Compile Data Set for Download or QSAR
maximum 50k data
Found 93 with Last Name = 'okawara' and Initial = 't'
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50142519(CHEMBL47027 | N-[2-(3,4,5-triihydroxy-benzoylamino...)
Affinity DataKi:  400nMAssay Description:Inhibition of relaxation activities of DNA topoisomerase I with respect to pBR322 DNAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha/2-beta(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50142519(CHEMBL47027 | N-[2-(3,4,5-triihydroxy-benzoylamino...)
Affinity DataKi:  7.41E+4nMAssay Description:Inhibition of relaxation activities of DNA topoisomerase II with respect to pBR322 DNAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha/2-beta(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50142519(CHEMBL47027 | N-[2-(3,4,5-triihydroxy-benzoylamino...)
Affinity DataIC50:  9nMAssay Description:Inhibitory concentration against relaxation activity of DNA topoisomerase II by detecting the conversion of supercoiled pBR322 DNA to its relaxed for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly(ADP-ribose) glycohydrolase(Rattus norvegicus)
Kumamoto Health Science University

Curated by ChEMBL
LigandPNGBDBM50350107(CHEMBL1230692)
Affinity DataIC50:  100nMAssay Description:Inhibition of rat testis GST-tagged PARG catalytic activity after 30 mins using [32P]poly(ADP-ribose) by radioassayMore data for this Ligand-Target Pair
TargetDNA topoisomerase 2-alpha/2-beta(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50142517(CHEMBL47885 | N-[4-(3,4,5-triihydroxy-benzoylamino...)
Affinity DataIC50:  150nMAssay Description:Inhibitory concentration against relaxation activity of DNA topoisomerase II by detecting the conversion of supercoiled pBR322 DNA to its relaxed for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha/2-beta(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50142507(CHEMBL47526 | N-[3-(3,4,5-triihydroxy-benzoylamino...)
Affinity DataIC50:  220nMAssay Description:Inhibitory concentration against relaxation activity of DNA topoisomerase II by detecting the conversion of supercoiled pBR322 DNA to its relaxed for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50142519(CHEMBL47027 | N-[2-(3,4,5-triihydroxy-benzoylamino...)
Affinity DataIC50:  900nMAssay Description:Inhibitory concentration against relaxation activity of DNA topoisomerase I by detecting the conversion of supercoiled pBR322 DNA to its relaxed formMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly(ADP-ribose) glycohydrolase(Rattus norvegicus)
Kumamoto Health Science University

Curated by ChEMBL
LigandPNGBDBM50052832(CHEMBL3318753)
Affinity DataIC50:  950nMAssay Description:Inhibition of rat testis GST-tagged PARG catalytic activity after 30 mins using [32P]poly(ADP-ribose) by radioassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly(ADP-ribose) glycohydrolase(Rattus norvegicus)
Kumamoto Health Science University

Curated by ChEMBL
LigandPNGBDBM50053036(CHEMBL3318737)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of rat testis GST-tagged PARG catalytic activity after 30 mins using [32P]poly(ADP-ribose) by radioassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50142517(CHEMBL47885 | N-[4-(3,4,5-triihydroxy-benzoylamino...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibitory concentration against relaxation activity of DNA topoisomerase I by detecting the conversion of supercoiled pBR322 DNA to its relaxed formMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly(ADP-ribose) glycohydrolase(Rattus norvegicus)
Kumamoto Health Science University

Curated by ChEMBL
LigandPNGBDBM50052838(CHEMBL3318748)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of rat testis GST-tagged PARG catalytic activity after 30 mins using [32P]poly(ADP-ribose) by radioassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50142507(CHEMBL47526 | N-[3-(3,4,5-triihydroxy-benzoylamino...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibitory concentration against relaxation activity of DNA topoisomerase I by detecting the conversion of supercoiled pBR322 DNA to its relaxed formMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly(ADP-ribose) glycohydrolase(Rattus norvegicus)
Kumamoto Health Science University

Curated by ChEMBL
LigandPNGBDBM50053035(CHEMBL3318738)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of rat testis GST-tagged PARG catalytic activity after 30 mins using [32P]poly(ADP-ribose) by radioassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50142526(CHEMBL44765 | N-[4-(3,4-dihydroxy-benzoylamino)-ph...)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibitory concentration against relaxation activity of DNA topoisomerase I by detecting the conversion of supercoiled pBR322 DNA to its relaxed formMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly(ADP-ribose) glycohydrolase(Rattus norvegicus)
Kumamoto Health Science University

Curated by ChEMBL
LigandPNGBDBM50052839(CHEMBL3318747)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of rat testis GST-tagged PARG catalytic activity after 30 mins using [32P]poly(ADP-ribose) by radioassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly(ADP-ribose) glycohydrolase(Rattus norvegicus)
Kumamoto Health Science University

Curated by ChEMBL
LigandPNGBDBM50052831(CHEMBL3318754)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of rat testis GST-tagged PARG catalytic activity after 30 mins using [32P]poly(ADP-ribose) by radioassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50410165(CHEMBL372661)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibitory concentration against DNA topoisomerase I activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly(ADP-ribose) glycohydrolase(Rattus norvegicus)
Kumamoto Health Science University

Curated by ChEMBL
LigandPNGBDBM50052840(CHEMBL3318746)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of rat testis GST-tagged PARG catalytic activity after 30 mins using [32P]poly(ADP-ribose) by radioassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly(ADP-ribose) glycohydrolase(Rattus norvegicus)
Kumamoto Health Science University

Curated by ChEMBL
LigandPNGBDBM50052843(CHEMBL3318743)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of rat testis GST-tagged PARG catalytic activity after 30 mins using [32P]poly(ADP-ribose) by radioassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly(ADP-ribose) glycohydrolase(Rattus norvegicus)
Kumamoto Health Science University

Curated by ChEMBL
LigandPNGBDBM50052842(CHEMBL3318744)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of rat testis GST-tagged PARG catalytic activity after 30 mins using [32P]poly(ADP-ribose) by radioassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50410153(CHEMBL197216)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibitory concentration against DNA topoisomerase I activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50142529(Acetic acid 2,3-diacetoxy-5-[2-(3,4,5-triacetoxy-b...)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibitory concentration against relaxation activity of DNA topoisomerase I by detecting the conversion of supercoiled pBR322 DNA to its relaxed formMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50410158(CHEMBL195195)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibitory concentration against DNA topoisomerase I activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50142509(CHEMBL44441 | N-[2-(3,4-dihydroxy-benzoylamino)-ph...)
Affinity DataIC50:  6.40E+3nMAssay Description:Inhibitory concentration against relaxation activity of DNA topoisomerase I by detecting the conversion of supercoiled pBR322 DNA to its relaxed formMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50142528(CHEMBL296351 | N-Benzothiazol-2-yl-3,4,5-trihydrox...)
Affinity DataIC50:  8.20E+3nMAssay Description:Inhibitory concentration against relaxation activity of DNA topoisomerase I by detecting the conversion of supercoiled pBR322 DNA to its relaxed formMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly(ADP-ribose) glycohydrolase(Rattus norvegicus)
Kumamoto Health Science University

Curated by ChEMBL
LigandPNGBDBM50052835(CHEMBL3318751)
Affinity DataIC50:  8.20E+3nMAssay Description:Inhibition of rat testis GST-tagged PARG catalytic activity after 30 mins using [32P]poly(ADP-ribose) by radioassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50142514(Acetic acid 2,3-diacetoxy-5-[4-(3,4,5-triacetoxy-b...)
Affinity DataIC50:  8.60E+3nMAssay Description:Inhibitory concentration against relaxation activity of DNA topoisomerase I by detecting the conversion of supercoiled pBR322 DNA to its relaxed formMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly(ADP-ribose) glycohydrolase(Rattus norvegicus)
Kumamoto Health Science University

Curated by ChEMBL
LigandPNGBDBM50052836(CHEMBL3318750)
Affinity DataIC50:  9.80E+3nMAssay Description:Inhibition of rat testis GST-tagged PARG catalytic activity after 30 mins using [32P]poly(ADP-ribose) by radioassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly(ADP-ribose) glycohydrolase(Rattus norvegicus)
Kumamoto Health Science University

Curated by ChEMBL
LigandPNGBDBM50053034(CHEMBL3318739)
Affinity DataIC50:  9.90E+3nMAssay Description:Inhibition of rat testis GST-tagged PARG catalytic activity after 30 mins using [32P]poly(ADP-ribose) by radioassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50142523(CHEMBL297255 | N-[3-(3,4-dihydroxy-benzoylamino)-p...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory concentration against relaxation activity of DNA topoisomerase I by detecting the conversion of supercoiled pBR322 DNA to its relaxed formMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50142510(Acetic acid 2,3-diacetoxy-5-[3-(3,4,5-triacetoxy-b...)
Affinity DataIC50:  1.12E+4nMAssay Description:Inhibitory concentration against relaxation activity of DNA topoisomerase I by detecting the conversion of supercoiled pBR322 DNA to its relaxed formMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly(ADP-ribose) glycohydrolase(Rattus norvegicus)
Kumamoto Health Science University

Curated by ChEMBL
LigandPNGBDBM50052834(CHEMBL3317464)
Affinity DataIC50:  1.39E+4nMAssay Description:Inhibition of rat testis GST-tagged PARG catalytic activity after 30 mins using [32P]poly(ADP-ribose) by radioassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly(ADP-ribose) glycohydrolase(Rattus norvegicus)
Kumamoto Health Science University

Curated by ChEMBL
LigandPNGBDBM50053033(CHEMBL3318740)
Affinity DataIC50:  1.48E+4nMAssay Description:Inhibition of rat testis GST-tagged PARG catalytic activity after 30 mins using [32P]poly(ADP-ribose) by radioassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly(ADP-ribose) glycohydrolase(Rattus norvegicus)
Kumamoto Health Science University

Curated by ChEMBL
LigandPNGBDBM50052837(CHEMBL3318749)
Affinity DataIC50:  1.54E+4nMAssay Description:Inhibition of rat testis GST-tagged PARG catalytic activity after 30 mins using [32P]poly(ADP-ribose) by radioassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50142515(CHEMBL44747 | N-Benzothiazol-2-yl-3,4-dihydroxy-be...)
Affinity DataIC50:  1.69E+4nMAssay Description:Inhibitory concentration against relaxation activity of DNA topoisomerase I by detecting the conversion of supercoiled pBR322 DNA to its relaxed formMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly(ADP-ribose) glycohydrolase(Rattus norvegicus)
Kumamoto Health Science University

Curated by ChEMBL
LigandPNGBDBM50052841(CHEMBL3318745)
Affinity DataIC50:  1.88E+4nMAssay Description:Inhibition of rat testis GST-tagged PARG catalytic activity after 30 mins using [32P]poly(ADP-ribose) by radioassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly(ADP-ribose) glycohydrolase(Rattus norvegicus)
Kumamoto Health Science University

Curated by ChEMBL
LigandPNGBDBM50052844(CHEMBL3318742)
Affinity DataIC50:  1.92E+4nMAssay Description:Inhibition of rat testis GST-tagged PARG catalytic activity after 30 mins using [32P]poly(ADP-ribose) by radioassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly(ADP-ribose) glycohydrolase(Rattus norvegicus)
Kumamoto Health Science University

Curated by ChEMBL
LigandPNGBDBM50052833(CHEMBL3318752)
Affinity DataIC50:  2.74E+4nMAssay Description:Inhibition of rat testis GST-tagged PARG catalytic activity after 30 mins using [32P]poly(ADP-ribose) by radioassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50142525(CHEMBL47524 | N-(4,5-Dihydro-thiazol-2-yl)-3,4,5-t...)
Affinity DataIC50:  3.44E+4nMAssay Description:Inhibitory concentration against relaxation activity of DNA topoisomerase I by detecting the conversion of supercoiled pBR322 DNA to its relaxed formMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly(ADP-ribose) glycohydrolase(Rattus norvegicus)
Kumamoto Health Science University

Curated by ChEMBL
LigandPNGBDBM50053032(CHEMBL3318741)
Affinity DataIC50:  4.01E+4nMAssay Description:Inhibition of rat testis GST-tagged PARG catalytic activity after 30 mins using [32P]poly(ADP-ribose) by radioassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50142513(Acetic acid 2-acetoxy-5-[3-(3,4-diacetoxy-benzoyla...)
Affinity DataIC50:  4.32E+4nMAssay Description:Inhibitory concentration against relaxation activity of DNA topoisomerase I by detecting the conversion of supercoiled pBR322 DNA to its relaxed formMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50338992(CHEMBL1687978 | N-[5-(2-Furyl)-1,3,4-oxadiazol-2-y...)
Affinity DataIC50:  5.50E+4nMAssay Description:Inhibition of STAT3 transcriptional activity in human HeLa cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50338996(2-(4-Chlorophenyl)-N-(5-phenyl-1,3,4-oxadiazol-2-y...)
Affinity DataIC50:  6.10E+4nMAssay Description:Inhibition of STAT3 transcriptional activity in human HeLa cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50338994(CHEMBL1687976 | N-[5-(2-Furyl)-1,3,4-oxadiazol-2-y...)
Affinity DataIC50:  6.30E+4nMAssay Description:Inhibition of STAT3 transcriptional activity in human HeLa cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50410153(CHEMBL197216)
Affinity DataIC50:  6.30E+4nMAssay Description:Inhibitory concentration against DNA topoisomerase II activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50338995(2-Phenyl-N-(5-phenyl-1,3,4-oxadiazol-2-yl)-4-quino...)
Affinity DataIC50:  6.60E+4nMAssay Description:Inhibition of STAT3 transcriptional activity in human HeLa cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50338993(2-(2-Furyl)-N-[5-(2-furyl)-1,3,4-oxadiazol-2-yl]-4...)
Affinity DataIC50:  6.60E+4nMAssay Description:Inhibition of STAT3 transcriptional activity in human HeLa cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50338998(CHEMBL1687965 | N-[5-(3-Furyl)-1,3,4-oxadiazol-2-y...)
Affinity DataIC50:  7.20E+4nMAssay Description:Inhibition of STAT3 transcriptional activity in human HeLa cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50338991(CHEMBL1687979 | N-[5-(2-Furyl)-1,3,4-oxadiazol-2-y...)
Affinity DataIC50:  7.40E+4nMAssay Description:Inhibition of STAT3 transcriptional activity in human HeLa cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly(ADP-ribose) glycohydrolase(Rattus norvegicus)
Kumamoto Health Science University

Curated by ChEMBL
LigandPNGBDBM50053038(CHEMBL3318735)
Affinity DataIC50: >7.50E+4nMAssay Description:Inhibition of rat testis GST-tagged PARG catalytic activity after 30 mins using [32P]poly(ADP-ribose) by radioassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 93 total ) | Next | Last >>
Jump to: