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Found 69 with Last Name = 'parrino' and Initial = 'b'
TargetHistamine H4 receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50021529(CHEMBL3290578)
Affinity DataKi:  520nMAssay Description:Displacement of [3H]histamine from human H4R expressed in Sf9 cell membranes co-expressed with G protein Gai2 and Gb1gamma2 incubated for 60 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50021557(CHEMBL3290582)
Affinity DataKi:  2.36E+3nMAssay Description:Displacement of [3H]histamine from human H4R expressed in Sf9 cell membranes co-expressed with G protein Gai2 and Gb1gamma2 incubated for 60 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM189355(4-(4-Methylpiperazin-1-yl)-6-(pyridin-4-yl)-1,3,5-...)
Affinity DataKi:  3.19E+3nMAssay Description:Displacement of [3H]histamine from human H4R expressed in Sf9 cell membranes co-expressed with G protein Gai2 and Gb1gamma2 incubated for 60 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM189352(4-(4-Methylpiperazin-1-yl)-6-(naphthalen-1-ylmethy...)
Affinity DataKi:  5.60E+3nMAssay Description:Displacement of [3H]histamine from human H4R expressed in Sf9 cell membranes co-expressed with G protein Gai2 and Gb1gamma2 incubated for 60 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM189353(4-Benzyl-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-...)
Affinity DataKi:  7.50E+3nMAssay Description:Displacement of [3H]histamine from human H4R expressed in Sf9 cell membranes co-expressed with G protein Gai2 and Gb1gamma2 incubated for 60 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM189351(4-(4-Methylpiperazin-1-yl)-6-(2-methylpropyl)-1,3,...)
Affinity DataKi:  8.26E+3nMAssay Description:Displacement of [3H]histamine from human H4R expressed in Sf9 cell membranes co-expressed with G protein Gai2 and Gb1gamma2 incubated for 60 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM189354(4-((4-Chlorophenoxy)methyl)-6-(4-methylpiperazin-1...)
Affinity DataKi:  1.06E+4nMAssay Description:Displacement of [3H]histamine from human H4R expressed in Sf9 cell membranes co-expressed with G protein Gai2 and Gb1gamma2 incubated for 60 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM189350(3-((4-Amino-6-(4-methylpiperazin-1-yl)-1,3,5-triaz...)
Affinity DataKi:  1.46E+4nMAssay Description:Displacement of [3H]histamine from human H4R expressed in Sf9 cell membranes co-expressed with G protein Gai2 and Gb1gamma2 incubated for 60 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50315213(2-(difluoromethyl)-1-(4,6-dimorpholin-4-yl-1,3,5-t...)
Affinity DataIC50:  4.60nMAssay Description:Inhibition of PI3K p110gamma/p85alpha (unknown origin) assessed as reduction in PIP2 to PIP3 conversion by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM369714(US10233160, Compound 4 | US9981925, Compound 4)
Affinity DataIC50: <25nMAssay Description:Inhibition of N-terminal 6His-tagged human recombinant p70S6K T412E mutant (1 to 421 residues) in Sf21 insect cells using FITC-AHA-AKRRRLSSLRA-OH sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM369712(US10233160, Compound 2 | US9981925, Compound 2)
Affinity DataIC50: <25nMAssay Description:Inhibition of N-terminal 6His-tagged human recombinant p70S6K T412E mutant (1 to 421 residues) in Sf21 insect cells using FITC-AHA-AKRRRLSSLRA-OH sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin-conjugating enzyme E2 B(Homo sapiens)
Universit£

Curated by ChEMBL
LigandPNGBDBM50468268(CHEMBL3787660)
Affinity DataIC50:  25nMAssay Description:Inhibition of human recombinant Rad6B using ubiquitin and histone H2A and ubiquitin-activating enzyme E1 preincubated for 1 hr before ubiquitin and h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM369718(US10233160, Compound 8 | US9981925, Compound 8)
Affinity DataIC50:  25nMAssay Description:Inhibition of N-terminal 6His-tagged human recombinant p70S6K T412E mutant (1 to 421 residues) in Sf21 insect cells using FITC-AHA-AKRRRLSSLRA-OH sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM369720(US10233160, Compound 10 | US9981925, Compound 10)
Affinity DataIC50: <25nMAssay Description:Inhibition of N-terminal 6His-tagged human recombinant p70S6K T412E mutant (1 to 421 residues) in Sf21 insect cells using FITC-AHA-AKRRRLSSLRA-OH sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM369721(US10233160, Compound 11 | US9981925, Compound 11)
Affinity DataIC50:  25nMAssay Description:Inhibition of N-terminal 6His-tagged human recombinant p70S6K T412E mutant (1 to 421 residues) in Sf21 insect cells using FITC-AHA-AKRRRLSSLRA-OH sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM369725(US10233160, Compound 15 | US9981925, Compound 15)
Affinity DataIC50: <25nMAssay Description:Inhibition of N-terminal 6His-tagged human recombinant p70S6K T412E mutant (1 to 421 residues) in Sf21 insect cells using FITC-AHA-AKRRRLSSLRA-OH sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM369726(US10233160, Compound 16 | US9981925, Compound 16)
Affinity DataIC50: <25nMAssay Description:Inhibition of N-terminal 6His-tagged human recombinant p70S6K T412E mutant (1 to 421 residues) in Sf21 insect cells using FITC-AHA-AKRRRLSSLRA-OH sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM369728(US10233160, Compound 18 | US9981925, Compound 18)
Affinity DataIC50: <25nMAssay Description:Inhibition of N-terminal 6His-tagged human recombinant p70S6K T412E mutant (1 to 421 residues) in Sf21 insect cells using FITC-AHA-AKRRRLSSLRA-OH sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM369724(US10233160, Compound 14 | US9981925, Compound 14)
Affinity DataIC50: <25nMAssay Description:Inhibition of N-terminal 6His-tagged human recombinant p70S6K T412E mutant (1 to 421 residues) in Sf21 insect cells using FITC-AHA-AKRRRLSSLRA-OH sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM369723(US10233160, Compound 13 | US9981925, Compound 13)
Affinity DataIC50: <25nMAssay Description:Inhibition of N-terminal 6His-tagged human recombinant p70S6K T412E mutant (1 to 421 residues) in Sf21 insect cells using FITC-AHA-AKRRRLSSLRA-OH sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM369727(US10233160, Compound 17 | US9981925, Compound 17)
Affinity DataIC50:  25nMAssay Description:Inhibition of N-terminal 6His-tagged human recombinant p70S6K T412E mutant (1 to 421 residues) in Sf21 insect cells using FITC-AHA-AKRRRLSSLRA-OH sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM369722(US10233160, Compound 12 | US9981925, Compound 12)
Affinity DataIC50: <25nMAssay Description:Inhibition of N-terminal 6His-tagged human recombinant p70S6K T412E mutant (1 to 421 residues) in Sf21 insect cells using FITC-AHA-AKRRRLSSLRA-OH sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM27217((2R)-2-{[4-(benzylamino)-8-(propan-2-yl)pyrazolo[1...)
Affinity DataIC50:  43nMAssay Description:Inhibition of human recombinant CDK7/cyclin H using histone H1 and [gamma-33P]ATP incubated fro 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM27217((2R)-2-{[4-(benzylamino)-8-(propan-2-yl)pyrazolo[1...)
Affinity DataIC50:  43nMAssay Description:Inhibition of human recombinant CDK2/cyclinE using histone H1 and [gamma-33P]ATP incubated fro 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM27217((2R)-2-{[4-(benzylamino)-8-(propan-2-yl)pyrazolo[1...)
Affinity DataIC50:  43nMAssay Description:Inhibition of human recombinant CDK5/p25 using histone H1 and [gamma-33P]ATP incubated fro 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM27217((2R)-2-{[4-(benzylamino)-8-(propan-2-yl)pyrazolo[1...)
Affinity DataIC50:  43nMAssay Description:Inhibition of human recombinant CDK2/cyclin A using histone H1 and [gamma-33P]ATP incubated fro 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM27217((2R)-2-{[4-(benzylamino)-8-(propan-2-yl)pyrazolo[1...)
Affinity DataIC50:  43nMAssay Description:Inhibition of human recombinant CDK9/cyclin T expressed in insect cells using pRb fragment (773 to 928 amino acids) and [gamma-33P]ATP incubated fro ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM369668(US10233160, Compound 1 | US9981925, Compound 1)
Affinity DataIC50:  101nMAssay Description:Inhibition of N-terminal 6His-tagged human recombinant p70S6K T412E mutant (1 to 421 residues) in Sf21 insect cells using FITC-AHA-AKRRRLSSLRA-OH sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFucose-binding lectin PA-IIL(Pseudomonas aeruginosa)
Universit£

Curated by ChEMBL
LigandPNGBDBM50506709(CHEMBL3218456)
Affinity DataIC50:  140nMAssay Description:Inhibition of biotinylated polymeric fucose binding to Pseudomonas aeruginosa LecB expressed in Escherichia coli BL21(DE3) preincubated for 1 hr foll...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
University Of Palermo

Curated by ChEMBL
LigandPNGBDBM109086(US10793535, Cmpd ID 727 | US8604016, 670 | US99382...)
Affinity DataIC50:  310nMAssay Description:Inhibition of GLS-1 (unknown origin)More data for this Ligand-Target Pair
TargetFucose-binding lectin PA-IIL(Pseudomonas aeruginosa)
Universit£

Curated by ChEMBL
LigandPNGBDBM50505593(CHEMBL4453855)
Affinity DataIC50:  340nMAssay Description:Inhibition of N-(Fluorescein-5-yl)-N'-(alpha-L-fucopyranosyl ethylen)thiocarbamide binding to Pseudomonas aeruginosa PA14 LecB after 22 to 24 hrs by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeparanase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50462074(CHEMBL4251007)
Affinity DataIC50:  350nMAssay Description:Inhibition of activation of recombinant human pro-heparanase expressed in CHO cells by dimethylmethylene blue based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFucose-binding lectin PA-IIL(Pseudomonas aeruginosa)
Universit£

Curated by ChEMBL
LigandPNGBDBM50505613(CHEMBL4441817)
Affinity DataIC50:  440nMAssay Description:Inhibition of N-(Fluorescein-5-yl)-N'-(alpha-L-fucopyranosyl ethylen)thiocarbamide binding to Pseudomonas aeruginosa PA14 LecB after 22 to 24 hrs by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM369716(US10233160, Compound 6 | US9981925, Compound 6)
Affinity DataIC50:  501nMAssay Description:Inhibition of N-terminal 6His-tagged human recombinant p70S6K T412E mutant (1 to 421 residues) in Sf21 insect cells using FITC-AHA-AKRRRLSSLRA-OH sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM369719(US10233160, Compound 9 | US9981925, Compound 9)
Affinity DataIC50:  501nMAssay Description:Inhibition of N-terminal 6His-tagged human recombinant p70S6K T412E mutant (1 to 421 residues) in Sf21 insect cells using FITC-AHA-AKRRRLSSLRA-OH sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM27216((2R)-2-({6-[(3-chlorophenyl)amino]-9-(propan-2-yl)...)
Affinity DataIC50:  610nMAssay Description:Inhibition of recombinant human full length His-tagged CDK1/Cyclin B expressed in baculovirus expression system using peptide substrate after 30 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50441366(CHEMBL2435287)
Affinity DataIC50:  750nMAssay Description:Inhibition of human recombinant CDK1/cyclin B after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50237830(CHEMBL3799807)
Affinity DataIC50:  790nMAssay Description:Inhibition of N-terminal His-tagged human PAK4 kinase domain (300 to 591 residues) expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50441365(CHEMBL2435289)
Affinity DataIC50:  860nMAssay Description:Inhibition of human recombinant CDK1/cyclin B after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50441367(CHEMBL2435286)
Affinity DataIC50:  890nMAssay Description:Inhibition of human recombinant CDK1/cyclin B after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFucose-binding lectin PA-IIL(Pseudomonas aeruginosa)
Universit£

Curated by ChEMBL
LigandPNGBDBM50505593(CHEMBL4453855)
Affinity DataIC50:  970nMAssay Description:Inhibition of N-(Fluorescein-5-yl)-N'-(alpha-L-fucopyranosyl ethylen)thiocarbamide binding to Pseudomonas aeruginosa PAO1 LecB after 22 to 24 hrs by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50441365(CHEMBL2435289)
Affinity DataIC50:  970nMAssay Description:Inhibition of recombinant human full length His-tagged CDK1/cyclin B expressed in baculovirus expression system after 60 mins in presence of omnia pe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM369715(US10233160, Compound 5 | US9981925, Compound 5)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of N-terminal 6His-tagged human recombinant p70S6K T412E mutant (1 to 421 residues) in Sf21 insect cells using FITC-AHA-AKRRRLSSLRA-OH sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50462075(CHEMBL4239130)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of N-terminal 6His-tagged human recombinant p70S6K T412E mutant (1 to 421 residues) in Sf21 insect cells using FITC-AHA-AKRRRLSSLRA-OH sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM369713(US10233160, Compound 3 | US9981925, Compound 3)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of N-terminal 6His-tagged human recombinant p70S6K T412E mutant (1 to 421 residues) in Sf21 insect cells using FITC-AHA-AKRRRLSSLRA-OH sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50456470(CHEMBL4217475)
Affinity DataIC50:  1.14E+3nMAssay Description:Inhibition of recombinant human full length His-tagged CDK1/cyclin B expressed in baculovirus expression system after 60 mins in presence of omnia pe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFucose-binding lectin PA-IIL(Pseudomonas aeruginosa)
Universit£

Curated by ChEMBL
LigandPNGBDBM50505613(CHEMBL4441817)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of N-(Fluorescein-5-yl)-N'-(alpha-L-fucopyranosyl ethylen)thiocarbamide binding to Pseudomonas aeruginosa PAO1 LecB after 22 to 24 hrs by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50245850(CHEMBL4071003)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of Staphylococcus aureus 1199B NorA assessed as reduction in ethidium bromide efflux by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuinolone resistance protein NorA(Staphylococcus aureus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50017712((-)-reserpine | (3beta,16beta,17alpha,18beta,20alp...)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of Staphylococcus aureus 1199B NorA assessed as reduction in ethidium bromide efflux by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50462073(CHEMBL4241245)
Affinity DataIC50: <1.00E+4nMAssay Description:Inhibition of JAK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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