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Found 31 with Last Name = 'ochiai' and Initial = 'e'
TargetVitamin D3 receptor(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50262540((3S,5S)-5-((R)-2-((1R,3aS,7aR)-4-(2-((3S,5R)-3,5-d...)
Affinity DataIC50:  207nMAssay Description:Antagonist activity assessed by differentiation of 1,25-D3-induced HL60 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50262542((3S,5S)-5-((R)-2-((1R,3aS,7aR)-4-(2-((3S,5R)-3,5-d...)
Affinity DataIC50:  390nMAssay Description:Antagonist activity assessed by differentiation of 1,25-D3-induced HL60 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50410853(CHEMBL203485)
Affinity DataIC50:  660nMAssay Description:Antagonist activity assessed by differentiation of 1,25-D3-induced HL60 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50262539((3S,5S)-1-benzyl-5-((R)-2-((1R,3aS,7aR)-4-(2-((3S,...)
Affinity DataIC50:  700nMAssay Description:Antagonist activity assessed by differentiation of 1,25-D3-induced HL60 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50410854(CHEMBL383450)
Affinity DataIC50: >1.00E+3nMAssay Description:Antagonist activity assessed by differentiation of 1,25-D3-induced HL60 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50313152((3R,5S)-5-((R)-2-((1R,3aS,7aR,E)-4-((Z)-2-((3S,5R)...)
Affinity DataIC50: >2.00E+3nMAssay Description:Antagonist activity assessed by differentiation of 1,25-D3-induced HL60 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50262541((3S,5S)-5-((R)-2-((1R,3aS,7aR)-4-(2-((3S,5R)-3,5-d...)
Affinity DataIC50:  2.20E+3nMAssay Description:Antagonist activity assessed by differentiation of 1,25-D3-induced HL60 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)
Affinity DataEC50:  0.0100nMAssay Description:Activity at human VDR expressed in human HOS cells transfected with pGL3-hOc, pCDNA-hVDR and phRL-TK assessed as assessed as transcriptional activati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetVitamin D3 receptor(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50437333(CHEMBL2407826)
Affinity DataEC50:  0.680nMAssay Description:Transactivation of VDR-mediated osteocalcin promoter in human HOS/SF cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50437334(CHEMBL2407825)
Affinity DataEC50:  0.210nMAssay Description:Transactivation of VDR-mediated osteocalcin promoter in human HOS/SF cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50437335(CHEMBL2407824)
Affinity DataEC50:  0.0440nMAssay Description:Transactivation of VDR-mediated osteocalcin promoter in human HOS/SF cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50437336(CHEMBL2407823)
Affinity DataEC50:  0.150nMAssay Description:Transactivation of VDR-mediated osteocalcin promoter in human HOS/SF cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50437337(CHEMBL2407822)
Affinity DataEC50:  0.290nMAssay Description:Transactivation of VDR-mediated osteocalcin promoter in human HOS/SF cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50437338(CHEMBL2407821)
Affinity DataEC50:  0.0100nMAssay Description:Transactivation of VDR-mediated osteocalcin promoter in human HOS/SF cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)
Affinity DataEC50:  0.0260nMAssay Description:Transactivation of VDR-mediated osteocalcin promoter in human HOS/SF cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetVitamin D3 receptor(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50520855(CHEMBL4449172)
Affinity DataEC50:  77nMAssay Description:Agonist activity at human VDR expressed in HOS cells co-expressing human RXR by Dual-Glo luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50520856(CHEMBL4437809)
Affinity DataEC50:  42nMAssay Description:Agonist activity at human VDR expressed in HOS cells co-expressing human RXR by Dual-Glo luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50520857(CHEMBL4435565)
Affinity DataEC50:  17nMAssay Description:Agonist activity at human VDR expressed in HOS cells co-expressing human RXR by Dual-Glo luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50520858(CHEMBL4538386)
Affinity DataEC50:  18nMAssay Description:Agonist activity at human VDR expressed in HOS cells co-expressing human RXR by Dual-Glo luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50520859(CHEMBL4524433)
Affinity DataEC50:  163nMAssay Description:Agonist activity at human VDR expressed in HOS cells co-expressing human RXR by Dual-Glo luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50329706((2S)-3-{4-[1-ethyl-1-(4-{[(2R)-2-hydroxy-3,3-dimet...)
Affinity DataEC50:  0.0400nMAssay Description:Agonist activity at human VDR expressed in HOS cells co-expressing human RXR by Dual-Glo luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50520860(CHEMBL4558352)
Affinity DataEC50:  77nMAssay Description:Agonist activity at human VDR expressed in HOS cells co-expressing human RXR by Dual-Glo luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50520861(CHEMBL4583069)
Affinity DataEC50:  9.30nMAssay Description:Agonist activity at human VDR expressed in HOS cells co-expressing human RXR by Dual-Glo luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50329706((2S)-3-{4-[1-ethyl-1-(4-{[(2R)-2-hydroxy-3,3-dimet...)
Affinity DataEC50:  0.0400nMAssay Description:Activity at human VDR expressed in human HOS cells transfected with pGL3-hOc, pCDNA-hVDR and phRL-TK assessed as assessed as transcriptional activati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50354991(CHEMBL1834894)
Affinity DataEC50:  1.29nMAssay Description:Activity at human VDR expressed in human HOS cells transfected with pGL3-hOc, pCDNA-hVDR and phRL-TK assessed as assessed as transcriptional activati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50354990(CHEMBL1834893)
Affinity DataEC50:  0.0600nMAssay Description:Activity at human VDR expressed in human HOS cells transfected with pGL3-hOc, pCDNA-hVDR and phRL-TK assessed as assessed as transcriptional activati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50354989(CHEMBL1834892)
Affinity DataEC50:  1.25nMAssay Description:Activity at human VDR expressed in human HOS cells transfected with pGL3-hOc, pCDNA-hVDR and phRL-TK assessed as assessed as transcriptional activati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50354988(CHEMBL1834891)
Affinity DataEC50:  0.920nMAssay Description:Activity at human VDR expressed in human HOS cells transfected with pGL3-hOc, pCDNA-hVDR and phRL-TK assessed as assessed as transcriptional activati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)
Affinity DataEC50:  0.0110nMAssay Description:Agonist activity at human VDR expressed in HOS cells co-expressing human RXR by Dual-Glo luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetVitamin D3 receptor(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50354986(CHEMBL1834889)
Affinity DataEC50:  19.4nMAssay Description:Activity at human VDR expressed in human HOS cells transfected with pGL3-hOc, pCDNA-hVDR and phRL-TK assessed as assessed as transcriptional activati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50354987(CHEMBL1834890)
Affinity DataEC50:  1.11nMAssay Description:Activity at human VDR expressed in human HOS cells transfected with pGL3-hOc, pCDNA-hVDR and phRL-TK assessed as assessed as transcriptional activati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed