TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Instituto Universitario De Bio-OrgáNica Antonio GonzáLez
Curated by ChEMBL
Instituto Universitario De Bio-OrgáNica Antonio GonzáLez
Curated by ChEMBL
Affinity DataKi: 420nMAssay Description:Inhibition of human MDR1 overexpressed in mouse NIH/3T3 cells assessed as daunorubicin accumulation by flow cytometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Instituto Universitario De Bio-OrgáNica Antonio GonzáLez
Curated by ChEMBL
Instituto Universitario De Bio-OrgáNica Antonio GonzáLez
Curated by ChEMBL
Affinity DataKi: 510nMAssay Description:Inhibition of human MDR1 overexpressed in mouse NIH/3T3 cells assessed as daunorubicin accumulation by flow cytometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Instituto Universitario De Bio-OrgáNica Antonio GonzáLez
Curated by ChEMBL
Instituto Universitario De Bio-OrgáNica Antonio GonzáLez
Curated by ChEMBL
Affinity DataKi: 770nMAssay Description:Inhibition of human MDR1 overexpressed in mouse NIH/3T3 cells assessed as daunorubicin accumulation by flow cytometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Instituto Universitario De Bio-OrgáNica Antonio GonzáLez
Curated by ChEMBL
Instituto Universitario De Bio-OrgáNica Antonio GonzáLez
Curated by ChEMBL
Affinity DataKi: 1.01E+3nMAssay Description:Inhibition of human MDR1 overexpressed in mouse NIH/3T3 cells assessed as daunorubicin accumulation by flow cytometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Instituto Universitario De Bio-OrgáNica Antonio GonzáLez
Curated by ChEMBL
Instituto Universitario De Bio-OrgáNica Antonio GonzáLez
Curated by ChEMBL
Affinity DataKi: 1.04E+3nMAssay Description:Inhibition of human MDR1 overexpressed in mouse NIH/3T3 cells assessed as daunorubicin accumulation by flow cytometryMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Universidad Nacional Del Sur
Curated by ChEMBL
Universidad Nacional Del Sur
Curated by ChEMBL
Affinity DataKi: 1.44E+5nMAssay Description:Uncompetitive inhibition of Pacific electric ray AChE using acetylthiocholine as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of BChE in horse serum using butyrylthiocholine iodide as substrate after 120 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Universidad Nacional Del Sur
Curated by ChEMBL
Universidad Nacional Del Sur
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of Pacific electric ray AChE using acetylthiocholine iodide as substrate after 60 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibition of BChE in horse serum using butyrylthiocholine iodide as substrate after 120 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Universidad Nacional Del Sur
Curated by ChEMBL
Universidad Nacional Del Sur
Curated by ChEMBL
Affinity DataIC50: 29nMAssay Description:Inhibition of Pacific electric ray AChE using acetylthiocholine iodide as substrate after 60 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 2.15E+4nMAssay Description:Inhibition of BChE in horse serum using butyrylthiocholine iodide as substrate after 120 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member B1(Homo sapiens (Human))
Universidad De La Laguna
Curated by ChEMBL
Universidad De La Laguna
Curated by ChEMBL
Affinity DataIC50: 5.69E+4nMAssay Description:Inhibition of human recombinant aldose reductaseMore data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member B1(Homo sapiens (Human))
Universidad De La Laguna
Curated by ChEMBL
Universidad De La Laguna
Curated by ChEMBL
Affinity DataIC50: 5.69E+4nMAssay Description:Inhibition of human recombinant aldose reductaseMore data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member B1(Homo sapiens (Human))
Universidad De La Laguna
Curated by ChEMBL
Universidad De La Laguna
Curated by ChEMBL
Affinity DataIC50: 5.72E+4nMAssay Description:Inhibition of human recombinant aldose reductaseMore data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member B1(Homo sapiens (Human))
Universidad De La Laguna
Curated by ChEMBL
Universidad De La Laguna
Curated by ChEMBL
Affinity DataIC50: 5.75E+4nMAssay Description:Inhibition of human recombinant aldose reductaseMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Universidad Nacional Del Sur
Curated by ChEMBL
Universidad Nacional Del Sur
Curated by ChEMBL
Affinity DataIC50: 5.88E+4nMAssay Description:Inhibition of Pacific electric ray AChE using acetylthiocholine iodide as substrate after 60 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 6.43E+4nMAssay Description:Inhibition of BChE in horse serum using butyrylthiocholine iodide as substrate after 120 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 8.06E+4nMAssay Description:Inhibition of BChE in horse serum using butyrylthiocholine iodide as substrate after 120 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.04E+5nMAssay Description:Inhibition of BChE in horse serum using butyrylthiocholine iodide as substrate after 120 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.88E+5nMAssay Description:Inhibition of BChE in horse serum using butyrylthiocholine iodide as substrate after 120 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Universidad Nacional Del Sur
Curated by ChEMBL
Universidad Nacional Del Sur
Curated by ChEMBL
Affinity DataIC50: 1.90E+5nMAssay Description:Inhibition of Pacific electric ray AChE using acetylthiocholine iodide as substrate after 60 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of BChE in horse serum using butyrylthiocholine iodide as substrate after 120 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of BChE in horse serum using butyrylthiocholine iodide as substrate after 120 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of BChE in horse serum using butyrylthiocholine iodide as substrate after 120 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Universidad Nacional Del Sur
Curated by ChEMBL
Universidad Nacional Del Sur
Curated by ChEMBL
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of Pacific electric ray AChE using acetylthiocholine iodide as substrate after 60 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Universidad Nacional Del Sur
Curated by ChEMBL
Universidad Nacional Del Sur
Curated by ChEMBL
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of Pacific electric ray AChE using acetylthiocholine iodide as substrate after 60 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Universidad Nacional Del Sur
Curated by ChEMBL
Universidad Nacional Del Sur
Curated by ChEMBL
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of Pacific electric ray AChE using acetylthiocholine iodide as substrate after 60 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Universidad Nacional Del Sur
Curated by ChEMBL
Universidad Nacional Del Sur
Curated by ChEMBL
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of Pacific electric ray AChE using acetylthiocholine iodide as substrate after 60 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Universidad Nacional Del Sur
Curated by ChEMBL
Universidad Nacional Del Sur
Curated by ChEMBL
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of Pacific electric ray AChE using acetylthiocholine iodide as substrate after 60 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Universidad Nacional Del Sur
Curated by ChEMBL
Universidad Nacional Del Sur
Curated by ChEMBL
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of Pacific electric ray AChE using acetylthiocholine iodide as substrate after 60 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Universidad Nacional Del Sur
Curated by ChEMBL
Universidad Nacional Del Sur
Curated by ChEMBL
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of Pacific electric ray AChE using acetylthiocholine iodide as substrate after 60 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Universidad Nacional Del Sur
Curated by ChEMBL
Universidad Nacional Del Sur
Curated by ChEMBL
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of Pacific electric ray AChE using acetylthiocholine iodide as substrate after 60 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Universidad Nacional Del Sur
Curated by ChEMBL
Universidad Nacional Del Sur
Curated by ChEMBL
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of Pacific electric ray AChE using acetylthiocholine iodide as substrate after 60 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of BChE in horse serum using butyrylthiocholine iodide as substrate after 120 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of BChE in horse serum using butyrylthiocholine iodide as substrate after 120 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of BChE in horse serum using butyrylthiocholine iodide as substrate after 120 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Universidad Nacional Del Sur
Curated by ChEMBL
Universidad Nacional Del Sur
Curated by ChEMBL
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of Pacific electric ray AChE using acetylthiocholine iodide as substrate after 60 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member B1(Homo sapiens (Human))
Universidad De La Laguna
Curated by ChEMBL
Universidad De La Laguna
Curated by ChEMBL
Affinity DataIC50: 2.62E+7nMAssay Description:Inhibition of human recombinant aldose reductaseMore data for this Ligand-Target Pair