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Found 82 with Last Name = 'peeters' and Initial = 'l'
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85994([leu13]pMOT(1-19))
Affinity DataKi:  0.980nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85614([Leu13]motilin | [leu13]pMOT(1-22))
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85979([ala3,leu13]pMOT(1-14))
Affinity DataKi:  1.32nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85987([leu13]pMOT(1-16))
Affinity DataKi:  2.14nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85389(CAS_52906-92-0 | Motilin)
Affinity DataKi:  2.82nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85981([ala1,leu13]pMOT(1-14) | [leu13]pMOT(1-14))
Affinity DataKi:  3.16nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50503158(CHEMBL4589377)
Affinity DataKi:  4.20nMAssay Description:Displacement of [3H]JNJ-46281222 from human mGlu2 receptor expressed in CHOK1 cell membranes preincubated for 3 hrs followed by [3H]JNJ-46281222 addi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85986([ala11,leu13]pMOT(1-14))
Affinity DataKi:  4.57nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85992([ala10,leu13]pMOT(1-14))
Affinity DataKi:  5.01nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50503158(CHEMBL4589377)
Affinity DataKi:  5.80nMAssay Description:Displacement of [3H]JNJ-46281222 from human mGlu2 receptor expressed in CHOK1 cell membranes after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85989(N-ethyl, N-methyl Erythromycin-A enol ether)
Affinity DataKi:  6.03nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50503157(CHEMBL4538850)
Affinity DataKi:  6.20nMAssay Description:Displacement of [3H]JNJ-46281222 from human mGlu2 receptor expressed in CHOK1 cell membranes preincubated for 3 hrs followed by [3H]JNJ-46281222 addi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85980([ala12,leu13]pMOT(1-14))
Affinity DataKi:  6.31nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85999([ala14,leu13]pMOT(1-14))
Affinity DataKi:  7.08nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85990([ala13,leu13]pMOT(1-14))
Affinity DataKi:  7.24nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85993(Erythromycin-B enol ether)
Affinity DataKi:  7.59nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50194613(CHEMBL3947764)
Affinity DataKi:  7.60nMAssay Description:Displacement of [3H]JNJ-46281222 from human mGlu2 receptor expressed in CHOK1 cell membranes after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50194613(CHEMBL3947764)
Affinity DataKi:  7.60nMAssay Description:Displacement of [3H]JNJ-46281222 from human mGlu2 receptor expressed in CHOK1 cell membranes preincubated for 3 hrs followed by [3H]JNJ-46281222 addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85846(CAS_33396-29-1 | EM523 | Erythromycin A 6,9-enolet...)
Affinity DataKi:  8.32nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50399088(CHEMBL2179319)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]8-Trifluoromethyl-3-cyclopropylmethyl-7-[(4-phenyl-1-piperidinyl)methyl]-1,2,4-triazolo[4,3-a]pyridine from mGlu2 receptor (unkno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85984([ala5,leu13]pMOT(1-14))
Affinity DataKi:  28.8nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85983([ala8,leu13]pMOT(1-14))
Affinity DataKi:  36.3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85978([ala6,leu13]pMOT(1-14))
Affinity DataKi:  46.8nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM86685(ABT-229)
Affinity DataKi:  58.9nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50503157(CHEMBL4538850)
Affinity DataKi:  62nMAssay Description:Displacement of [3H]JNJ-46281222 from human mGlu2 receptor expressed in CHOK1 cell membranes after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85991([ala9,leu13]pMOT(1-14))
Affinity DataKi:  75.9nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85995([leu13]pMOT(1-11))
Affinity DataKi:  89.1nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50503156(CHEMBL4468977)
Affinity DataKi:  112nMAssay Description:Displacement of [3H]JNJ-46281222 from human mGlu2 receptor expressed in CHOK1 cell membranes after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85998(Erythromycin-B)
Affinity DataKi:  145nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50194617(CHEMBL3926416)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]8-Trifluoromethyl-3-cyclopropylmethyl-7-[(4-phenyl-1-piperidinyl)methyl]-1,2,4-triazolo[4,3-a]pyridine from mGlu2 receptor (unkno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50503156(CHEMBL4468977)
Affinity DataKi:  166nMAssay Description:Displacement of [3H]JNJ-46281222 from human mGlu2 receptor expressed in CHOK1 cell membranes preincubated for 3 hrs followed by [3H]JNJ-46281222 addi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50503157(CHEMBL4538850)
Affinity DataKi:  174nMAssay Description:Displacement of [3H]JNJ-46281222 from human mGlu2 receptor transiently expressed in CHOK1 cell membranes after 1 hr by liquid scintillation counting ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50051408(CHEMBL3337527 | US11071729, Compound 2)
Affinity DataKi:  180nMAssay Description:Displacement of [3H]8-Trifluoromethyl-3-cyclopropylmethyl-7-[(4-phenyl-1-piperidinyl)methyl]-1,2,4-triazolo[4,3-a]pyridine from mGlu2 receptor (unkno...More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50503157(CHEMBL4538850)
Affinity DataKi:  234nMAssay Description:Irreversible displacement of [3H]JNJ-46281222 from human mGlu2 receptor expressed in CHOK1 cell membranes preincubated for 1 hr in presence of glutam...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85988(N-ethyl, N-Methyl Erythromycin-A)
Affinity DataKi:  240nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85846(CAS_33396-29-1 | EM523 | Erythromycin A 6,9-enolet...)
Affinity DataKi:  257nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM86688(EM-B enolether)
Affinity DataKi:  324nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM86686(Erythromycin A Enol Ether | ME4)
Affinity DataKi:  537nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85981([ala1,leu13]pMOT(1-14) | [leu13]pMOT(1-14))
Affinity DataKi:  589nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85982([ala7,leu13]pMOT(1-14))
Affinity DataKi:  1.45E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM86000([ala4,leu13]pMOT(1-14))
Affinity DataKi:  2.57E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM86313(CAS_114-07-8 | NSC_12560 | erythromycin-A)
Affinity DataKi:  3.09E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85996([leu13]pMOT(1-9))
Affinity DataKi:  4.07E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM86001([leu13]pMOT(1-7))
Affinity DataKi:  6.92E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM85985([leu13]pMOT(1-5))
Affinity DataKi:  8.91E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPromotilin(Homo sapiens (Human))
Katholieke Universiteit Leuven

Curated by PDSP Ki Database
LigandPNGBDBM86687(ME36)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Janssen Pharmaceutica

Curated by ChEMBL
LigandPNGBDBM50194617(CHEMBL3926416)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Janssen Pharmaceutica

Curated by ChEMBL
LigandPNGBDBM50194617(CHEMBL3926416)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Janssen Pharmaceutica

Curated by ChEMBL
LigandPNGBDBM50194617(CHEMBL3926416)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of CYP1A2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C8(Homo sapiens (Human))
Janssen Pharmaceutica

Curated by ChEMBL
LigandPNGBDBM50194617(CHEMBL3926416)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of CYP2C8 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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