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Found 745 with Last Name = 'pati' and Initial = 'b'
TargetD(4) dopamine receptor(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061349(CHEMBL129534 | [2-(3-Chloro-phenoxy)-ethyl]-(3-phe...)
Affinity DataKi:  0.309nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061345(CHEMBL129927 | [2-(3,4-Dimethyl-phenoxy)-ethyl]-(3...)
Affinity DataKi:  0.347nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061351((3-Phenoxy-propyl)-(2-m-tolyloxy-ethyl)-amine | CH...)
Affinity DataKi:  0.457nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061339(CHEMBL132884 | [2-(4-Chloro-phenoxy)-ethyl]-(3-phe...)
Affinity DataKi:  0.525nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061334(CHEMBL131997 | [2-(3-Chloro-4-methyl-phenoxy)-ethy...)
Affinity DataKi:  0.525nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061332((3-Phenoxy-propyl)-(2-p-tolyloxy-ethyl)-amine | CH...)
Affinity DataKi:  0.525nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061330(CHEMBL129757 | [2-(4-Chloro-phenoxy)-ethyl]-[3-(4-...)
Affinity DataKi:  0.832nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061325(CHEMBL131357 | [3-(4-Fluoro-phenoxy)-propyl]-(2-p-...)
Affinity DataKi:  0.955nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061324((2-p-Tolyloxy-ethyl)-(3-o-tolyloxy-propyl)-amine |...)
Affinity DataKi:  1.10nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50058234(CHEMBL300956 | N-[4-(2-Cyano-phenyl)-piperazin-1-y...)
Affinity DataKi:  1.20nMAssay Description:Binding affinity towards human dopamine receptor D4 expressed in CHO cells was determined by using [3H]thymidine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061327((2-p-Tolyloxy-ethyl)-(3-m-tolyloxy-propyl)-amine |...)
Affinity DataKi:  1.20nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061346((2-Phenoxy-ethyl)-(3-phenoxy-propyl)-amine | CHEMB...)
Affinity DataKi:  2nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061337((2-Phenoxy-ethyl)-(3-p-tolyloxy-propyl)-amine | CH...)
Affinity DataKi:  2.69nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061336(4-[2-(3-Phenoxy-propylamino)-ethoxy]-phenol | CHEM...)
Affinity DataKi:  3.09nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50058222(CHEMBL51023 | N-[4-(2-Methoxy-phenyl)-piperazin-1-...)
Affinity DataKi:  3.39nMAssay Description:Binding affinity towards human dopamine receptor D4 expressed in CHO cells was determined by using [3H]thymidine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50058223(4-Chloro-N-[4-(2-methoxy-phenyl)-piperazin-1-ylmet...)
Affinity DataKi:  3.47nMAssay Description:Binding affinity towards human dopamine receptor D4 expressed in CHO cells was determined by using [3H]thymidine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50058233(4-Chloro-N-[4-(2-cyano-phenyl)-piperazin-1-ylmethy...)
Affinity DataKi:  3.89nMAssay Description:Binding affinity towards human dopamine receptor D4 expressed in CHO cells was determined by using [3H]thymidine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061334(CHEMBL131997 | [2-(3-Chloro-4-methyl-phenoxy)-ethy...)
Affinity DataKi:  3.89nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D3 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061340(CHEMBL131396 | [2-(2-Chloro-phenoxy)-ethyl]-(3-phe...)
Affinity DataKi:  4.37nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061348(CHEMBL132455 | [2-(4-Nitro-phenoxy)-ethyl]-(3-phen...)
Affinity DataKi:  4.37nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50175151(3-(3-(bis(4-fluorophenyl)methoxy)-8-aza-bicyclo[3....)
Affinity DataKi:  5.01nMAssay Description:Ability of compound to inhibit dopamine uptake of receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50058230(4-Chloro-N-[4-(2-chloro-phenyl)-piperazin-1-ylmeth...)
Affinity DataKi:  5.25nMAssay Description:Binding affinity of compound towards human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50058226(3-Chloro-N-[4-(2-cyano-phenyl)-piperazin-1-ylmethy...)
Affinity DataKi:  5.25nMAssay Description:Binding affinity towards human dopamine receptor D4 expressed in CHO cells was determined by using [3H]thymidine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061343(CHEMBL128276 | [2-(4-Methoxy-phenoxy)-ethyl]-(3-ph...)
Affinity DataKi:  5.37nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50058233(4-Chloro-N-[4-(2-cyano-phenyl)-piperazin-1-ylmethy...)
Affinity DataKi:  5.5nMAssay Description:Binding affinity of compound towards human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061326(CHEMBL131484 | [2-(4-Chloro-phenoxy)-ethyl]-(3-p-t...)
Affinity DataKi:  5.62nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50058234(CHEMBL300956 | N-[4-(2-Cyano-phenyl)-piperazin-1-y...)
Affinity DataKi:  6.46nMAssay Description:Binding affinity of compound towards human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50148744(CHEMBL115253 | N-(2-{3-[Bis-(4-fluoro-phenyl)-meth...)
Affinity DataKi:  6.46nMAssay Description:Ability of compound to inhibit dopamine uptake of receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50058232(CHEMBL296506 | N-[4-(2-Methoxy-phenyl)-piperazin-1...)
Affinity DataKi:  6.76nMAssay Description:Binding affinity of compound towards human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50058222(CHEMBL51023 | N-[4-(2-Methoxy-phenyl)-piperazin-1-...)
Affinity DataKi:  7.76nMAssay Description:Binding affinity of compound towards human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-4(Homo sapiens (Human))
Depaul University

Curated by ChEMBL
LigandPNGBDBM50200547(CHEMBL3949842)
Affinity DataKi:  8nMAssay Description:Inhibition of human recombinant N-terminal His-tagged DTT-activated caspase-4 expressed in Escherichia coli using Ac-LEVD-AMC as substrate preincubat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50148741(Benzyl-(2-{3-[bis-(4-fluoro-phenyl)-methoxy]-8-aza...)
Affinity DataKi:  8.13nMAssay Description:Ability of compound to inhibit dopamine uptake of receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50058230(4-Chloro-N-[4-(2-chloro-phenyl)-piperazin-1-ylmeth...)
Affinity DataKi:  8.32nMAssay Description:Binding affinity towards human dopamine receptor D4 expressed in CHO cells was determined by using [3H]thymidine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50058225(CHEMBL45244 | N-((4-(2-cyanophenyl)piperazin-1-yl)...)
Affinity DataKi:  8.71nMAssay Description:Binding affinity of compound towards human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061344((2-p-Tolyloxy-ethyl)-(3-p-tolyloxy-propyl)-amine |...)
Affinity DataKi:  11.0nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50058220(CHEMBL51536 | N-[4-(2-Chloro-phenyl)-piperazin-1-y...)
Affinity DataKi:  12.0nMAssay Description:Binding affinity of compound towards human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50058232(CHEMBL296506 | N-[4-(2-Methoxy-phenyl)-piperazin-1...)
Affinity DataKi:  12.9nMAssay Description:Binding affinity towards human dopamine receptor D4 expressed in CHO cells was determined by using [3H]thymidine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM86701(3-(bis(4-fluorophenyl)methoxy)-8-methyl-8-aza-bicy...)
Affinity DataKi:  13.8nMAssay Description:Ability of compound to inhibit dopamine uptake of receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50058223(4-Chloro-N-[4-(2-methoxy-phenyl)-piperazin-1-ylmet...)
Affinity DataKi:  14.1nMAssay Description:Binding affinity of compound towards human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50148736(CHEMBL112528 | N-(2-{3-[Bis-(4-fluoro-phenyl)-meth...)
Affinity DataKi:  14.1nMAssay Description:Ability of compound to inhibit dopamine uptake of receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50058228(3-Chloro-N-[4-(2-methoxy-phenyl)-piperazin-1-ylmet...)
Affinity DataKi:  15.1nMAssay Description:Binding affinity of compound towards human dopamine receptor D4 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50058228(3-Chloro-N-[4-(2-methoxy-phenyl)-piperazin-1-ylmet...)
Affinity DataKi:  15.1nMAssay Description:Binding affinity towards human dopamine receptor D4 expressed in CHO cells was determined by using [3H]thymidine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50058224(CHEMBL298166 | N-[4-(2-Chloro-phenyl)-piperazin-1-...)
Affinity DataKi:  15.8nMAssay Description:Binding affinity towards human dopamine receptor D4 expressed in CHO cells was determined by using [3H]thymidine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-5(Homo sapiens (Human))
Depaul University

Curated by ChEMBL
LigandPNGBDBM50200547(CHEMBL3949842)
Affinity DataKi:  16nMAssay Description:Inhibition of human recombinant DTT-activated caspase-5 expressed in Escherichia coli using Ac-WEHD-AMC as substrate preincubated for 30 mins followe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-1(Homo sapiens (Human))
Depaul University

Curated by ChEMBL
LigandPNGBDBM50200547(CHEMBL3949842)
Affinity DataKi:  16nMAssay Description:Inhibition of human recombinant N-terminal His-tagged DTT-activated caspase-1 expressed in Escherichia coli using Ac-WEHD-AMC as substrate preincubat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061340(CHEMBL131396 | [2-(2-Chloro-phenoxy)-ethyl]-(3-phe...)
Affinity DataKi:  17.0nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D3 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50058225(CHEMBL45244 | N-((4-(2-cyanophenyl)piperazin-1-yl)...)
Affinity DataKi:  17.0nMAssay Description:Binding affinity towards human dopamine receptor D4 expressed in CHO cells was determined by using [3H]thymidine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50148742(3-[Bis-(4-fluoro-phenyl)-methoxy]-8-[2-(thiophen-2...)
Affinity DataKi:  18.6nMAssay Description:Ability of compound to inhibit dopamine uptake of receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061335((3-Phenoxy-propyl)-(2-o-tolyloxy-ethyl)-amine | CH...)
Affinity DataKi:  19.9nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D2 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Pomona College

Curated by ChEMBL
LigandPNGBDBM50061349(CHEMBL129534 | [2-(3-Chloro-phenoxy)-ethyl]-(3-phe...)
Affinity DataKi:  21.9nMAssay Description:Binding affinity to displace [3H]spiperone from cloned human dopamine receptor D2 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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