Affinity DataKi: 0.510nMAssay Description:Displacement of [3H]substance P from human NK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.610nMAssay Description:Displacement of [3H]substance P from human NK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.740nMAssay Description:Displacement of [3H]SR142801 from human NK3 receptor expressed in HEK-293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.780nMAssay Description:Displacement of [3H]substance P from human NK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.860nMAssay Description:Displacement of [3H]substance P from human NK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.910nMAssay Description:Displacement of [3H]substance P from human NK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.910nMAssay Description:Displacement of [3H]SR142801 from human NK3 receptor expressed in HEK-293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.910nMAssay Description:Displacement of [3H]SR142801 from human NK3 receptor expressed in HEK-293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.950nMAssay Description:Displacement of [3H]SR142801 from human NK3 receptor expressed in HEK-293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Displacement of [3H]MPEP from recombinant human mGlu5 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Displacement of [3H]substance P from human NK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.12nMAssay Description:Displacement of [3H]SR142801 from human NK3 receptor expressed in HEK-293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.12nMAssay Description:Displacement of [3H]substance P from human NK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.15nMAssay Description:Displacement of [3H]substance P from human NK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity to rat 5HT5A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.38nMAssay Description:Displacement of [3H]substance P from human NK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.48nMAssay Description:Displacement of [3H]SR142801 from human NK3 receptor expressed in HEK-293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.58nMAssay Description:Displacement of [3H]substance P from human NK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.58nMAssay Description:Displacement of [3H]substance P from human NK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Binding affinity to human 5HT5A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.72nMAssay Description:Displacement of [3H]substance P from human NK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Binding affinity to human 5HT5A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.24nMAssay Description:Displacement of [3H]substance P from human NK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.27nMAssay Description:Displacement of [3H]substance P from human NK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Binding affinity to histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.62nMAssay Description:Displacement of [3H]substance P from human NK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Binding affinity to rat 5HT5A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.91nMAssay Description:Displacement of [3H]SR142801 from human NK3 receptor expressed in HEK-293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.05nMAssay Description:Displacement of [3H]substance P from human NK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
F. Hoffmann-La Roche
Curated by PDSP Ki Database
F. Hoffmann-La Roche
Curated by PDSP Ki Database
Affinity DataKi: 3.37nMAssay Description:Displacement of [3H]substance P from human NK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Binding affinity to human 5HT7 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:Displacement of [3H]MPEP from recombinant human mGlu5 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:Binding affinity to dopamine D2 receptor (unknown origin) by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Displacement of [3H]MPEP from recombinant human mGlu5 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.10nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
F. Hoffmann-La Roche
Curated by PDSP Ki Database
F. Hoffmann-La Roche
Curated by PDSP Ki Database
Affinity DataKi: 5.40nMAssay Description:Displacement of [3H]SR142801 from human NK3 receptor expressed in HEK-293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.70nMAssay Description:Binding affinity to human 5HT5A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Binding affinity to human 5HT7 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Displacement of [3H]MPEP from recombinant human mGlu5 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair