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Found 36 with Last Name = 'parrotta' and Initial = 'l'
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50310892(CHEMBL1078511 | N,N'-(9-(2-(1-methylpyrrolidin-2-y...)
Affinity DataIC50:  18nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50440391(CHEMBL2425367)
Affinity DataIC50:  28nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50134018(CHEMBL335819 | N,N'-(9-(4-aminophenylamino)acridin...)
Affinity DataIC50:  60nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50440389(CHEMBL1997011)
Affinity DataIC50:  100nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50440390(ISOMETAMIDIUM)
Affinity DataIC50:  100nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50440388(CHEMBL2425366)
Affinity DataIC50:  130nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50440387(CHEMBL2425365)
Affinity DataIC50:  220nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094895(1,4-diamino-9,10-anthraquinone | 1,4-diamino-anthr...)
Affinity DataIC50:  330nMAssay Description:Inhibition of CK1deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50176906(CHEMBL219728 | N'-(10H-indolo[3,2-b]quinolin-11-yl...)
Affinity DataIC50:  440nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50111322(CHEMBL274335 | N,N-Dimethyl-N'-(11-nitro-13H-5,13-...)
Affinity DataIC50:  500nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094893(1-Amino-4-hydroxy-anthraquinone | 1-hydroxy-4-amin...)
Affinity DataIC50:  660nMAssay Description:Inhibition of CK1deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50440386(CHEMBL2425364)
Affinity DataIC50:  750nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50008516(IC261)
Affinity DataIC50:  1.24E+3nMAssay Description:Inhibition of CK1alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50440385(CHEMBL2425363)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50068304(CHEMBL343445 | N-[9,10-Dioxo-6-(3-pyrrolidin-1-yl-...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50008516(IC261)
Affinity DataIC50:  2.57E+3nMAssay Description:Inhibition of CK1deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHomeodomain-interacting protein kinase 2(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094895(1,4-diamino-9,10-anthraquinone | 1,4-diamino-anthr...)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of HIPK2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094895(1,4-diamino-9,10-anthraquinone | 1,4-diamino-anthr...)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of DYRK1aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094893(1-Amino-4-hydroxy-anthraquinone | 1-hydroxy-4-amin...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of CK1alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094895(1,4-diamino-9,10-anthraquinone | 1,4-diamino-anthr...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of CK1alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50440384(CHEMBL2425362)
Affinity DataIC50:  5.40E+3nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412201(CRYPTOLEPINE HYDROCHLORIDE | Cryptolepine)
Affinity DataIC50:  9.40E+3nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50440382(CHEMBL2425361)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50440381(MERIDINE)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Fgr(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094895(1,4-diamino-9,10-anthraquinone | 1,4-diamino-anthr...)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibition of FgrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094895(1,4-diamino-9,10-anthraquinone | 1,4-diamino-anthr...)
Affinity DataIC50:  2.47E+4nMAssay Description:Inhibition of PIM1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform gamma-1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094893(1-Amino-4-hydroxy-anthraquinone | 1-hydroxy-4-amin...)
Affinity DataIC50:  2.62E+4nMAssay Description:Inhibition of CK1gamma1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform gamma-1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094895(1,4-diamino-9,10-anthraquinone | 1,4-diamino-anthr...)
Affinity DataIC50:  3.40E+4nMAssay Description:Inhibition of CK1gamma1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094895(1,4-diamino-9,10-anthraquinone | 1,4-diamino-anthr...)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of SykMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094895(1,4-diamino-9,10-anthraquinone | 1,4-diamino-anthr...)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of LynMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase CSK(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094895(1,4-diamino-9,10-anthraquinone | 1,4-diamino-anthr...)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of CSKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50240382(1,4-Dihydroxyanthrachinon | 1,4-dihydroxy-9,10-ant...)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of CK1alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform gamma-1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50240382(1,4-Dihydroxyanthrachinon | 1,4-dihydroxy-9,10-ant...)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of CK1gamma1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform delta(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50240382(1,4-Dihydroxyanthrachinon | 1,4-dihydroxy-9,10-ant...)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of CK1deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase I isoform gamma-1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50008516(IC261)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of CK1gamma1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50094895(1,4-diamino-9,10-anthraquinone | 1,4-diamino-anthr...)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of GST tagged ALKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed