Affinity DataKi: 0.110nMAssay Description:Inhibitory potency was measured against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.110nM ΔG°: -56.3kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme activities were determined kinetically as the initial rate of cleavage of a peptide p-nitroanilide. Km for enzyme and substrate was determ...More data for this Ligand-Target Pair
Affinity DataKi: 0.110nM ΔG°: -56.3kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme activities were determined kinetically as the initial rate of cleavage of a peptide p-nitroanilide. Km for enzyme and substrate was determ...More data for this Ligand-Target Pair
Affinity DataKi: 0.110nM ΔG°: -56.3kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme activities were determined kinetically as the initial rate of cleavage of a peptide p-nitroanilide. Km for enzyme and substrate was determ...More data for this Ligand-Target Pair
Affinity DataKi: 0.120nMAssay Description:Binding affinity at histamine H3 receptor in rat cortical membranes by [3H]-Nalpha-methylhistamine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.180nMAssay Description:Histamine H3 receptor affinity of compound was determined in rat cortical membranes using the H3 selective agonist ligand, [3H]N-alpha-methylhistamin...More data for this Ligand-Target Pair
Affinity DataKi: 0.180nMAssay Description:Inhibition of [3H]- N-alpha-methylhistamine from histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.240nMAssay Description:Inhibitory potency was measured against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.260nMAssay Description:Inhibitory potency was measured against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.270nM ΔG°: -54.1kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme activities were determined kinetically as the initial rate of cleavage of a peptide p-nitroanilide. Km for enzyme and substrate was determ...More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Histamine H3 receptor affinity of compound was determined in rat cortical membranes using the H3 selective agonist ligand, [3H]N-alpha-methylhistamin...More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:The enzyme activities were determined kinetically as the initial rate of cleavage of a peptide p-nitroanilide. Km for enzyme and substrate was determ...More data for this Ligand-Target Pair
Affinity DataKi: 0.310nMAssay Description:Inhibitory potency was measured against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.320nMAssay Description:Inhibition constant against human factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.330nMAssay Description:Inhibitory potency was measured against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.330nM ΔG°: -53.6kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme activities were determined kinetically as the initial rate of cleavage of a peptide p-nitroanilide. Km for enzyme and substrate was determ...More data for this Ligand-Target Pair
Affinity DataKi: 0.330nMAssay Description:Binding affinity at histamine H3 receptor in rat cortical membranes by [3H]-Nalpha-methylhistamine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.380nMAssay Description:The enzyme activities were determined kinetically as the initial rate of cleavage of a peptide p-nitroanilide. Km for enzyme and substrate was determ...More data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:The enzyme activities were determined kinetically as the initial rate of cleavage of a peptide p-nitroanilide. Km for enzyme and substrate was determ...More data for this Ligand-Target Pair
Affinity DataKi: 0.410nMAssay Description:Inhibitory potency was measured against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.430nMAssay Description:Inhibitory potency was measured against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.450nMAssay Description:The enzyme activities were determined kinetically as the initial rate of cleavage of a peptide p-nitroanilide. Km for enzyme and substrate was determ...More data for this Ligand-Target Pair
Affinity DataKi: 0.460nMAssay Description:Inhibition constant against human factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Binding affinity against [3H]- -8-OH-DPAT -labeled 5-hydroxytryptamine 1A sites in cloned CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Inhibition of [3H]- N-alpha-methylhistamine from histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.520nMAssay Description:The enzyme activities were determined kinetically as the initial rate of cleavage of a peptide p-nitroanilide. Km for enzyme and substrate was determ...More data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Antagonist activity against platelet activating factor (PAF) receptor in rabbit platelet membranes using [3H]C18-PAF as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nM ΔG°: -52.1kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme activities were determined kinetically as the initial rate of cleavage of a peptide p-nitroanilide. Km for enzyme and substrate was determ...More data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Inhibition constant against human factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:The enzyme activities were determined kinetically as the initial rate of cleavage of a peptide p-nitroanilide. Km for enzyme and substrate was determ...More data for this Ligand-Target Pair
Affinity DataKi: 0.650nMAssay Description:Inhibitory potency was measured against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.660nMAssay Description:Inhibitory potency was measured against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.660nMAssay Description:Compound was tested for inhibition activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.660nM ΔG°: -51.9kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme activities were determined kinetically as the initial rate of cleavage of a peptide p-nitroanilide. Km for enzyme and substrate was determ...More data for this Ligand-Target Pair
Affinity DataKi: 0.710nMAssay Description:Inhibitory potency was measured against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:The enzyme activities were determined kinetically as the initial rate of cleavage of a peptide p-nitroanilide. Km for enzyme and substrate was determ...More data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Antagonist activity against platelet activating factor (PAF) receptor in rabbit platelet membranes using [3H]C18-PAF as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Binding affinity at histamine H3 receptor in rat cortical membranes by [3H]-Nalpha-methylhistamine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Inhibition of [3H]- N-alpha-methylhistamine from histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:The enzyme activities were determined kinetically as the initial rate of cleavage of a peptide p-nitroanilide. Km for enzyme and substrate was determ...More data for this Ligand-Target Pair
Affinity DataKi: 0.820nM ΔG°: -51.3kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme activities were determined kinetically as the initial rate of cleavage of a peptide p-nitroanilide. Km for enzyme and substrate was determ...More data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Binding affinity at histamine H3 receptor in rat cortical membranes by [3H]-Nalpha-methylhistamine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.950nMAssay Description:Inhibition of [3H]- N-alpha-methylhistamine from histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.950nM ΔG°: -51.0kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme activities were determined kinetically as the initial rate of cleavage of a peptide p-nitroanilide. Km for enzyme and substrate was determ...More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Antagonist activity against platelet activating factor (PAF) receptor in rabbit platelet membranes using [3H]C18-PAF as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Antagonist activity against platelet activating factor (PAF) receptor in rabbit platelet membranes using [3H]C18-PAF as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of [3H]- N-alpha-methylhistamine from histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1nM ΔG°: -50.9kJ/molepH: 7.5 T: 2°CAssay Description:The enzyme activities were determined kinetically as the initial rate of cleavage of a peptide p-nitroanilide. Km for enzyme and substrate was determ...More data for this Ligand-Target Pair