataKi:  0.254nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50101510((R)-N*1*-((S)-2-Cyclohexyl-1-phenethylcarbamoyl-et...)
Affinity DataKi:  0.300nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50101529((R)-N*1*-((S)-2-Cyclohexyl-1-phenethylcarbamoyl-et...)
Affinity DataKi:  0.330nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283712(4-{2-[(S)-3-Cyclohexyl-2-((R)-2-hydroxycarbamoylme...)
Affinity DataKi:  0.590nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283701(3-{(S)-2-[(R)-5-(4-Chloro-phenyl)-2-hydroxycarbamo...)
Affinity DataKi:  0.800nMAssay Description:Inhibition of the stromelysin enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50101523((R)-3-{(S)-2-Cyclohexyl-1-[2-(4-sulfamoyl-phenyl)-...)
Affinity DataKi:  0.900nMAssay Description:Inhibition of the Gelatinase-A enzyme was determined from purified NSO cells.More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283708(3-{(S)-2-[(R)-5-(4-Chloro-phenyl)-2-hydroxycarbamo...)
Affinity DataKi:  0.960nMAssay Description:Inhibition of the stromelysin enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50101515((R)-3-(((S)-3-cyclohexyl-1-oxo-1-(phenethylamino)p...)
Affinity DataKi:  1nMAssay Description:Inhibition of the Gelatinase-A enzyme was determined from purified NSO cells.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50101525((R)-6-(4-Chloro-phenyl)-3-{(S)-2-cyclohexyl-1-[2-(...)
Affinity DataKi:  1nMAssay Description:Inhibition of the Gelatinase-A enzyme was determined from purified NSO cells.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50101496((R)-3-(((S)-3-cyclohexyl-1-(3-methoxy-3-oxopropyla...)
Affinity DataKi:  1.20nMAssay Description:Inhibition of the Gelatinase-A enzyme was determined from purified NSO cells.More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283711((R)-2-[3-(4-Chloro-phenyl)-propyl]-N*1*-[(S)-2-cyc...)
Affinity DataKi:  1.40nMAssay Description:Inhibition of the stromelysin enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283705((R)-2-[3-(4-Chloro-phenyl)-propyl]-N*1*-{(S)-2-cyc...)
Affinity DataKi:  1.70nMAssay Description:Inhibition of the stromelysin enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50101521((R)-3-{(S)-2-Cyclohexyl-1-[2-(4-sulfamoyl-phenyl)-...)
Affinity DataKi:  1.80nMAssay Description:Inhibition of the Gelatinase-A enzyme was determined from purified NSO cells.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50101514((R)-N*1*-((S)-2-Cyclohexyl-1-phenethylcarbamoyl-et...)
Affinity DataKi:  2.20nMAssay Description:Inhibition of the gelatinase-A enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283707((R)-2-[3-(4-Chloro-phenyl)-propyl]-N*1*-[(S)-2-cyc...)
Affinity DataKi:  2.40nMAssay Description:Inhibition of the stromelysin enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50101522(CHEMBL76869 | [(S)-2-((S)-2-Cyclohexyl-1-phenethyl...)
Affinity DataKi:  2.5nMAssay Description:Inhibition of the Collagenase enzyme was determined from purified NSO cells.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50101522(CHEMBL76869 | [(S)-2-((S)-2-Cyclohexyl-1-phenethyl...)
Affinity DataKi:  2.5nMAssay Description:Inhibition of the Gelatinase-A enzyme was determined from purified NSO cells.More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283710((R)-N*1*-[(S)-2-Cyclohexyl-1-(4-morpholin-4-yl-but...)
Affinity DataKi:  2.60nMAssay Description:Inhibition of the stromelysin enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283715((R)-N*1*-{(S)-2-Cyclohexyl-1-[2-(morpholine-4-sulf...)
Affinity DataKi:  2.80nMAssay Description:Inhibition of the stromelysin enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50087826(CHEMBL3426789)
Affinity DataKi:  3nMAssay Description:Positive allosteric modulation of human delta opioid receptor expressed in CHO cell membranes assessed as TAN67 Ki at 10 uM after 90 mins by [3H]-dip...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283703((R)-N*1*-{(S)-2-Cyclohexyl-1-[2-(4-sulfamoyl-pheny...)
Affinity DataKi:  3nMAssay Description:Inhibition of the stromelysin enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50101501((R)-3-(((S)-1-(4-amino-4-oxobutylamino)-3-cyclohex...)
Affinity DataKi:  3.10nMAssay Description:Inhibition of the Gelatinase-A enzyme was determined from purified NSO cells.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50101524((R)-3-(((S)-1-(2-carboxyethylamino)-3-cyclohexyl-1...)
Affinity DataKi:  3.80nMAssay Description:Inhibition of the Gelatinase-A enzyme was determined from purified NSO cells.More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50101530((R)-N*1*-((S)-2-Cyclohexyl-1-phenethylcarbamoyl-et...)
Affinity DataKi:  4.20nMAssay Description:Inhibition of the stromelysin enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50087826(CHEMBL3426789)
Affinity DataKi:  5nMAssay Description:Positive allosteric modulation of human delta opioid receptor expressed in CHO cell membranes assessed as SNC80 Ki at 10 uM after 90 mins by [3H]-dip...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50101494((R)-N*1*-((S)-2-Cyclohexyl-1-phenethylcarbamoyl-et...)
Affinity DataKi:  5.40nMAssay Description:Inhibition of the stromelysin enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283713((R)-N*1*-[(S)-2-Cyclohexyl-1-(4-dimethylamino-buty...)
Affinity DataKi:  5.90nMAssay Description:Inhibition of the stromelysin enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50101507((R)-3-(((S)-3-cyclohexyl-1-(3-methoxy-3-oxopropyla...)
Affinity DataKi:  6nMAssay Description:Inhibition of the Gelatinase-A enzyme was determined from purified NSO cells.More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283704((R)-N*1*-[(S)-2-Cyclohexyl-1-(2-morpholin-4-yl-eth...)
Affinity DataKi:  6.30nMAssay Description:Inhibition of the stromelysin enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50101506((R)-3-{(S)-2-cyclohexyl-1-[2-(4-sulfamoyl-phenyl)-...)
Affinity DataKi:  6.40nMAssay Description:Inhibition of the Gelatinase-A enzyme was determined from purified NSO cells.More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283702((R)-2-[3-(4-Chloro-phenyl)-propyl]-N*1*-{(S)-2-cyc...)
Affinity DataKi:  6.40nMAssay Description:Inhibition of the stromelysin enzyme.More data for this Ligand-Target Pair
In DepthDetails Article
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