Affinity DataIC50: 20nMAssay Description:The compounds II-2a to II-2m and controls in Table II were tested in 10-dose IC50 mode, with 3-fold serial dilution at a starting concentration of 10...More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:5 μl of enzyme (150 nM for ALDH1a1 and 200 nM for ALDH2 in reaction buffer) were delivered to assay wells in coming black, 384 well plate. 5 ...More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of ALDH1A1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:FAAH inhibition assay was performed using Fatty Acid Amide Hydrolase Inhibitor Screening Assay Kit (Item #10005196), Cayman (1180 E Ellsworth Rd Ann ...More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:5 μl of enzyme (150 nM for ALDH1a1 and 200 nM for ALDH2 in reaction buffer) were delivered to assay wells in coming black, 384 well plate. 5 ...More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of ALDH1A1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of ALDH1A1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:5 μl of enzyme (150 nM for ALDH1a1 and 200 nM for ALDH2 in reaction buffer) were delivered to assay wells in coming black, 384 well plate. 5 ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Centre D'Etudes Et De Recherche Sur Le MÉDicament De Normandie
Centre D'Etudes Et De Recherche Sur Le MÉDicament De Normandie
Affinity DataIC50: 60nMpH: 7.4Assay Description:Inhibitory ability of compounds on AChE activity was evaluated through the use of the spectrometic method of Ellman. Lyophilized electric eel AChE (...More data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibition of ALDH1A1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:5 μl of enzyme (150 nM for ALDH1a1 and 200 nM for ALDH2 in reaction buffer) were delivered to assay wells in coming black, 384 well plate. 5 ...More data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:5 μl of enzyme (150 nM for ALDH1a1 and 200 nM for ALDH2 in reaction buffer) were delivered to assay wells in coming black, 384 well plate. 5 ...More data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Inhibition of ALDH1A1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:5 μl of enzyme (150 nM for ALDH1a1 and 200 nM for ALDH2 in reaction buffer) were delivered to assay wells in coming black, 384 well plate. 5 ...More data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:5 μl of enzyme (150 nM for ALDH1a1 and 200 nM for ALDH2 in reaction buffer) were delivered to assay wells in coming black, 384 well plate. 5 ...More data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Inhibition of ALDH1A1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 210nMAssay Description:5 μl of enzyme (150 nM for ALDH1a1 and 200 nM for ALDH2 in reaction buffer) were delivered to assay wells in coming black, 384 well plate. 5 ...More data for this Ligand-Target Pair
Affinity DataIC50: 210nMAssay Description:Inhibition of ALDH1A1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 270nMAssay Description:Inhibition of ALDH1A1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 270nMAssay Description:5 μl of enzyme (150 nM for ALDH1a1 and 200 nM for ALDH2 in reaction buffer) were delivered to assay wells in coming black, 384 well plate. 5 ...More data for this Ligand-Target Pair
Affinity DataIC50: 310nMAssay Description:5 μl of enzyme (150 nM for ALDH1a1 and 200 nM for ALDH2 in reaction buffer) were delivered to assay wells in coming black, 384 well plate. 5 ...More data for this Ligand-Target Pair
Affinity DataIC50: 320nMAssay Description:5 μl of enzyme (150 nM for ALDH1a1 and 200 nM for ALDH2 in reaction buffer) were delivered to assay wells in coming black, 384 well plate. 5 ...More data for this Ligand-Target Pair
Affinity DataIC50: 320nMAssay Description:Inhibition of ALDH2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 390nMAssay Description:5 μl of enzyme (150 nM for ALDH1a1 and 200 nM for ALDH2 in reaction buffer) were delivered to assay wells in coming black, 384 well plate. 5 ...More data for this Ligand-Target Pair
Affinity DataIC50: 390nMAssay Description:5 μl of enzyme (150 nM for ALDH1a1 and 200 nM for ALDH2 in reaction buffer) were delivered to assay wells in coming black, 384 well plate. 5 ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Centre D'Etudes Et De Recherche Sur Le MÉDicament De Normandie
Centre D'Etudes Et De Recherche Sur Le MÉDicament De Normandie
Affinity DataIC50: 400nMpH: 7.4Assay Description:Inhibitory ability of compounds on AChE activity was evaluated through the use of the spectrometic method of Ellman. Lyophilized electric eel AChE (...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Centre D'Etudes Et De Recherche Sur Le MÉDicament De Normandie
Centre D'Etudes Et De Recherche Sur Le MÉDicament De Normandie
Affinity DataIC50: 400nMpH: 7.4Assay Description:Inhibitory ability of compounds on AChE activity was evaluated through the use of the spectrometic method of Ellman. Lyophilized electric eel AChE (...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Centre D'Etudes Et De Recherche Sur Le MÉDicament De Normandie
Centre D'Etudes Et De Recherche Sur Le MÉDicament De Normandie
Affinity DataIC50: 560nMpH: 7.4Assay Description:Inhibitory ability of compounds on AChE activity was evaluated through the use of the spectrometic method of Ellman. Lyophilized electric eel AChE (...More data for this Ligand-Target Pair
Affinity DataIC50: 580nMAssay Description:5 μl of enzyme (150 nM for ALDH1a1 and 200 nM for ALDH2 in reaction buffer) were delivered to assay wells in coming black, 384 well plate. 5 ...More data for this Ligand-Target Pair
Affinity DataIC50: 590nMAssay Description:5 μl of enzyme (150 nM for ALDH1a1 and 200 nM for ALDH2 in reaction buffer) were delivered to assay wells in coming black, 384 well plate. 5 ...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Centre D'Etudes Et De Recherche Sur Le MÉDicament De Normandie
Centre D'Etudes Et De Recherche Sur Le MÉDicament De Normandie
Affinity DataIC50: 630nMpH: 7.4Assay Description:Inhibitory ability of compounds on AChE activity was evaluated through the use of the spectrometic method of Ellman. Lyophilized electric eel AChE (...More data for this Ligand-Target Pair
Affinity DataIC50: 720nMAssay Description:The compounds II-2a to II-2m and controls in Table II were tested in 10-dose IC50 mode, with 3-fold serial dilution at a starting concentration of 10...More data for this Ligand-Target Pair
Affinity DataIC50: 850nMAssay Description:Inhibition of ALDH2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 850nMAssay Description:5 μl of enzyme (150 nM for ALDH1a1 and 200 nM for ALDH2 in reaction buffer) were delivered to assay wells in coming black, 384 well plate. 5 ...More data for this Ligand-Target Pair
Affinity DataIC50: 860nMAssay Description:5 μl of enzyme (150 nM for ALDH1a1 and 200 nM for ALDH2 in reaction buffer) were delivered to assay wells in coming black, 384 well plate. 5 ...More data for this Ligand-Target Pair
Affinity DataIC50: 870nMAssay Description:The compounds II-2a to II-2m and controls in Table II were tested in 10-dose IC50 mode, with 3-fold serial dilution at a starting concentration of 10...More data for this Ligand-Target Pair
Affinity DataIC50: 950nMAssay Description:The compounds II-2a to II-2m and controls in Table II were tested in 10-dose IC50 mode, with 3-fold serial dilution at a starting concentration of 10...More data for this Ligand-Target Pair
Affinity DataIC50: 1.43E+3nMAssay Description:5 μl of enzyme (150 nM for ALDH1a1 and 200 nM for ALDH2 in reaction buffer) were delivered to assay wells in coming black, 384 well plate. 5 ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.43E+3nMAssay Description:Inhibition of ALDH2 (unknown origin)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Centre D'Etudes Et De Recherche Sur Le MÉDicament De Normandie
Centre D'Etudes Et De Recherche Sur Le MÉDicament De Normandie
Affinity DataIC50: 1.50E+3nMpH: 7.4Assay Description:Inhibitory ability of compounds on AChE activity was evaluated through the use of the spectrometic method of Ellman. Lyophilized electric eel AChE (...More data for this Ligand-Target Pair
Affinity DataIC50: 1.51E+3nMAssay Description:5 μl of enzyme (150 nM for ALDH1a1 and 200 nM for ALDH2 in reaction buffer) were delivered to assay wells in coming black, 384 well plate. 5 ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.51E+3nMAssay Description:Inhibition of ALDH2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.89E+3nMAssay Description:The compounds II-2a to II-2m and controls in Table II were tested in 10-dose IC50 mode, with 3-fold serial dilution at a starting concentration of 10...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Centre D'Etudes Et De Recherche Sur Le MÉDicament De Normandie
Centre D'Etudes Et De Recherche Sur Le MÉDicament De Normandie
Affinity DataIC50: 2.30E+3nMpH: 7.4Assay Description:Inhibitory ability of compounds on AChE activity was evaluated through the use of the spectrometic method of Ellman. Lyophilized electric eel AChE (...More data for this Ligand-Target Pair
Affinity DataIC50: 2.54E+3nMAssay Description:5 μl of enzyme (150 nM for ALDH1a1 and 200 nM for ALDH2 in reaction buffer) were delivered to assay wells in coming black, 384 well plate. 5 ...More data for this Ligand-Target Pair
Affinity DataIC50: 2.54E+3nMAssay Description:Inhibition of ALDH1A1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.85E+3nMAssay Description:5 μl of enzyme (150 nM for ALDH1a1 and 200 nM for ALDH2 in reaction buffer) were delivered to assay wells in coming black, 384 well plate. 5 ...More data for this Ligand-Target Pair
Affinity DataIC50: 2.85E+3nMAssay Description:Inhibition of ALDH1A1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.95E+3nMAssay Description:Inhibition of ALDH1A1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.95E+3nMAssay Description:5 μl of enzyme (150 nM for ALDH1a1 and 200 nM for ALDH2 in reaction buffer) were delivered to assay wells in coming black, 384 well plate. 5 ...More data for this Ligand-Target Pair