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Found 158 with Last Name = 'ragab' and Initial = 'fa'
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
Egypt National Research Centre

Curated by ChEMBL
LigandPNGBDBM50263771(1-benzoyl-3-((2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(...)
Affinity DataKi:  4.60E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase bMore data for this Ligand-Target Pair
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
Egypt National Research Centre

Curated by ChEMBL
LigandPNGBDBM50295859((2S,3R,4R,5S,6R)-2-(1H-benzo[d]imidazol-2-yl)-6-(h...)
Affinity DataKi:  9.00E+3nMAssay Description:Inhibition of rabbit skeletal muscle glycogen phosphorylase b assessed as inorganic phosphate release using glucose-1-phosphate as substrate by doubl...More data for this Ligand-Target Pair
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
Egypt National Research Centre

Curated by ChEMBL
LigandPNGBDBM50295859((2S,3R,4R,5S,6R)-2-(1H-benzo[d]imidazol-2-yl)-6-(h...)
Affinity DataKi:  1.10E+4nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase b using alpha-D-glucose-1-phosphate as substrateMore data for this Ligand-Target Pair
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
Egypt National Research Centre

Curated by ChEMBL
LigandPNGBDBM50295860((2R,3R,4S,5S,6R)-2-(benzo[d]thiazol-2-yl)-6-(hydro...)
Affinity DataKi:  7.60E+4nMAssay Description:Inhibition of rabbit skeletal muscle glycogen phosphorylase b assessed as inorganic phosphate release using glucose-1-phosphate as substrate by doubl...More data for this Ligand-Target Pair
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
Egypt National Research Centre

Curated by ChEMBL
LigandPNGBDBM50295860((2R,3R,4S,5S,6R)-2-(benzo[d]thiazol-2-yl)-6-(hydro...)
Affinity DataKi:  2.29E+5nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase b using alpha-D-glucose-1-phosphate as substrateMore data for this Ligand-Target Pair
LigandPNGBDBM50145416(GSK2126458 | Omipalisib)
Affinity DataIC50:  0.0190nMAssay Description:Competitive inhibition of human PI3K p110alpha/p85alpha using PIP2 as substrate preincubated for 10 mins followed by ATP addition measured after 30 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50145416(GSK2126458 | Omipalisib)
Affinity DataIC50:  0.180nMAssay Description:Competitive inhibition of human mTOR using 4EBP1 as substrate in presence of [33gammaP]-ATP after 120 mins by filter binding methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50243194(CHEMBL4097194)
Affinity DataIC50:  0.240nMAssay Description:Competitive inhibition of human PI3K p110alpha/p85alpha using PIP2 as substrate preincubated for 10 mins followed by ATP addition measured after 30 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50243144(CHEMBL4065928)
Affinity DataIC50:  0.400nMAssay Description:Competitive inhibition of human PI3K p110alpha/p85alpha using PIP2 as substrate preincubated for 10 mins followed by ATP addition measured after 30 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50243193(CHEMBL4060651)
Affinity DataIC50: <0.5nMAssay Description:Competitive inhibition of human PI3K p110alpha/p85alpha using PIP2 as substrate preincubated for 10 mins followed by ATP addition measured after 30 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50243339(CHEMBL4089494)
Affinity DataIC50: <0.5nMAssay Description:Competitive inhibition of human PI3K p110alpha/p85alpha using PIP2 as substrate preincubated for 10 mins followed by ATP addition measured after 30 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50243292(CHEMBL4092587)
Affinity DataIC50:  0.570nMAssay Description:Competitive inhibition of human PI3K p110alpha/p85alpha using PIP2 as substrate preincubated for 10 mins followed by ATP addition measured after 30 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50243304(CHEMBL4104902)
Affinity DataIC50:  0.630nMAssay Description:Competitive inhibition of human PI3K p110alpha/p85alpha using PIP2 as substrate preincubated for 10 mins followed by ATP addition measured after 30 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50243145(CHEMBL3109141)
Affinity DataIC50:  1nMAssay Description:Competitive inhibition of human mTOR using 4EBP1 as substrate in presence of [33gammaP]-ATP after 120 mins by filter binding methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50243144(CHEMBL4065928)
Affinity DataIC50:  1.60nMAssay Description:Competitive inhibition of human mTOR using 4EBP1 as substrate in presence of [33gammaP]-ATP after 120 mins by filter binding methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50243176(CHEMBL4081617)
Affinity DataIC50:  1.70nMAssay Description:Competitive inhibition of human PI3K p110alpha/p85alpha using PIP2 as substrate preincubated for 10 mins followed by ATP addition measured after 30 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50243146(CHEMBL4102783)
Affinity DataIC50:  1.90nMAssay Description:Competitive inhibition of human PI3K p110alpha/p85alpha using PIP2 as substrate preincubated for 10 mins followed by ATP addition measured after 30 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM25045(3-(4-morpholin-4-ylpyrido[2,3]furo[2,4-b]pyrimidin...)
Affinity DataIC50:  2nMAssay Description:Competitive inhibition of human PI3K p110alpha/p85alpha using PIP2 as substrate preincubated for 10 mins followed by ATP addition measured after 30 m...More data for this Ligand-Target Pair
LigandPNGBDBM50243195(CHEMBL4079178)
Affinity DataIC50:  2.5nMAssay Description:Competitive inhibition of human PI3K p110alpha/p85alpha using PIP2 as substrate preincubated for 10 mins followed by ATP addition measured after 30 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50243313(CHEMBL4103534)
Affinity DataIC50:  2.5nMAssay Description:Competitive inhibition of human PI3K p110alpha/p85alpha using PIP2 as substrate preincubated for 10 mins followed by ATP addition measured after 30 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50243196(CHEMBL4087043)
Affinity DataIC50:  2.80nMAssay Description:Competitive inhibition of human PI3K p110alpha/p85alpha using PIP2 as substrate preincubated for 10 mins followed by ATP addition measured after 30 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50429701(AZD-2014 | CHEMBL2336325 | US9102670, 1ap)
Affinity DataIC50:  2.80nMAssay Description:Competitive inhibition of human mTOR using 4EBP1 as substrate in presence of [33gammaP]-ATP after 120 mins by filter binding methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50243293(CHEMBL4088235)
Affinity DataIC50:  2.90nMAssay Description:Competitive inhibition of human PI3K p110alpha/p85alpha using PIP2 as substrate preincubated for 10 mins followed by ATP addition measured after 30 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50243172(CHEMBL4059989)
Affinity DataIC50:  3.30nMAssay Description:Competitive inhibition of human PI3K p110alpha/p85alpha using PIP2 as substrate preincubated for 10 mins followed by ATP addition measured after 30 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50243230(CHEMBL4092840)
Affinity DataIC50:  3.60nMAssay Description:Competitive inhibition of human PI3K p110alpha/p85alpha using PIP2 as substrate preincubated for 10 mins followed by ATP addition measured after 30 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50243304(CHEMBL4104902)
Affinity DataIC50:  3.60nMAssay Description:Competitive inhibition of human mTOR using 4EBP1 as substrate in presence of [33gammaP]-ATP after 120 mins by filter binding methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50243251(CHEMBL4088056)
Affinity DataIC50:  3.70nMAssay Description:Competitive inhibition of human PI3K p110alpha/p85alpha using PIP2 as substrate preincubated for 10 mins followed by ATP addition measured after 30 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50243248(CHEMBL4102715)
Affinity DataIC50:  4.10nMAssay Description:Competitive inhibition of human PI3K p110alpha/p85alpha using PIP2 as substrate preincubated for 10 mins followed by ATP addition measured after 30 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50243143(CHEMBL3109142)
Affinity DataIC50:  5nMAssay Description:Competitive inhibition of human mTOR using 4EBP1 as substrate in presence of [33gammaP]-ATP after 120 mins by filter binding methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50243296(CHEMBL4065878)
Affinity DataIC50:  5.40nMAssay Description:Competitive inhibition of human PI3K p110alpha/p85alpha using PIP2 as substrate preincubated for 10 mins followed by ATP addition measured after 30 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50243249(CHEMBL4079272)
Affinity DataIC50:  5.60nMAssay Description:Competitive inhibition of human PI3K p110alpha/p85alpha using PIP2 as substrate preincubated for 10 mins followed by ATP addition measured after 30 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50243246(CHEMBL4064842)
Affinity DataIC50:  5.70nMAssay Description:Competitive inhibition of human PI3K p110alpha/p85alpha using PIP2 as substrate preincubated for 10 mins followed by ATP addition measured after 30 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50243314(CHEMBL4087157)
Affinity DataIC50:  6.10nMAssay Description:Competitive inhibition of human PI3K p110alpha/p85alpha using PIP2 as substrate preincubated for 10 mins followed by ATP addition measured after 30 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50243247(CHEMBL4092544)
Affinity DataIC50:  7.80nMAssay Description:Competitive inhibition of human PI3K p110alpha/p85alpha using PIP2 as substrate preincubated for 10 mins followed by ATP addition measured after 30 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50243253(CHEMBL4095781)
Affinity DataIC50:  8.80nMAssay Description:Competitive inhibition of human mTOR using 4EBP1 as substrate in presence of [33gammaP]-ATP after 120 mins by filter binding methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50243254(CHEMBL4069475)
Affinity DataIC50:  9.90nMAssay Description:Competitive inhibition of human mTOR using 4EBP1 as substrate in presence of [33gammaP]-ATP after 120 mins by filter binding methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50243252(CHEMBL4059778)
Affinity DataIC50:  16nMAssay Description:Competitive inhibition of human mTOR using 4EBP1 as substrate in presence of [33gammaP]-ATP after 120 mins by filter binding methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50243251(CHEMBL4088056)
Affinity DataIC50:  19nMAssay Description:Competitive inhibition of human mTOR using 4EBP1 as substrate in presence of [33gammaP]-ATP after 120 mins by filter binding methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM25045(3-(4-morpholin-4-ylpyrido[2,3]furo[2,4-b]pyrimidin...)
Affinity DataIC50:  20nMAssay Description:Competitive inhibition of human mTOR using 4EBP1 as substrate in presence of [33gammaP]-ATP after 120 mins by filter binding methodMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50243194(CHEMBL4097194)
Affinity DataIC50:  23nMAssay Description:Competitive inhibition of human mTOR using 4EBP1 as substrate in presence of [33gammaP]-ATP after 120 mins by filter binding methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50243231(CHEMBL4072084)
Affinity DataIC50:  26nMAssay Description:Competitive inhibition of human mTOR using 4EBP1 as substrate in presence of [33gammaP]-ATP after 120 mins by filter binding methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
National Center For Radiation Research And Technology (Ncrrt)

Curated by ChEMBL
LigandPNGBDBM16673(4-[4-({[4-chloro-3-(trifluoromethyl)phenyl]carbamo...)
Affinity DataIC50:  30nMAssay Description:Inhibition of human VEGFR-2 after 2.5 hrs by ELISAMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50243313(CHEMBL4103534)
Affinity DataIC50:  31nMAssay Description:Competitive inhibition of human mTOR using 4EBP1 as substrate in presence of [33gammaP]-ATP after 120 mins by filter binding methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
National Center For Radiation Research And Technology (Ncrrt)

Curated by ChEMBL
LigandPNGBDBM50461329(CHEMBL4225623)
Affinity DataIC50:  33nMAssay Description:Inhibition of human VEGFR-2 after 2.5 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50243249(CHEMBL4079272)
Affinity DataIC50:  33nMAssay Description:Competitive inhibition of human mTOR using 4EBP1 as substrate in presence of [33gammaP]-ATP after 120 mins by filter binding methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50243303(CHEMBL4084790)
Affinity DataIC50:  35nMAssay Description:Competitive inhibition of human PI3K p110alpha/p85alpha using PIP2 as substrate preincubated for 10 mins followed by ATP addition measured after 30 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
National Center For Radiation Research And Technology (Ncrrt)

Curated by ChEMBL
LigandPNGBDBM50461332(CHEMBL4226159)
Affinity DataIC50:  37nMAssay Description:Inhibition of human VEGFR-2 after 2.5 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
National Center For Radiation Research And Technology (Ncrrt)

Curated by ChEMBL
LigandPNGBDBM50461334(CHEMBL4225317)
Affinity DataIC50:  37nMAssay Description:Inhibition of human VEGFR-2 after 2.5 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50243248(CHEMBL4102715)
Affinity DataIC50:  37nMAssay Description:Competitive inhibition of human mTOR using 4EBP1 as substrate in presence of [33gammaP]-ATP after 120 mins by filter binding methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50243145(CHEMBL3109141)
Affinity DataIC50:  40nMAssay Description:Competitive inhibition of human PI3K p110alpha/p85alpha using PIP2 as substrate preincubated for 10 mins followed by ATP addition measured after 30 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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