Affinity DataKi: 1nMAssay Description:Binding affinity to human wild type adenosine A2B receptor expressed in Expi293F cells assessed as inhibition constant by surface plasmon resonance a...More data for this Ligand-Target Pair
Affinity DataKi: 76nMAssay Description:Binding affinity to human wild type adenosine A2A receptor expressed in Expi293F cells assessed as inhibition constant by surface plasmon resonance a...More data for this Ligand-Target Pair
Affinity DataKi: 150nMAssay Description:Binding affinity to human wild type adenosine A2A receptor expressed in Expi293F cells assessed as inhibition constant by surface plasmon resonance a...More data for this Ligand-Target Pair
Affinity DataKi: 290nMAssay Description:Binding affinity to human wild type adenosine A3 receptor expressed in Expi293F cells assessed as inhibition constant by surface plasmon resonance as...More data for this Ligand-Target Pair
Affinity DataKi: 395nMAssay Description:Binding affinity to human wild type adenosine A2A receptor expressed in Expi293F cells assessed as inhibition constant by surface plasmon resonance a...More data for this Ligand-Target Pair
Affinity DataKi: 1.30E+3nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluKK1(Q)1b receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.40E+3nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluKK1(Q)1b receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 3.00E+3nMAssay Description:Displacement of [3H]-(2S,4R)-4-methylglutamic acid from full length recombinant rat GluKK1(Q)1b receptor expressed in sf9 cells by liquid scintillati...More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKi: 4.70E+3nMAssay Description:Displacement of [3H]-(2S,4R)-4-methylglutamic acid from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation cou...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKi: 5.80E+3nMAssay Description:Mixed-type inhibition of electric eel acetylcholinesterase assessed as enzyme-inhibitor complex by Lineweaver-Burk plot methodMore data for this Ligand-Target Pair
Affinity DataKi: 6.30E+3nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluKK1(Q)1b receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKi: 1.12E+4nMAssay Description:Mixed-type inhibition of electric eel acetylcholinesterase assessed as enzyme-substrate-inhibitor complex by Lineweaver-Burk plot methodMore data for this Ligand-Target Pair
Affinity DataKi: 1.23E+4nMAssay Description:Displacement of [3H]-(2S,4R)-4-methylglutamic acid from full length recombinant rat GluKK1(Q)1b receptor expressed in sf9 cells by liquid scintillati...More data for this Ligand-Target Pair
Affinity DataKi: 1.33E+4nMAssay Description:Displacement of [3H]-(2S,4R)-4-methylglutamic acid from full length recombinant rat GluKK1(Q)1b receptor expressed in sf9 cells by liquid scintillati...More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKi: 1.44E+4nMAssay Description:Displacement of [3H]-(2S,4R)-4-methylglutamic acid from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation cou...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKi: 1.69E+4nMAssay Description:Mixed-type inhibition of electric eel acetylcholinesterase assessed as enzyme-substrate-inhibitor complex by Lineweaver-Burk plot methodMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKi: 1.70E+4nMAssay Description:Displacement of [3H]-(2S,4R)-4-methylglutamic acid from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation cou...More data for this Ligand-Target Pair
Affinity DataKi: 1.90E+4nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluKK1(Q)1b receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKi: 2.10E+4nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.40E+4nMAssay Description:Displacement of [3H]SYM2081 from full length recombinant rat GluKK1(Q)1b receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKi: 2.90E+4nMAssay Description:Displacement of [3H]SYM2081 from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 3.20E+4nMAssay Description:Displacement of [3H]SYM2081 from full length recombinant rat GluKK1(Q)1b receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKi: 3.40E+4nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKi: 4.00E+4nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 5.00E+4nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluKK1(Q)1b receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 5.00E+4nMAssay Description:Displacement of [3H]SYM2081 from full length recombinant rat GluKK1(Q)1b receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKi: 5.00E+4nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 5.00E+4nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluKK1(Q)1b receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKi: 5.00E+4nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKi: 5.00E+4nMAssay Description:Displacement of [3H]SYM2081 from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKi: 5.00E+4nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKi: 5.88E+4nMAssay Description:Mixed-type inhibition of electric eel acetylcholinesterase assessed as enzyme-substrate-inhibitor complex by Lineweaver-Burk plot methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKi: 8.31E+4nMAssay Description:Mixed-type inhibition of electric eel acetylcholinesterase assessed as enzyme-inhibitor complex by Lineweaver-Burk plot methodMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluKK1(Q)1b receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluKK1(Q)1b receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluKK1(Q)1b receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]SYM2081 from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluKK1(Q)1b receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 3(Rattus norvegicus)
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]SYM2081 from full length recombinant rat GluK3 receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]SYM2081 from full length recombinant rat GluKK1(Q)1b receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]KA from full length recombinant rat GluKK1(Q)1b receptor expressed in sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKi: 1.05E+5nMAssay Description:Mixed-type inhibition of electric eel acetylcholinesterase assessed as enzyme-inhibitor complex by Lineweaver-Burk plot methodMore data for this Ligand-Target Pair
Affinity DataKi: 2.70E+5nMAssay Description:Inhibition of jack bean alpha-mannosidase using p-nitrophenyl-mannopyranoside as substrate measured every 2 minsMore data for this Ligand-Target Pair
Affinity DataKi: 2.90E+5nMAssay Description:Mixed-type inhibition of jack bean alpha-mannosidase assessed as enzyme-substrate-inhibitor complex using o-orp-nitrophenyl-glycopyranoside as substr...More data for this Ligand-Target Pair
Affinity DataKi: 3.90E+5nMAssay Description:Mixed-type inhibition of jack bean alpha-mannosidase assessed as enzyme-inhibitor complex using o-orp-nitrophenyl-glycopyranoside as substrate by Lin...More data for this Ligand-Target Pair