Affinity DataKi: 0.0300nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human MT1 receptor transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
Affinity DataKi: 0.372nMAssay Description:Displacement of [3H]RAMHA from rat histamine H3 receptor in rat cerebral cortex membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.390nMAssay Description:Displacement of [3H]GR65630 from 5-HT3 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.398nMAssay Description:Displacement of [3H]GR65630 from 5-HT3 receptor (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of Perugia
Curated by ChEMBL
University Of Perugia
Curated by ChEMBL
Affinity DataKi: 0.400nMAssay Description:Inhibition of P38alpha MAPK (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.513nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in GPCR97 transfected human SK-N-MC cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.661nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in GPCR97 transfected human SK-N-MC cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human MT1 receptor transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
Affinity DataKi: 0.871nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in GPCR97 transfected human SK-N-MC cellsMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of Perugia
Curated by ChEMBL
University Of Perugia
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Inhibition of P38alpha MAPK (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.26nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in GPCR97 transfected human SK-N-MC cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.26nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in GPCR97 transfected human SK-N-MC cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.29nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in GPCR97 transfected human SK-N-MC cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Displacement of [3H]5-HT from human 5-HT7 receptor expressed in HEK293 cells after 30 mins by microbeta counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.41nMAssay Description:Displacement of [3H]RAMHA from rat histamine H3 receptor in rat cerebral cortex membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.48nMAssay Description:Displacement of [3H]RAMHA from rat histamine H3 receptor in rat cerebral cortex membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.48nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in GPCR97 transfected human SK-N-MC cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.55nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in GPCR97 transfected human SK-N-MC cellsMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 3-kinase regulatory subunit alpha/4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 1.58nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged PI3K p110delta/p85alpha expressed in baculovirus infected Sf9 insect cells using P...More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human MT1 receptor transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University Of Missouri
Curated by ChEMBL
University Of Missouri
Curated by ChEMBL
Affinity DataKi: 1.66nMAssay Description:Displacement of [3H](+)Pentazocine from sigma 1 receptor (unknown origin)More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University Of Missouri
Curated by ChEMBL
University Of Missouri
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:Displacement of [3H](+)Pentazocine from sigma 1 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.78nMAssay Description:Displacement of [3H]RAMHA from rat histamine H3 receptor in rat cerebral cortex membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in GPCR97 transfected human SK-N-MC cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.04nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in GPCR97 transfected human SK-N-MC cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.09nMAssay Description:Displacement of [3H]RAMHA from rat histamine H3 receptor in rat cerebral cortex membranesMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University Of Perugia
Curated by ChEMBL
University Of Perugia
Curated by ChEMBL
Affinity DataKi: 2.30nMAssay Description:Inhibition of P38alpha MAPK (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 2.34nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in GPCR97 transfected human SK-N-MC cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.45nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in GPCR97 transfected human SK-N-MC cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.45nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in GPCR97 transfected human SK-N-MC cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.57nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in GPCR97 transfected human SK-N-MC cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Displacement of [3H]5-HT from human 5-HT7 receptor expressed in HEK293 cells after 30 mins by microbeta counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 3.02nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in GPCR97 transfected human SK-N-MC cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Displacement of [3H]5-HT from human 5-HT7 receptor expressed in HEK293 cells after 30 mins by microbeta counting analysisMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 3-kinase regulatory subunit alpha/4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 3.16nMAssay Description:Inhibition of human recombinant full length N-terminal His6-tagged PI3K p110delta/p85alpha expressed in baculovirus infected Sf9 insect cells using P...More data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Displacement of [3H]N-Methylspiperone from dopamine D2 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 3.55nMAssay Description:Displacement of [3H]RAMHA from rat histamine H3 receptor in rat cerebral cortex membranesMore data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Displacement of [3H]N-Methylspiperone from dopamine D2 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 4.27nMAssay Description:Displacement of [3H]RAMHA from rat histamine H3 receptor in rat cerebral cortex membranesMore data for this Ligand-Target Pair
Affinity DataKi: 4.47nMAssay Description:Displacement of [3H]Pyrilamine from histamine H1 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 4.5nMAssay Description:Displacement of [3H]Pyrilamine from histamine H1 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 4.68nMAssay Description:Displacement of [3H]RAMHA from rat histamine H3 receptor in rat cerebral cortex membranesMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human MT1 receptor transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
Affinity DataKi: 5.30nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human MT1 receptor transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
Affinity DataKi: 5.62nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in GPCR97 transfected human SK-N-MC cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.70nMAssay Description:Displacement of [3H]Cimetidine from histamine H2 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 5.80nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human MT1 receptor transfected in CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
Affinity DataKi: 5.80nMAssay Description:Displacement of [3H]Cimetidine from histamine H2 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 6.60nMAssay Description:Displacement of [3H]5-HT from human 5-HT7 receptor expressed in HEK293 cells after 30 mins by microbeta counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 6.61nMAssay Description:Displacement of [3H]RAMHA from rat histamine H3 receptor in rat cerebral cortex membranesMore data for this Ligand-Target Pair