TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Signal Pharmaceuticals
Curated by ChEMBL
Signal Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Concentration required to inhibit activator protein-1(AP-1) mediated transcriptional activation in human Jurkat T-cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Concentration required to inhibit activator protein-1(AP-1) mediated transcriptional activation in human Jurkat T-cellsMore data for this Ligand-Target Pair
TargetNuclear factor NF-kappa-B p105 subunit(Homo sapiens (Human))
Signal Pharmaceuticals
Curated by ChEMBL
Signal Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:In vitro inhibitory activity against human Jurkat T-Cells stably transfected with an Nuclear factor kappa B transcription factorMore data for this Ligand-Target Pair
TargetCyclic AMP-dependent transcription factor ATF-1(Homo sapiens (Human))
Signal Pharmaceuticals
Curated by ChEMBL
Signal Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:In vitro inhibitory activity against human Jurkat T-Cells stably transfected with activating transcription factor 1More data for this Ligand-Target Pair
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Signal Pharmaceuticals
Curated by ChEMBL
Signal Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Signal Pharmaceuticals
Curated by ChEMBL
Signal Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Concentration required to inhibit activator protein-1(AP-1) mediated transcriptional activation in human Jurkat T-cellsMore data for this Ligand-Target Pair
TargetCyclic AMP-dependent transcription factor ATF-1(Homo sapiens (Human))
Signal Pharmaceuticals
Curated by ChEMBL
Signal Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:In vitro inhibitory activity against human Jurkat T-Cells stably transfected with activating transcription factor 1More data for this Ligand-Target Pair
TargetCyclic AMP-dependent transcription factor ATF-1(Homo sapiens (Human))
Signal Pharmaceuticals
Curated by ChEMBL
Signal Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:In vitro inhibitory activity against human Jurkat T-Cells stably transfected with activating transcription factor 1More data for this Ligand-Target Pair
TargetNuclear factor NF-kappa-B p105 subunit(Homo sapiens (Human))
Signal Pharmaceuticals
Curated by ChEMBL
Signal Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:In vitro inhibitory activity against human Jurkat T-Cells stably transfected with an Nuclear factor kappa B transcription factorMore data for this Ligand-Target Pair
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Signal Pharmaceuticals
Curated by ChEMBL
Signal Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Signal Pharmaceuticals
Curated by ChEMBL
Signal Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Signal Pharmaceuticals
Curated by ChEMBL
Signal Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Signal Pharmaceuticals
Curated by ChEMBL
Signal Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Signal Pharmaceuticals
Curated by ChEMBL
Signal Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Concentration required to inhibit activator protein-1(AP-1) mediated transcriptional activation in human Jurkat T-cellsMore data for this Ligand-Target Pair
TargetNuclear factor NF-kappa-B p105 subunit(Homo sapiens (Human))
Signal Pharmaceuticals
Curated by ChEMBL
Signal Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 280nMAssay Description:In vitro inhibitory activity against human Jurkat T-Cells stably transfected with an Nuclear factor kappa B transcription factorMore data for this Ligand-Target Pair
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Signal Pharmaceuticals
Curated by ChEMBL
Signal Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Signal Pharmaceuticals
Curated by ChEMBL
Signal Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Signal Pharmaceuticals
Curated by ChEMBL
Signal Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Signal Pharmaceuticals
Curated by ChEMBL
Signal Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Concentration required to inhibit activator protein-1(AP-1) mediated transcriptional activation in human Jurkat T-cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Concentration required to inhibit activator protein-1(AP-1) mediated transcriptional activation in human Jurkat T-cellsMore data for this Ligand-Target Pair
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Signal Pharmaceuticals
Curated by ChEMBL
Signal Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
TargetNuclear factor NF-kappa-B p105 subunit(Homo sapiens (Human))
Signal Pharmaceuticals
Curated by ChEMBL
Signal Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 380nMAssay Description:In vitro inhibitory activity against human Jurkat T-Cells stably transfected with an Nuclear factor kappa B transcription factorMore data for this Ligand-Target Pair
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Signal Pharmaceuticals
Curated by ChEMBL
Signal Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Concentration required to inhibit activator protein-1(AP-1) mediated transcriptional activation in human Jurkat T-cellsMore data for this Ligand-Target Pair
TargetCyclic AMP-dependent transcription factor ATF-1(Homo sapiens (Human))
Signal Pharmaceuticals
Curated by ChEMBL
Signal Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 490nMAssay Description:In vitro inhibitory activity against human Jurkat T-Cells stably transfected with activating transcription factor 1More data for this Ligand-Target Pair
TargetCyclic AMP-dependent transcription factor ATF-1(Homo sapiens (Human))
Signal Pharmaceuticals
Curated by ChEMBL
Signal Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:In vitro inhibitory activity against human Jurkat T-Cells stably transfected with activating transcription factor 1More data for this Ligand-Target Pair
TargetNuclear factor NF-kappa-B p105 subunit(Homo sapiens (Human))
Signal Pharmaceuticals
Curated by ChEMBL
Signal Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:In vitro inhibitory activity against human Jurkat T-Cells stably transfected with an Nuclear factor kappa B transcription factorMore data for this Ligand-Target Pair
TargetCyclic AMP-dependent transcription factor ATF-1(Homo sapiens (Human))
Signal Pharmaceuticals
Curated by ChEMBL
Signal Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:In vitro inhibitory activity against human Jurkat T-Cells stably transfected with activating transcription factor 1More data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Concentration required to inhibit activator protein-1(AP-1) mediated transcriptional activation in human Jurkat T-cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Concentration required to inhibit activator protein-1(AP-1) mediated transcriptional activation in human Jurkat T-cellsMore data for this Ligand-Target Pair
TargetNuclear factor NF-kappa-B p105 subunit(Homo sapiens (Human))
Signal Pharmaceuticals
Curated by ChEMBL
Signal Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 620nMAssay Description:In vitro inhibitory activity against human Jurkat T-Cells stably transfected with an Nuclear factor kappa B transcription factorMore data for this Ligand-Target Pair
TargetCyclic AMP-dependent transcription factor ATF-1(Homo sapiens (Human))
Signal Pharmaceuticals
Curated by ChEMBL
Signal Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 660nMAssay Description:In vitro inhibitory activity against human Jurkat T-Cells stably transfected with activating transcription factor 1More data for this Ligand-Target Pair
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Signal Pharmaceuticals
Curated by ChEMBL
Signal Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Signal Pharmaceuticals
Curated by ChEMBL
Signal Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Signal Pharmaceuticals
Curated by ChEMBL
Signal Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
TargetNuclear factor NF-kappa-B p105 subunit(Homo sapiens (Human))
Signal Pharmaceuticals
Curated by ChEMBL
Signal Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:In vitro inhibitory activity against human Jurkat T-Cells stably transfected with an Nuclear factor kappa B transcription factorMore data for this Ligand-Target Pair
TargetCyclic AMP-dependent transcription factor ATF-1(Homo sapiens (Human))
Signal Pharmaceuticals
Curated by ChEMBL
Signal Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:In vitro inhibitory activity against human Jurkat T-Cells stably transfected with activating transcription factor 1More data for this Ligand-Target Pair
TargetNuclear factor NF-kappa-B p105 subunit(Homo sapiens (Human))
Signal Pharmaceuticals
Curated by ChEMBL
Signal Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:In vitro inhibitory activity against human Jurkat T-Cells stably transfected with an Nuclear factor kappa B transcription factorMore data for this Ligand-Target Pair
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Signal Pharmaceuticals
Curated by ChEMBL
Signal Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Signal Pharmaceuticals
Curated by ChEMBL
Signal Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Signal Pharmaceuticals
Curated by ChEMBL
Signal Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Signal Pharmaceuticals
Curated by ChEMBL
Signal Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Signal Pharmaceuticals
Curated by ChEMBL
Signal Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
TargetProtein c-Fos/Transcription factor Jun(Homo sapiens (Human))
Signal Pharmaceuticals
Curated by ChEMBL
Signal Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
TargetCyclic AMP-dependent transcription factor ATF-1(Homo sapiens (Human))
Signal Pharmaceuticals
Curated by ChEMBL
Signal Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:In vitro inhibitory activity against human Jurkat T-Cells stably transfected with activating transcription factor 1More data for this Ligand-Target Pair
TargetNuclear factor NF-kappa-B p105 subunit(Homo sapiens (Human))
Signal Pharmaceuticals
Curated by ChEMBL
Signal Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:In vitro inhibitory activity against human Jurkat T-Cells stably transfected with an Nuclear factor kappa B transcription factorMore data for this Ligand-Target Pair