Affinity DataKi: 160nMAssay Description:Competitive inhibition of ATP binding to EGF-RMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibitory activity against S- adenosylmethionine decarboxylase (SAMDC) from rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibitory concentration of compound against S-Adenosylmethionine decarboxylase (SAMDC) from rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibitory concentration of compound against S-Adenosylmethionine decarboxylase (SAMDC) from rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against S- adenosylmethionine decarboxylase (SAMDC) from rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibitory activity against Rat liver ornithine decarboxylase(ODC)More data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Homo sapiens (Human))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibition of recombinant PDHK1 (unknown origin) expressed in Escherichia coli incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Homo sapiens (Human))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of recombinant PDHK1 (unknown origin) expressed in Escherichia coli incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Homo sapiens (Human))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Inhibition of recombinant PDHK1 (unknown origin) expressed in Escherichia coli incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Inhibitory activity against Rat liver ornithine decarboxylase(ODC)More data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Inhibitory activity against Rat liver ornithine decarboxylase(ODC)More data for this Ligand-Target Pair
Affinity DataIC50: 36nMAssay Description:Inhibitory concentration of compound against S-Adenosylmethionine decarboxylase (SAMDC) from rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 39nMAssay Description:Inhibitory activity against Rat liver ornithine decarboxylase(ODC)More data for this Ligand-Target Pair
Affinity DataIC50: 49nMAssay Description:Inhibitory activity against Rat liver ornithine decarboxylase(ODC)More data for this Ligand-Target Pair
Affinity DataIC50: 54nMAssay Description:Inhibition of the epidermal growth factor receptor expressed in A431 cell lineMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Homo sapiens (Human))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 59nMAssay Description:Inhibition of recombinant PDHK1 (unknown origin) expressed in Escherichia coli incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 61nMAssay Description:Inhibitory concentration of compound against S-Adenosylmethionine decarboxylase (SAMDC) from rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 66nMAssay Description:Inhibitory concentration of compound against S-Adenosylmethionine decarboxylase (SAMDC) from rat liverMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Homo sapiens (Human))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 68nMAssay Description:Inhibition of recombinant PDHK1 (unknown origin) expressed in Escherichia coli incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 84nMAssay Description:Inhibitory concentration of compound against S-Adenosylmethionine decarboxylase (SAMDC) from rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 88nMAssay Description:Inhibitory concentration of compound against S-Adenosylmethionine decarboxylase (SAMDC) from rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Inhibitory concentration of compound against S-Adenosylmethionine decarboxylase (SAMDC) from rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 92nMAssay Description:Inhibitory concentration of compound against S-Adenosylmethionine decarboxylase (SAMDC) from rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 93nMAssay Description:Inhibitory activity against Rat liver ornithine decarboxylase(ODC)More data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Inhibitory concentration of compound against S-Adenosylmethionine decarboxylase (SAMDC) from rat liverMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Homo sapiens (Human))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of recombinant PDHK1 (unknown origin) expressed in Escherichia coli incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Homo sapiens (Human))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Inhibition of recombinant PDHK1 (unknown origin) expressed in Escherichia coli incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Homo sapiens (Human))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibition of recombinant PDHK1 (unknown origin) expressed in Escherichia coli incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Inhibitory concentration of compound against S-Adenosylmethionine decarboxylase (SAMDC) from rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Inhibitory concentration of compound against S-Adenosylmethionine decarboxylase (SAMDC) from rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:In vitro inhibition of the Epidermal growth factor receptor activity in A431 membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 210nMAssay Description:Inhibitory concentration of compound against S-Adenosylmethionine decarboxylase (SAMDC) from rat liverMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Homo sapiens (Human))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 210nMAssay Description:Inhibition of recombinant PDHK1 (unknown origin) expressed in Escherichia coli incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 230nMAssay Description:In vitro inhibition of the Epidermal growth factor receptor activity in A431 membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 240nMAssay Description:Inhibitory concentration of compound against S-Adenosylmethionine decarboxylase (SAMDC) from rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:In vitro inhibition of the Epidermal growth factor receptor activity in A431 membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibitory activity against recombinant tyrosine kinase EGF-R (EGF-R ICD)More data for this Ligand-Target Pair
Affinity DataIC50: 310nMAssay Description:Inhibition of the epidermal growth factor receptor expressed in A431 cell lineMore data for this Ligand-Target Pair
Affinity DataIC50: 330nMAssay Description:Inhibitory concentration of compound against S-Adenosylmethionine decarboxylase (SAMDC) from rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 360nMAssay Description:In vitro inhibition of the Epidermal growth factor receptor activity in A431 membranesMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Homo sapiens (Human))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 380nMAssay Description:Inhibition of recombinant PDHK1 (unknown origin) expressed in Escherichia coli incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibition of the epidermal growth factor receptor expressed in A431 cell lineMore data for this Ligand-Target Pair
Affinity DataIC50: 470nMAssay Description:In vitro inhibition of the Epidermal growth factor receptor activity in A431 membranesMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Homo sapiens (Human))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 491nMAssay Description:Inhibition of recombinant PDHK1 (unknown origin) expressed in Escherichia coli incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition of the epidermal growth factor receptor expressed in A431 cell lineMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Homo sapiens (Human))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 521nMAssay Description:Inhibition of recombinant PDHK1 (unknown origin) expressed in Escherichia coli incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 530nMAssay Description:Inhibitory concentration of compound against S-Adenosylmethionine decarboxylase (SAMDC) from rat liverMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Homo sapiens (Human))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 557nMAssay Description:Inhibition of recombinant PDHK1 (unknown origin) expressed in Escherichia coli incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Homo sapiens (Human))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 580nMAssay Description:Inhibition of recombinant PDHK1 (unknown origin) expressed in Escherichia coli incubated for 1 hr by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Inhibition of the epidermal growth factor receptor expressed in A431 cell lineMore data for this Ligand-Target Pair