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Found 2255 with Last Name = 'patterson' and Initial = 'j'
TargetSerine/threonine-protein kinase TNNI3K(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50578225(CHEMBL4869303)
Affinity DataKi:  0.540nMAssay Description:Binding affinity to full length human His-MBP-TNNI3K assessed as off-rate constant in presence of rhodamine green labeled GW805818X by fluorescence c...More data for this Ligand-Target Pair
TargetGalanin receptor type 1(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM50273370(CHEMBL503473 | GWTLNSAGYLLGPPPGFSPFR-CONH2 | Galan...)
Affinity DataKi:  11.5nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase TNNI3K(Mus musculus)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50578225(CHEMBL4869303)
Affinity DataKi:  13nMAssay Description:Binding affinity to full length mouse His-MBP-TNNI3K assessed as off-rate constant in presence of rhodamine green labeled GW805818X by fluorescence c...More data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50073987(1,1,1-Trifluoro-9-phenyl-nonan-2-one | 1,1,1-trifl...)
Affinity DataKi:  25nMAssay Description:Inhibitory concentration of the compound against Fatty-acid amide hydrolase (FAAH) in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM85070(Galanin, Porcine)
Affinity DataKi:  25.2nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM85530(Nor-d-fenfluramine | Nor-dexfenfluramine | Norfenf...)
Affinity DataKi:  27nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM50273369(CHEMBL526003 | GWTLNSAGYLLGPQQFFGLM-CONH2 | Galani...)
Affinity DataKi:  27.4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM85072(Galanin, Human)
Affinity DataKi:  30.9nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM85530(Nor-d-fenfluramine | Nor-dexfenfluramine | Norfenf...)
Affinity DataKi:  56nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM85598(l-norfenfluramine)
Affinity DataKi:  65nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50069273((Z)-1,1,1-Trifluoro-nonadec-10-en-2-one | 1,1,1-tr...)
Affinity DataKi:  82nMAssay Description:Inhibitory concentration of the compound against Fatty-acid amide hydrolase (FAAH) in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50073986(1,1,1-Trifluoro-8-(4-heptyl-phenyl)-octan-2-one | ...)
Affinity DataKi:  96nMAssay Description:Inhibitory constant of the compound against Fatty-acid amide hydrolase (FAAH) in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM85598(l-norfenfluramine)
Affinity DataKi:  99nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50073974(1,1,1-Trifluoro-8-phenyl-octan-2-one | 1,1,1-Trifl...)
Affinity DataKi:  100nMAssay Description:Inhibitory constant of the compound against Fatty-acid amide hydrolase (FAAH) in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM85205(Galanin (1-16) | Galanin (1-16), rat)
Affinity DataKi:  106nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM50307254(CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2 | M40)
Affinity DataKi:  109nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50073985(1,1,1-Trifluoro-undecan-2-one | 1,1,1-trifluoround...)
Affinity DataKi:  130nMAssay Description:Inhibitory constant of the compound against Fatty-acid amide hydrolase (FAAH) in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50073975(1,1,1-Trifluoro-tridecan-2-one | 1,1,1-trifluorotr...)
Affinity DataKi:  140nMAssay Description:Inhibitory constant of the compound against Fatty-acid amide hydrolase (FAAH) in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50073984(1,1,1-Trifluoro-8-(3-hexyl-phenyl)-octan-2-one | C...)
Affinity DataKi:  140nMAssay Description:Inhibitory constant of the compound against Fatty-acid amide hydrolase (FAAH) in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM50273370(CHEMBL503473 | GWTLNSAGYLLGPPPGFSPFR-CONH2 | Galan...)
Affinity DataKi:  170nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50073989(1,1,1-Trifluoro-7-phenyl-heptan-2-one | 1,1,1-Trif...)
Affinity DataKi:  170nMAssay Description:Inhibitory concentration of the compound against Fatty-acid amide hydrolase (FAAH) in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50073973((E)-1,1,1-Trifluoro-nonadec-10-en-2-one | 1,1,1-Tr...)
Affinity DataKi:  170nMAssay Description:Inhibitory constant of the compound against Fatty-acid amide hydrolase (FAAH) in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM85530(Nor-d-fenfluramine | Nor-dexfenfluramine | Norfenf...)
Affinity DataKi:  187nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Institute For Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50069276(4-Bromo-3-oxo-butyric acid (Z)-tetradec-5-enyl est...)
Affinity DataKi:  190nMpH: 9.0Assay Description:Compound was tested for inhibitory potency against Fatty-acid amide hydrolase (FAAH) at pH 9.0More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM85070(Galanin, Porcine)
Affinity DataKi:  227nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM85072(Galanin, Human)
Affinity DataKi:  232nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50073981(1,1,1-Trifluoro-nonadecan-2-one | 1,1,1-trifluoron...)
Affinity DataKi:  240nMAssay Description:Inhibitory constant of the compound against Fatty-acid amide hydrolase (FAAH) in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Institute For Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50069273((Z)-1,1,1-Trifluoro-nonadec-10-en-2-one | 1,1,1-tr...)
Affinity DataKi:  250nMpH: 9.0Assay Description:Compound was tested for inhibitory potency against Fatty-acid amide hydrolase (FAAH) at pH 9.0More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM50273369(CHEMBL526003 | GWTLNSAGYLLGPQQFFGLM-CONH2 | Galani...)
Affinity DataKi:  256nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM85598(l-norfenfluramine)
Affinity DataKi:  267nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50073982(1,1,1-Trifluoro-9-(2-octyl-phenyl)-nonan-2-one | C...)
Affinity DataKi:  320nMAssay Description:Inhibitory constant of the compound against Fatty-acid amide hydrolase (FAAH) in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Institute For Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50069272((Z)-1-Bromo-nonadec-10-en-2-one | CHEMBL157736)
Affinity DataKi:  390nMpH: 9.0Assay Description:Compound was tested for inhibitory potency against Fatty-acid amide hydrolase (FAAH) at pH 9.0More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50073980(5-((1R,6R)-6-Butoxymethyl-cyclohex-3-enylmethoxy)-...)
Affinity DataKi:  440nMAssay Description:Inhibitory concentration of the compound against Fatty-acid amide hydrolase (FAAH) in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50073970(1,1,1-Trifluoro-pentadecan-2-one | 1,1,1-trifluoro...)
Affinity DataKi:  490nMAssay Description:Inhibitory concentration of the compound against Fatty-acid amide hydrolase (FAAH) in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Institute For Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50069270(4-Bromo-3-oxo-butyric acid heptyl ester | CHEMBL15...)
Affinity DataKi:  550nMpH: 9.0Assay Description:Inhibitory concentration against Fatty-acid amide hydrolase (FAAH) at pH 9.0More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50073978(5-((1R,6S)-6-Butoxymethyl-cyclohex-3-enylmethoxy)-...)
Affinity DataKi:  570nMAssay Description:Inhibitory constant of the compound against Fatty-acid amide hydrolase (FAAH) in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM85597(CAS_37577-24-5 | NSC_65801 | l-Fenfluramine)
Affinity DataKi:  680nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM85068(Gal(1-13)-Std I)
Affinity DataKi:  685nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM50307254(CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2 | M40)
Affinity DataKi:  713nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50073990(5-((1R,2S)-2-Butoxymethyl-cyclohexylmethoxy)-1,1,1...)
Affinity DataKi:  780nMAssay Description:Inhibitory constant of the compound against Fatty-acid amide hydrolase (FAAH) in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Institute For Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50069269((R)-octan-2-yl 4-bromo-3-oxobutanoate | 4-Bromo-3-...)
Affinity DataKi:  800nMpH: 9.0Assay Description:Concentration of the compound required to inhibit fatty acid amide hydrolase (FAAH) at pH 7.0More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Institute For Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50069271(4-Chloro-3-oxo-butyric acid (R)-1-methyl-heptyl es...)
Affinity DataKi:  1.10E+3nMpH: 9.0Assay Description:Concentration of the compound required to inhibit Fatty-acid amide hydrolase (FAAH) at pH 7.0More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Institute For Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50069280(4-Bromo-3-oxo-butyric acid (S)-1-methyl-heptyl est...)
Affinity DataKi:  1.10E+3nMpH: 9.0Assay Description:Concentration of the compound required to inhibit fatty acid amide hydrolase (FAAH) at pH 7.0More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50073971(5-((1R,2R)-2-Butoxymethyl-cyclohexylmethoxy)-1,1,1...)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibitory constant of the compound against Fatty-acid amide hydrolase (FAAH) in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50073977(1,1,1-Trifluoro-nonan-2-one | 1,1,1-trifluorononan...)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibitory constant of the compound against Fatty-acid amide hydrolase (FAAH) in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM85597(CAS_37577-24-5 | NSC_65801 | l-Fenfluramine)
Affinity DataKi:  1.43E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM85597(CAS_37577-24-5 | NSC_65801 | l-Fenfluramine)
Affinity DataKi:  1.62E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM85596(CAS_3239-45-0 | NSC_65801 | d-Fenfluramine)
Affinity DataKi:  2.08E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50073979(1,1,1-Trifluoro-7-(2-hexyl-phenyl)-heptan-2-one | ...)
Affinity DataKi:  2.80E+3nMAssay Description:Inhibitory constant of the compound against Fatty-acid amide hydrolase (FAAH) in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM85596(CAS_3239-45-0 | NSC_65801 | d-Fenfluramine)
Affinity DataKi:  3.92E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
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