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Found 20 with Last Name = 'quéléver' and Initial = 'g'
TargetBeta-secretase 1(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50180393(CHEMBL205309 | tert-butyl 4-(4-bromo-2-(2-(7-metho...)
Affinity DataIC50:  93nMAssay Description:Inhibition of BACE1 activity by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM16741(2,2,2-trifluoroacetic acid; N-[5-bromo-2-(piperazi...)
Affinity DataIC50:  670nMAssay Description:Inhibition of BACE1 activity by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM16740(CHEMBL206442 | Coumarin Compound, 9c | N-[2-(4-ben...)
Affinity DataIC50:  760nMAssay Description:Inhibition of BACE1 activity by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM16739(CHEMBL207083 | Coumarin Compound, 9b | tert-butyl ...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of BACE1 activity by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM16726(CHEMBL203120 | N-[5-bromo-2-(piperazin-1-yl)phenyl...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of BACE1 activity by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50180395(CHEMBL205637 | N-(5-bromo-2-(4-(thiophen-2-ylsulfo...)
Affinity DataIC50:  1.13E+3nMAssay Description:Inhibition of BACE1 activity by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50180396(4-Oxo-4H-chromene-2-carboxylic acid (5-bromo-2-pip...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of BACE1 activity by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50180391(CHEMBL206651 | tert-butyl 4-(4-bromo-2-(quinoline-...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of BACE1 activity by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM16724(CHEMBL381618 | Naphthyl Compound, 3b | tert-butyl ...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of BACE1 activity by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50180394(CHEMBL205241 | N-(5-bromo-2-piperazin-1-yl-phenyl)...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of BACE1 activity by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50180398(CHEMBL206665 | tert-butyl 4-(4-bromo-2-(4-oxo-4H-c...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of BACE1 activity by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM16744(CHEMBL206854 | Coumarin Compound, 10b | tert-butyl...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of BACE1 activity by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50180399(CHEMBL206097 | N-(5-bromo-2-(4-(thiophen-2-ylsulfo...)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of BACE1 activity by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50180392(CHEMBL377745 | quinoline-2-carboxylic acid (5-brom...)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of BACE1 activity by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM16746(2,2,2-trifluoroacetic acid; N-[5-bromo-2-(piperazi...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of BACE1 activity by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM16725(CHEMBL380521 | N-[2-(4-benzylpiperazin-1-yl)-5-bro...)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of BACE1 activity by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM16745(CHEMBL381617 | Coumarin Compound, 10c | N-[2-(4-be...)
Affinity DataIC50:  5.50E+3nMAssay Description:Inhibition of BACE1 activity by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50157216(2-Bromomethyl-8-nitro-benzo[c]chromen-6-one | CHEM...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory concentration against HIV aspartyl proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50157217(2-Methyl-8-nitro-benzo[c]chromen-6-one | CHEMBL182...)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibitory concentration against HIV aspartyl proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of The Mediterranean

Curated by ChEMBL
LigandPNGBDBM50157215(8-Amino-2-bromomethyl-benzo[c]chromen-6-one | CHEM...)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibitory concentration against HIV aspartyl proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed