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Found 50 with Last Name = 'rajagopalan' and Initial = 'dr'
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50000492((zacopride)4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3-yl...)
Affinity DataKi:  0.390nMAssay Description:Displacement of [3H]GR65630 from 5-HT3 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50000492((zacopride)4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3-yl...)
Affinity DataKi:  0.398nMAssay Description:Displacement of [3H]GR65630 from 5-HT3 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  1.66nMAssay Description:Displacement of [3H](+)Pentazocine from sigma 1 receptor (unknown origin)More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H](+)Pentazocine from sigma 1 receptor (unknown origin)More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]N-Methylspiperone from dopamine D2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]N-Methylspiperone from dopamine D2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM35938(1-(p-chlorophenyl)-1-(2-pyridyl)-3-N,N-dimethylpro...)
Affinity DataKi:  4.47nMAssay Description:Displacement of [3H]Pyrilamine from histamine H1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM35938(1-(p-chlorophenyl)-1-(2-pyridyl)-3-N,N-dimethylpro...)
Affinity DataKi:  4.5nMAssay Description:Displacement of [3H]Pyrilamine from histamine H1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetHistamine H2 receptor(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50445613(Asenapine maleate | CHEBI:71246 | ORG-5222 | Saphr...)
Affinity DataKi:  5.70nMAssay Description:Displacement of [3H]Cimetidine from histamine H2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50445613(Asenapine maleate | CHEBI:71246 | ORG-5222 | Saphr...)
Affinity DataKi:  5.80nMAssay Description:Displacement of [3H]Cimetidine from histamine H2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50445615(CHEMBL3104092)
Affinity DataKi:  48nMAssay Description:Displacement of [3H]Pyrilamine from histamine H1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50445615(CHEMBL3104092)
Affinity DataKi:  48nMAssay Description:Displacement of [3H]Pyrilamine from histamine H1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50445616(CHEMBL3104091)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]Pyrilamine from histamine H1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50445616(CHEMBL3104091)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]Pyrilamine from histamine H1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50403559(Brumetadina | CIMETIDINE)
Affinity DataKi:  70nMAssay Description:Displacement of [3H]Cimetidine from histamine H2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50403559(Brumetadina | CIMETIDINE)
Affinity DataKi:  71nMAssay Description:Displacement of [3H]Cimetidine from histamine H2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50445616(CHEMBL3104091)
Affinity DataKi:  81nMAssay Description:Displacement of [3H]Cimetidine from histamine H2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50445616(CHEMBL3104091)
Affinity DataKi:  81nMAssay Description:Displacement of [3H]Cimetidine from histamine H2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50445614(CHEMBL3104093)
Affinity DataKi:  104nMAssay Description:Binding affinity to 5-HT2B receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50445614(CHEMBL3104093)
Affinity DataKi:  195nMAssay Description:Binding affinity to 5-HT7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50445614(CHEMBL3104093)
Affinity DataKi:  219nMAssay Description:Displacement of [3H](+)Pentazocine from sigma 1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50445614(CHEMBL3104093)
Affinity DataKi:  220nMAssay Description:Binding affinity to sigma1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50445614(CHEMBL3104093)
Affinity DataKi:  220nMAssay Description:Displacement of [3H](+)Pentazocine from sigma 1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50445614(CHEMBL3104093)
Affinity DataKi:  257nMAssay Description:Binding affinity to 5-HT2A receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50445614(CHEMBL3104093)
Affinity DataKi:  286nMAssay Description:Binding affinity to adrenergic alpha 1A receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50445614(CHEMBL3104093)
Affinity DataKi:  293nMAssay Description:Binding affinity to adrenergic alpha 1D receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50445614(CHEMBL3104093)
Affinity DataKi:  407nMAssay Description:Binding affinity to adrenergic alpha 2A receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50445614(CHEMBL3104093)
Affinity DataKi:  446nMAssay Description:Binding affinity to adrenergic alpha 2C receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50445614(CHEMBL3104093)
Affinity DataKi:  501nMAssay Description:Displacement of [3H]GR65630 from 5-HT3 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50445614(CHEMBL3104093)
Affinity DataKi:  529nMAssay Description:Displacement of [3H]GR65630 from 5-HT3 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50445616(CHEMBL3104091)
Affinity DataKi:  832nMAssay Description:Displacement of [3H]N-Methylspiperone from dopamine D2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50445616(CHEMBL3104091)
Affinity DataKi:  835nMAssay Description:Displacement of [3H]N-Methylspiperone from dopamine D2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50445614(CHEMBL3104093)
Affinity DataKi:  933nMAssay Description:Displacement of [3H]Cimetidine from histamine H2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50445614(CHEMBL3104093)
Affinity DataKi:  943nMAssay Description:Displacement of [3H]Cimetidine from histamine H2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50445616(CHEMBL3104091)
Affinity DataKi:  6.14E+3nMAssay Description:Displacement of [3H](+)Pentazocine from sigma 1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50445616(CHEMBL3104091)
Affinity DataKi:  6.31E+3nMAssay Description:Displacement of [3H](+)Pentazocine from sigma 1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50445614(CHEMBL3104093)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]N-Methylspiperone from dopamine D2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50445614(CHEMBL3104093)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Pyrilamine from histamine H1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50445616(CHEMBL3104091)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]GR65630 from 5-HT3 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50445615(CHEMBL3104092)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]GR65630 from 5-HT3 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50445615(CHEMBL3104092)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]N-Methylspiperone from dopamine D2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50445615(CHEMBL3104092)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Cimetidine from histamine H2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50445615(CHEMBL3104092)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H](+)Pentazocine from sigma 1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50445614(CHEMBL3104093)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to SST4 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50445614(CHEMBL3104093)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to SST2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50445614(CHEMBL3104093)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to cannabinoid CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50445614(CHEMBL3104093)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to cannabinoid CB1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50445614(CHEMBL3104093)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to adenosine A3 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50445614(CHEMBL3104093)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to adenosine A1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Missouri

Curated by ChEMBL
LigandPNGBDBM50445614(CHEMBL3104093)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to adenosine A2A receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed