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Found 51 with Last Name = 'parmentier' and Initial = 'm'
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Upr Centre

Curated by PDSP Ki Database
LigandPNGBDBM50004051(2-Amino-4-phosphono-butyric acid | 2-Amino-4-phosp...)
Affinity DataKi:  400nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Upr Centre

Curated by PDSP Ki Database
LigandPNGBDBM50034504((1S,2S)-2-((S)-Amino-carboxy-methyl)-cyclopropanec...)
Affinity DataKi:  490nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Upr Centre

Curated by PDSP Ki Database
LigandPNGBDBM17664((2S)-2-amino-3-(phosphonooxy)propanoic acid | CHEM...)
Affinity DataKi:  2.30E+3nMMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Upr Centre

Curated by PDSP Ki Database
LigandPNGBDBM50034504((1S,2S)-2-((S)-Amino-carboxy-methyl)-cyclopropanec...)
Affinity DataKi:  8.90E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Upr Centre

Curated by PDSP Ki Database
LigandPNGBDBM50030628((S)-4C3HPG | 4-(Amino-carboxy-methyl)-2-hydroxy-be...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Upr Centre

Curated by PDSP Ki Database
LigandPNGBDBM50030629((R,S)-4-Carboxy-3-hydroxyphenylglycine | (S)-4CPG ...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Upr Centre

Curated by PDSP Ki Database
LigandPNGBDBM17657((2S)-2-aminopentanedioic acid | (S)-Glu | D-Glutam...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Upr Centre

Curated by PDSP Ki Database
LigandPNGBDBM82355(Amino-(3-hydroxy-isoxazol-5-yl)-acetic acid(Iboten...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Upr Centre

Curated by PDSP Ki Database
LigandPNGBDBM85016(CAS_1795545 | MAP4 | NSC_1795545)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Upr Centre

Curated by PDSP Ki Database
LigandPNGBDBM50062500((S)-2-((R)-1-Amino-1-carboxy-ethyl)-cyclopropaneca...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Upr Centre

Curated by PDSP Ki Database
LigandPNGBDBM50089910(2-Amino-2-(4-phosphono-phenyl)-propionic acid | 2-...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Upr Centre

Curated by PDSP Ki Database
LigandPNGBDBM85015(CAS_3964410 | MSPG | NSC_3964410)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Upr Centre

Curated by PDSP Ki Database
LigandPNGBDBM85014(CAS_5311456 | MTPG | NSC_5311456)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Upr Centre

Curated by PDSP Ki Database
LigandPNGBDBM17660((2S)-2-amino-3-(3,5-dioxo-1,2,4-oxadiazolidin-2-yl...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Upr Centre

Curated by PDSP Ki Database
LigandPNGBDBM50004863((+/-)-trans-ACPD | (1S,3S)-1-Amino-cyclopentane-1,...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Upr Centre

Curated by PDSP Ki Database
LigandPNGBDBM50004863((+/-)-trans-ACPD | (1S,3S)-1-Amino-cyclopentane-1,...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Upr Centre

Curated by PDSP Ki Database
LigandPNGBDBM85017((1S,3S)-1-AMINO-1-CARBOXYCYCLOPENTANE-3-ACETIC ACI...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Upr Centre

Curated by PDSP Ki Database
LigandPNGBDBM17657((2S)-2-aminopentanedioic acid | (S)-Glu | D-Glutam...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Upr Centre

Curated by PDSP Ki Database
LigandPNGBDBM82355(Amino-(3-hydroxy-isoxazol-5-yl)-acetic acid(Iboten...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Upr Centre

Curated by PDSP Ki Database
LigandPNGBDBM85017((1S,3S)-1-AMINO-1-CARBOXYCYCLOPENTANE-3-ACETIC ACI...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Upr Centre

Curated by PDSP Ki Database
LigandPNGBDBM50004863((+/-)-trans-ACPD | (1S,3S)-1-Amino-cyclopentane-1,...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Upr Centre

Curated by PDSP Ki Database
LigandPNGBDBM50004863((+/-)-trans-ACPD | (1S,3S)-1-Amino-cyclopentane-1,...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Upr Centre

Curated by PDSP Ki Database
LigandPNGBDBM50030627((+-)-MCPG | (R,S)-alpha-Methyl-4-carboxyphenylglyc...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Upr Centre

Curated by PDSP Ki Database
LigandPNGBDBM50004863((+/-)-trans-ACPD | (1S,3S)-1-Amino-cyclopentane-1,...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Upr Centre

Curated by PDSP Ki Database
LigandPNGBDBM17660((2S)-2-amino-3-(3,5-dioxo-1,2,4-oxadiazolidin-2-yl...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Upr Centre

Curated by PDSP Ki Database
LigandPNGBDBM85015(CAS_3964410 | MSPG | NSC_3964410)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Upr Centre

Curated by PDSP Ki Database
LigandPNGBDBM50089910(2-Amino-2-(4-phosphono-phenyl)-propionic acid | 2-...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Upr Centre

Curated by PDSP Ki Database
LigandPNGBDBM85016(CAS_1795545 | MAP4 | NSC_1795545)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50088301((E)-N,N-dimethyl-N-(4-(2-p-tolyl-6,7-dihydro-5H-be...)
Affinity DataIC50:  0.0300nMAssay Description:Displacement of [125I]MCP1 from CCR2/CXCR4 (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50035696(1,1''-{1,4-phenylenebis(methylene)}-bis{1,4,8,11-t...)
Affinity DataIC50:  0.0400nMAssay Description:Displacement of [125I]SDF1alpha from CCR2/CXCR4 (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50088301((E)-N,N-dimethyl-N-(4-(2-p-tolyl-6,7-dihydro-5H-be...)
Affinity DataIC50:  0.0800nMAssay Description:Displacement of [125I]SDF1alpha from CCR2/CXCR4 (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50035696(1,1''-{1,4-phenylenebis(methylene)}-bis{1,4,8,11-t...)
Affinity DataIC50:  0.0900nMAssay Description:Displacement of [125I]MCP1 from CCR2/CXCR4 (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50088301((E)-N,N-dimethyl-N-(4-(2-p-tolyl-6,7-dihydro-5H-be...)
Affinity DataIC50:  0.25nMAssay Description:Displacement of [125I]MCP1 from CCR2 (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50035696(1,1''-{1,4-phenylenebis(methylene)}-bis{1,4,8,11-t...)
Affinity DataIC50:  0.810nMAssay Description:Displacement of [125I]SDF1alpha from CXCR4 (unknown origin) expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Cnrs Umr 7175-Lc1

Curated by ChEMBL
LigandPNGBDBM50205734(1-(6-thiophen-2-yl-pyridazin-3-yl)-piperidine-4-ca...)
Affinity DataIC50:  5.80E+3nMAssay Description:Displacement of [125I]MIP1beta from CCR5 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Cnrs Umr 7175-Lc1

Curated by ChEMBL
LigandPNGBDBM50205735(CHEMBL219770 | N-(2-methyl-4-((4-methylpiperazin-1...)
Affinity DataIC50:  1.41E+4nMAssay Description:Displacement of [125I]MIP1beta from CCR5 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromal cell-derived factor 1(Homo sapiens (Human))
UniversitÉ

LigandPNGBDBM86004(Chalcone 2 | Chalcone, 3)
Affinity DataIC50:  1.50E+4nMT: 2°CAssay Description:Binding of chalcone 4 and chlcone 1 to CSCL12 was examined by monitoring changes in the emission intensity of intrinsic Trp fluorescence of the chemo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Cnrs Umr 7175-Lc1

Curated by ChEMBL
LigandPNGBDBM50205736(2-(4-benzyl-5-(2-(piperidin-1-yl)ethyl)-4H-1,2,4-t...)
Affinity DataIC50:  1.70E+4nMAssay Description:Displacement of [125I]MIP1beta from CCR5 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Cnrs Umr 7175-Lc1

Curated by ChEMBL
LigandPNGBDBM50205732(1-(3-diethylamino-propylamino)-3-methyl-2-(2-methy...)
Affinity DataIC50:  2.24E+4nMAssay Description:Displacement of [125I]MIP1beta from CCR5 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromal cell-derived factor 1(Homo sapiens (Human))
UniversitÉ

LigandPNGBDBM50042978((E)-1-(2-hydroxyphenyl)-3-(4-hydroxyphenyl)prop-2-...)
Affinity DataIC50:  2.42E+4nMT: 2°CAssay Description:Binding of chalcone 4 and chlcone 1 to CSCL12 was examined by monitoring changes in the emission intensity of intrinsic Trp fluorescence of the chemo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Cnrs Umr 7175-Lc1

Curated by ChEMBL
LigandPNGBDBM50205738(2-(4-oxo-3-(3-(piperidin-1-yl)propyl)-3,4-dihydroq...)
Affinity DataIC50:  4.90E+4nMAssay Description:Displacement of [125I]MIP1beta from CCR5 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Cnrs Umr 7175-Lc1

Curated by ChEMBL
LigandPNGBDBM50205737(1-((1-(4-fluorobenzyl)-1H-tetrazol-5-yl)(2-fluorop...)
Affinity DataIC50:  7.94E+4nMAssay Description:Displacement of [125I]MIP1beta from CCR5 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromal cell-derived factor 1(Homo sapiens (Human))
UniversitÉ

LigandPNGBDBM50042947(1-(4-Chloro-phenyl)-3-(4-hydroxy-3-methoxy-phenyl)...)
Affinity DataIC50:  1.50E+5nMT: 2°CAssay Description:Binding of chalcone 4 and chlcone 1 to CSCL12 was examined by monitoring changes in the emission intensity of intrinsic Trp fluorescence of the chemo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Cnrs Umr 7175-Lc1

Curated by ChEMBL
LigandPNGBDBM50205733(CHEMBL219769 | N-(1-benzylpiperidin-4-yl)-2-(5-met...)
Affinity DataIC50:  2.69E+5nMAssay Description:Displacement of [125I]MIP1beta from CCR5 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromal cell-derived factor 1(Homo sapiens (Human))
UniversitÉ

LigandPNGBDBM29143(CHEMBL7976 | Chalcone 1 | Chalcone, 13 | cid_63776...)
Affinity DataIC50: >5.00E+5nMT: 2°CAssay Description:Binding of chalcone 4 and chlcone 1 to CSCL12 was examined by monitoring changes in the emission intensity of intrinsic Trp fluorescence of the chemo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Cnrs Umr 7175-Lc1

Curated by ChEMBL
LigandPNGBDBM50205732(1-(3-diethylamino-propylamino)-3-methyl-2-(2-methy...)
Affinity DataEC50:  1.90E+3nMAssay Description:Agonist activity at CCR5 expressed in CHO-K1 cells in aqeuorin based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Cnrs Umr 7175-Lc1

Curated by ChEMBL
LigandPNGBDBM50205737(1-((1-(4-fluorobenzyl)-1H-tetrazol-5-yl)(2-fluorop...)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at CCR5 expressed in CHO-K1 cells in aqeuorin based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Cnrs Umr 7175-Lc1

Curated by ChEMBL
LigandPNGBDBM50205734(1-(6-thiophen-2-yl-pyridazin-3-yl)-piperidine-4-ca...)
Affinity DataEC50:  1.10E+3nMAssay Description:Agonist activity at CCR5 expressed in CHO-K1 cells in aqeuorin based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Cnrs Umr 7175-Lc1

Curated by ChEMBL
LigandPNGBDBM50205735(CHEMBL219770 | N-(2-methyl-4-((4-methylpiperazin-1...)
Affinity DataEC50:  2.00E+3nMAssay Description:Agonist activity at CCR5 expressed in CHO-K1 cells in aqeuorin based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Cnrs Umr 7175-Lc1

Curated by ChEMBL
LigandPNGBDBM50205736(2-(4-benzyl-5-(2-(piperidin-1-yl)ethyl)-4H-1,2,4-t...)
Affinity DataEC50:  3.00E+3nMAssay Description:Agonist activity at CCR5 expressed in CHO-K1 cells in aqeuorin based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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