Affinity DataKi: 0.540nMAssay Description:Binding affinity to full length human His-MBP-TNNI3K assessed as off-rate constant in presence of rhodamine green labeled GW805818X by fluorescence c...More data for this Ligand-Target Pair
TargetGalanin receptor type 1(Homo sapiens (Human))
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataKi: 13nMAssay Description:Binding affinity to full length mouse His-MBP-TNNI3K assessed as off-rate constant in presence of rhodamine green labeled GW805818X by fluorescence c...More data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Scripps Research Institute
Curated by ChEMBL
Scripps Research Institute
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Inhibitory concentration of the compound against Fatty-acid amide hydrolase (FAAH) in rat liverMore data for this Ligand-Target Pair
TargetGalanin receptor type 1(Homo sapiens (Human))
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Dupont Pharmaceuticals
Curated by PDSP Ki Database
TargetGalanin receptor type 1(Homo sapiens (Human))
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Dupont Pharmaceuticals
Curated by PDSP Ki Database
TargetGalanin receptor type 1(Homo sapiens (Human))
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Dupont Pharmaceuticals
Curated by PDSP Ki Database
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Scripps Research Institute
Curated by ChEMBL
Scripps Research Institute
Curated by ChEMBL
Affinity DataKi: 82nMAssay Description:Inhibitory concentration of the compound against Fatty-acid amide hydrolase (FAAH) in rat liverMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Scripps Research Institute
Curated by ChEMBL
Scripps Research Institute
Curated by ChEMBL
Affinity DataKi: 96nMAssay Description:Inhibitory constant of the compound against Fatty-acid amide hydrolase (FAAH) in rat liverMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Dupont Pharmaceuticals
Curated by PDSP Ki Database
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Scripps Research Institute
Curated by ChEMBL
Scripps Research Institute
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:Inhibitory constant of the compound against Fatty-acid amide hydrolase (FAAH) in rat liverMore data for this Ligand-Target Pair
TargetGalanin receptor type 1(Homo sapiens (Human))
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Dupont Pharmaceuticals
Curated by PDSP Ki Database
TargetGalanin receptor type 1(Homo sapiens (Human))
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Dupont Pharmaceuticals
Curated by PDSP Ki Database
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Scripps Research Institute
Curated by ChEMBL
Scripps Research Institute
Curated by ChEMBL
Affinity DataKi: 130nMAssay Description:Inhibitory constant of the compound against Fatty-acid amide hydrolase (FAAH) in rat liverMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Scripps Research Institute
Curated by ChEMBL
Scripps Research Institute
Curated by ChEMBL
Affinity DataKi: 140nMAssay Description:Inhibitory constant of the compound against Fatty-acid amide hydrolase (FAAH) in rat liverMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Scripps Research Institute
Curated by ChEMBL
Scripps Research Institute
Curated by ChEMBL
Affinity DataKi: 140nMAssay Description:Inhibitory constant of the compound against Fatty-acid amide hydrolase (FAAH) in rat liverMore data for this Ligand-Target Pair
TargetGalanin receptor type 1(Homo sapiens (Human))
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Dupont Pharmaceuticals
Curated by PDSP Ki Database
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Scripps Research Institute
Curated by ChEMBL
Scripps Research Institute
Curated by ChEMBL
Affinity DataKi: 170nMAssay Description:Inhibitory concentration of the compound against Fatty-acid amide hydrolase (FAAH) in rat liverMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Scripps Research Institute
Curated by ChEMBL
Scripps Research Institute
Curated by ChEMBL
Affinity DataKi: 170nMAssay Description:Inhibitory constant of the compound against Fatty-acid amide hydrolase (FAAH) in rat liverMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Dupont Pharmaceuticals
Curated by PDSP Ki Database
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Institute For Chemical Biology
Curated by ChEMBL
Institute For Chemical Biology
Curated by ChEMBL
Affinity DataKi: 190nMpH: 9.0Assay Description:Compound was tested for inhibitory potency against Fatty-acid amide hydrolase (FAAH) at pH 9.0More data for this Ligand-Target Pair
TargetGalanin receptor type 1(Homo sapiens (Human))
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Dupont Pharmaceuticals
Curated by PDSP Ki Database
TargetGalanin receptor type 1(Homo sapiens (Human))
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Dupont Pharmaceuticals
Curated by PDSP Ki Database
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Scripps Research Institute
Curated by ChEMBL
Scripps Research Institute
Curated by ChEMBL
Affinity DataKi: 240nMAssay Description:Inhibitory constant of the compound against Fatty-acid amide hydrolase (FAAH) in rat liverMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Institute For Chemical Biology
Curated by ChEMBL
Institute For Chemical Biology
Curated by ChEMBL
Affinity DataKi: 250nMpH: 9.0Assay Description:Compound was tested for inhibitory potency against Fatty-acid amide hydrolase (FAAH) at pH 9.0More data for this Ligand-Target Pair
TargetGalanin receptor type 1(Homo sapiens (Human))
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Dupont Pharmaceuticals
Curated by PDSP Ki Database
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Scripps Research Institute
Curated by ChEMBL
Scripps Research Institute
Curated by ChEMBL
Affinity DataKi: 320nMAssay Description:Inhibitory constant of the compound against Fatty-acid amide hydrolase (FAAH) in rat liverMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Institute For Chemical Biology
Curated by ChEMBL
Institute For Chemical Biology
Curated by ChEMBL
Affinity DataKi: 390nMpH: 9.0Assay Description:Compound was tested for inhibitory potency against Fatty-acid amide hydrolase (FAAH) at pH 9.0More data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Scripps Research Institute
Curated by ChEMBL
Scripps Research Institute
Curated by ChEMBL
Affinity DataKi: 440nMAssay Description:Inhibitory concentration of the compound against Fatty-acid amide hydrolase (FAAH) in rat liverMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Scripps Research Institute
Curated by ChEMBL
Scripps Research Institute
Curated by ChEMBL
Affinity DataKi: 490nMAssay Description:Inhibitory concentration of the compound against Fatty-acid amide hydrolase (FAAH) in rat liverMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Institute For Chemical Biology
Curated by ChEMBL
Institute For Chemical Biology
Curated by ChEMBL
Affinity DataKi: 550nMpH: 9.0Assay Description:Inhibitory concentration against Fatty-acid amide hydrolase (FAAH) at pH 9.0More data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Scripps Research Institute
Curated by ChEMBL
Scripps Research Institute
Curated by ChEMBL
Affinity DataKi: 570nMAssay Description:Inhibitory constant of the compound against Fatty-acid amide hydrolase (FAAH) in rat liverMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Dupont Pharmaceuticals
Curated by PDSP Ki Database
TargetGalanin receptor type 1(Homo sapiens (Human))
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Dupont Pharmaceuticals
Curated by PDSP Ki Database
TargetGalanin receptor type 1(Homo sapiens (Human))
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Dupont Pharmaceuticals
Curated by PDSP Ki Database
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Scripps Research Institute
Curated by ChEMBL
Scripps Research Institute
Curated by ChEMBL
Affinity DataKi: 780nMAssay Description:Inhibitory constant of the compound against Fatty-acid amide hydrolase (FAAH) in rat liverMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Institute For Chemical Biology
Curated by ChEMBL
Institute For Chemical Biology
Curated by ChEMBL
Affinity DataKi: 800nMpH: 9.0Assay Description:Concentration of the compound required to inhibit fatty acid amide hydrolase (FAAH) at pH 7.0More data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Institute For Chemical Biology
Curated by ChEMBL
Institute For Chemical Biology
Curated by ChEMBL
Affinity DataKi: 1.10E+3nMpH: 9.0Assay Description:Concentration of the compound required to inhibit Fatty-acid amide hydrolase (FAAH) at pH 7.0More data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Institute For Chemical Biology
Curated by ChEMBL
Institute For Chemical Biology
Curated by ChEMBL
Affinity DataKi: 1.10E+3nMpH: 9.0Assay Description:Concentration of the compound required to inhibit fatty acid amide hydrolase (FAAH) at pH 7.0More data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Scripps Research Institute
Curated by ChEMBL
Scripps Research Institute
Curated by ChEMBL
Affinity DataKi: 1.20E+3nMAssay Description:Inhibitory constant of the compound against Fatty-acid amide hydrolase (FAAH) in rat liverMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Scripps Research Institute
Curated by ChEMBL
Scripps Research Institute
Curated by ChEMBL
Affinity DataKi: 1.20E+3nMAssay Description:Inhibitory constant of the compound against Fatty-acid amide hydrolase (FAAH) in rat liverMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Dupont Pharmaceuticals
Curated by PDSP Ki Database
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Scripps Research Institute
Curated by ChEMBL
Scripps Research Institute
Curated by ChEMBL
Affinity DataKi: 2.80E+3nMAssay Description:Inhibitory constant of the compound against Fatty-acid amide hydrolase (FAAH) in rat liverMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Dupont Pharmaceuticals
Curated by PDSP Ki Database