Affinity DataKi: 12.9nMAssay Description:Inhibition of Yes kinaseMore data for this Ligand-Target Pair
Affinity DataKi: 19.4nMAssay Description:Inhibition of Abl kinaseMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
Targegen
Curated by ChEMBL
Targegen
Curated by ChEMBL
Affinity DataKi: 2.09E+3nMAssay Description:Inhibition of PDGFRbetaMore data for this Ligand-Target Pair
Affinity DataKi: 6.70E+3nMAssay Description:Inhibitory activity against bovine adrenal phenylethanolamine N-methyltransferase(PNMT)More data for this Ligand-Target Pair
TargetAndrogen receptor(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:Displacement of [3H]DHT from androgen receptor in human MDA-MB-435 cells after 30 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Inhibition of VEGFR2More data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair