Compile Data Set for Download or QSAR
maximum 50k data
Found 89 with Last Name = 'oamppound39malley' and Initial = 'cf'
LigandPNGBDBM27476(2-amino-5-(pyridin-4-yl)-3-(4-sulfamoylphenyl)benz...)
Affinity DataIC50:  79nMpH: 7.4 T: 2°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM27467(2-amino-5-(4-chlorophenyl)-3-(4-sulfamoylphenyl)be...)
Affinity DataIC50:  100nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM27477(2-amino-5-(4-methanesulfonylphenyl)-3-(4-sulfamoyl...)
Affinity DataIC50:  158nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM27489(2-amino-3-{4-[(2-aminoethyl)sulfamoyl]phenyl}-5-ph...)
Affinity DataIC50:  158nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM27466(2-amino-5-(4-fluorophenyl)-3-(4-sulfamoylphenyl)be...)
Affinity DataIC50:  200nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM27490(2-amino-3-{4-[(3-methoxypropyl)sulfamoyl]phenyl}-5...)
Affinity DataIC50:  251nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM27471(2-amino-5-phenyl-3-(4-sulfamoylphenyl)benzamide | ...)
Affinity DataIC50:  251nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM27476(2-amino-5-(pyridin-4-yl)-3-(4-sulfamoylphenyl)benz...)
Affinity DataIC50:  251nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM27492(2-amino-5-phenyl-3-(4-{[2-(pyrrolidin-1-yl)ethyl]s...)
Affinity DataIC50:  251nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM27487(2-amino-3-(4-{[3-(dimethylamino)propyl]sulfamoyl}p...)
Affinity DataIC50:  316nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM27491(2-amino-3-[4-(cyclopropylsulfamoyl)phenyl]-5-pheny...)
Affinity DataIC50:  316nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM27488(2-amino-3-(4-{[3-(morpholin-4-yl)propyl]sulfamoyl}...)
Affinity DataIC50:  316nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM27467(2-amino-5-(4-chlorophenyl)-3-(4-sulfamoylphenyl)be...)
Affinity DataIC50:  398nMpH: 7.4 T: 2°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM27478(2-amino-5-(4-methanesulfonylphenyl)-3-[4-(pyrrolid...)
Affinity DataIC50:  398nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM27466(2-amino-5-(4-fluorophenyl)-3-(4-sulfamoylphenyl)be...)
Affinity DataIC50:  501nMpH: 7.4 T: 2°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM27489(2-amino-3-{4-[(2-aminoethyl)sulfamoyl]phenyl}-5-ph...)
Affinity DataIC50:  631nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM27465(2-amino-5-(4-fluorophenyl)-3-[4-(pyrrolidine-1-sul...)
Affinity DataIC50:  631nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM27492(2-amino-5-phenyl-3-(4-{[2-(pyrrolidin-1-yl)ethyl]s...)
Affinity DataIC50:  794nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM27490(2-amino-3-{4-[(3-methoxypropyl)sulfamoyl]phenyl}-5...)
Affinity DataIC50:  794nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM27471(2-amino-5-phenyl-3-(4-sulfamoylphenyl)benzamide | ...)
Affinity DataIC50:  1.00E+3nMpH: 7.4 T: 2°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
LigandPNGBDBM27485(2-hydroxy-3-(4-methanesulfonamidophenyl)-5-phenylb...)
Affinity DataIC50:  1.00E+3nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM27488(2-amino-3-(4-{[3-(morpholin-4-yl)propyl]sulfamoyl}...)
Affinity DataIC50:  1.00E+3nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM27487(2-amino-3-(4-{[3-(dimethylamino)propyl]sulfamoyl}p...)
Affinity DataIC50:  1.00E+3nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM27491(2-amino-3-[4-(cyclopropylsulfamoyl)phenyl]-5-pheny...)
Affinity DataIC50:  1.00E+3nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM27469(2-amino-3-(4-methanesulfonamidophenyl)-5-phenylben...)
Affinity DataIC50:  1.59E+3nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM27468(2-amino-5-(4-chlorophenyl)-3-(4-methanesulfonamido...)
Affinity DataIC50:  1.59E+3nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM27464(2-amino-5-(4-fluorophenyl)-3-(pyridin-4-yl)benzami...)
Affinity DataIC50:  1.59E+3nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM27476(2-amino-5-(pyridin-4-yl)-3-(4-sulfamoylphenyl)benz...)
Affinity DataIC50:  1.59E+3nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM27484(5-(4-chlorophenyl)-2-hydroxy-3-(4-sulfamoylphenyl)...)
Affinity DataIC50:  1.59E+3nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM27477(2-amino-5-(4-methanesulfonylphenyl)-3-(4-sulfamoyl...)
Affinity DataIC50:  2.00E+3nMpH: 7.4 T: 2°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM27484(5-(4-chlorophenyl)-2-hydroxy-3-(4-sulfamoylphenyl)...)
Affinity DataIC50:  2.00E+3nMpH: 7.4 T: 2°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM27485(2-hydroxy-3-(4-methanesulfonamidophenyl)-5-phenylb...)
Affinity DataIC50:  2.00E+3nMpH: 7.4 T: 2°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM27465(2-amino-5-(4-fluorophenyl)-3-[4-(pyrrolidine-1-sul...)
Affinity DataIC50:  2.51E+3nMpH: 7.4 T: 2°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM27475(2-amino-3-phenyl-5-(pyridin-4-yl)benzamide | Amino...)
Affinity DataIC50:  3.16E+3nMpH: 7.4 T: 2°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM27475(2-amino-3-phenyl-5-(pyridin-4-yl)benzamide | Amino...)
Affinity DataIC50:  3.98E+3nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM27473(2-amino-5-phenyl-3-[4-(sulfamoylmethyl)phenyl]benz...)
Affinity DataIC50:  3.98E+3nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM27475(2-amino-3-phenyl-5-(pyridin-4-yl)benzamide | Amino...)
Affinity DataIC50:  3.98E+3nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM27464(2-amino-5-(4-fluorophenyl)-3-(pyridin-4-yl)benzami...)
Affinity DataIC50:  5.01E+3nMpH: 7.4 T: 2°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM27486(3-[4-(dimethylsulfamoyl)phenyl]-2-hydroxy-5-(pyrid...)
Affinity DataIC50:  5.01E+3nMpH: 7.4 T: 2°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM27478(2-amino-5-(4-methanesulfonylphenyl)-3-[4-(pyrrolid...)
Affinity DataIC50:  5.01E+3nMpH: 7.4 T: 2°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM27468(2-amino-5-(4-chlorophenyl)-3-(4-methanesulfonamido...)
Affinity DataIC50:  6.31E+3nMpH: 7.4 T: 2°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM27486(3-[4-(dimethylsulfamoyl)phenyl]-2-hydroxy-5-(pyrid...)
Affinity DataIC50:  7.94E+3nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM27470(2-amino-3-(3-methanesulfonamidophenyl)-5-phenylben...)
Affinity DataIC50:  7.94E+3nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM27472(2-amino-5-phenyl-3-(3-sulfamoylphenyl)benzamide | ...)
Affinity DataIC50:  7.94E+3nMAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM27473(2-amino-5-phenyl-3-[4-(sulfamoylmethyl)phenyl]benz...)
Affinity DataIC50:  7.94E+3nMpH: 7.4 T: 2°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM27470(2-amino-3-(3-methanesulfonamidophenyl)-5-phenylben...)
Affinity DataIC50:  1.00E+4nMpH: 7.4 T: 2°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM27469(2-amino-3-(4-methanesulfonamidophenyl)-5-phenylben...)
Affinity DataIC50:  1.26E+4nMpH: 7.4 T: 2°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM27460(2-amino-5-(4-fluorophenyl)-3-(4-methanesulfonylphe...)
Affinity DataIC50: >1.58E+4nMpH: 7.4 T: 2°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM27461(2-amino-5-(4-fluorophenyl)-N-methyl-3-[4-(pyrrolid...)
Affinity DataIC50: >1.58E+4nMpH: 7.4 T: 2°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM27462(2-amino-5-phenylbenzamide | Amino-substituted benz...)
Affinity DataIC50: >1.58E+4nMpH: 7.4 T: 2°CAssay Description:IKK kinase activity was assessed using a time-resolved fluorescence resonance energy transfer (TR-FRET) assay. The reaction was initiated by the addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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