TargetGABA A receptor alpha-4/beta-3/gamma-2(Homo sapiens (Human))
University Of Utah
Curated by ChEMBL
University Of Utah
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Negative allosteric modulation activity at human GABAA alpha4beta3gamma2 stably expressed in HEK cells by patch clamp methodMore data for this Ligand-Target Pair
TargetGABA A receptor alpha-1/beta-1/gamma-2(Homo sapiens (Human))
University Of Utah
Curated by ChEMBL
University Of Utah
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Negative allosteric modulation activity at human GABAA alpha1beta1gamma2 stably expressed in HEK cells by whole cell patch clamp methodMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Roseman University Of Health Sciences
Curated by ChEMBL
Roseman University Of Health Sciences
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human recombinant FAAH using AMC arachidonoyl amide as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Roseman University Of Health Sciences
Curated by ChEMBL
Roseman University Of Health Sciences
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human recombinant COX2 assessed as inhibition of ADHP to fluorescent resorufin conversion by fluorescence assayMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-3/gamma-2(Homo sapiens (Human))
University Of Utah
Curated by ChEMBL
University Of Utah
Curated by ChEMBL
Affinity DataIC50: 5.50E+3nMAssay Description:Negative allosteric modulation activity at human GABAA alpha3beta3gamma2 stably expressed in HEK cells by whole cell patch clamp methodMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Roseman University Of Health Sciences
Curated by ChEMBL
Roseman University Of Health Sciences
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of human TRPV1 overexpressed in BEAS-2B cells assessed as calcium flux after 30 mins by Fluo-4 AM fluorescence assayMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Roseman University Of Health Sciences
Curated by ChEMBL
Roseman University Of Health Sciences
Curated by ChEMBL
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of human recombinant COX2 assessed as inhibition of ADHP to fluorescent resorufin conversion by fluorescence assayMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Roseman University Of Health Sciences
Curated by ChEMBL
Roseman University Of Health Sciences
Curated by ChEMBL
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of human recombinant COX2 assessed as inhibition of ADHP to fluorescent resorufin conversion by fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Roseman University Of Health Sciences
Curated by ChEMBL
Roseman University Of Health Sciences
Curated by ChEMBL
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of human TRPV1 overexpressed in BEAS-2B cells assessed as calcium flux after 30 mins by Fluo-4 AM fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Roseman University Of Health Sciences
Curated by ChEMBL
Roseman University Of Health Sciences
Curated by ChEMBL
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of human TRPV1 overexpressed in BEAS-2B cells assessed as calcium flux after 30 mins by Fluo-4 AM fluorescence assayMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Roseman University Of Health Sciences
Curated by ChEMBL
Roseman University Of Health Sciences
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant COX2 assessed as inhibition of ADHP to fluorescent resorufin conversion by fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Roseman University Of Health Sciences
Curated by ChEMBL
Roseman University Of Health Sciences
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human TRPV1 overexpressed in BEAS-2B cells assessed as calcium flux after 30 mins by Fluo-4 AM fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Roseman University Of Health Sciences
Curated by ChEMBL
Roseman University Of Health Sciences
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human TRPV1 overexpressed in BEAS-2B cells assessed as calcium flux after 30 mins by Fluo-4 AM fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Roseman University Of Health Sciences
Curated by ChEMBL
Roseman University Of Health Sciences
Curated by ChEMBL
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of human TRPV1 overexpressed in BEAS-2B cells assessed as calcium flux after 30 mins by Fluo-4 AM fluorescence assayMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Roseman University Of Health Sciences
Curated by ChEMBL
Roseman University Of Health Sciences
Curated by ChEMBL
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of human recombinant FAAH using AMC arachidonoyl amide as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetGABA-A receptor; alpha-2/beta-3/gamma-2(Homo sapiens (Human))
University Of Utah
Curated by ChEMBL
University Of Utah
Curated by ChEMBL
Affinity DataIC50: 1.57E+4nMAssay Description:Negative allosteric modulation activity at human GABAA alpha2beta3gamma2 stably expressed in HEK cells by whole cell patch clamp methodMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Roseman University Of Health Sciences
Curated by ChEMBL
Roseman University Of Health Sciences
Curated by ChEMBL
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of human recombinant FAAH using AMC arachidonoyl amide as substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Roseman University Of Health Sciences
Curated by ChEMBL
Roseman University Of Health Sciences
Curated by ChEMBL
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of human recombinant COX2 assessed as inhibition of ADHP to fluorescent resorufin conversion by fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Roseman University Of Health Sciences
Curated by ChEMBL
Roseman University Of Health Sciences
Curated by ChEMBL
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of human TRPV1 overexpressed in BEAS-2B cells assessed as calcium flux after 30 mins by Fluo-4 AM fluorescence assayMore data for this Ligand-Target Pair
TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Homo sapiens (Human))
University Of Utah
Curated by ChEMBL
University Of Utah
Curated by ChEMBL
Affinity DataIC50: 1.94E+4nMAssay Description:Negative allosteric modulation activity at human GABAA alpha5beta3gamma2 stably expressed in HEK cells by patch clamp methodMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Homo sapiens (Human))
University Of Utah
Curated by ChEMBL
University Of Utah
Curated by ChEMBL
Affinity DataIC50: 2.10E+4nMAssay Description:Negative allosteric modulation activity at human GABAA alpha1beta3gamma2 stably expressed in HEK cells by whole cell patch clamp methodMore data for this Ligand-Target Pair
Target InfoGoogleScholar
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Roseman University Of Health Sciences
Curated by ChEMBL
Roseman University Of Health Sciences
Curated by ChEMBL
Affinity DataIC50: 4.50E+4nMAssay Description:Inhibition of human TRPV1 overexpressed in BEAS-2B cells assessed as calcium flux after 30 mins by Fluo-4 AM fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Roseman University Of Health Sciences
Curated by ChEMBL
Roseman University Of Health Sciences
Curated by ChEMBL
Affinity DataIC50: 4.80E+4nMAssay Description:Inhibition of human TRPV1 overexpressed in BEAS-2B cells assessed as calcium flux after 30 mins by Fluo-4 AM fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Roseman University Of Health Sciences
Curated by ChEMBL
Roseman University Of Health Sciences
Curated by ChEMBL
Affinity DataIC50: 7.00E+4nMAssay Description:Inhibition of human TRPV1 overexpressed in BEAS-2B cells assessed as calcium flux after 30 mins by Fluo-4 AM fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Roseman University Of Health Sciences
Curated by ChEMBL
Roseman University Of Health Sciences
Curated by ChEMBL
Affinity DataIC50: 7.00E+4nMAssay Description:Inhibition of human TRPV1 overexpressed in BEAS-2B cells assessed as calcium flux after 30 mins by Fluo-4 AM fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Roseman University Of Health Sciences
Curated by ChEMBL
Roseman University Of Health Sciences
Curated by ChEMBL
Affinity DataIC50: 2.03E+5nMAssay Description:Inhibition of human TRPV1 overexpressed in BEAS-2B cells assessed as calcium flux after 30 mins by Fluo-4 AM fluorescence assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Mus musculus)
University Of Utah
Curated by ChEMBL
University Of Utah
Curated by ChEMBL
Affinity DataIC50: 2.27E+5nMAssay Description:Antagonist activity at TRPV1 channel in C57B1 mouse dorsal root ganglion cells assessed as inhibition of capsaicin-induced calcium flux by fluorometr...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Roseman University Of Health Sciences
Curated by ChEMBL
Roseman University Of Health Sciences
Curated by ChEMBL
Affinity DataIC50: 2.27E+5nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cell assessed as inhibition of capsaicin-induced calcium flux by fluorometric analysisMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Mus musculus)
University Of Utah
Curated by ChEMBL
University Of Utah
Curated by ChEMBL
Affinity DataIC50: 2.75E+5nMAssay Description:Antagonist activity at TRPV1 channel in C57B1 mouse dorsal root ganglion cells assessed as inhibition of capsaicin-induced calcium flux by fluorometr...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Roseman University Of Health Sciences
Curated by ChEMBL
Roseman University Of Health Sciences
Curated by ChEMBL
Affinity DataIC50: 2.75E+5nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cell assessed as inhibition of capsaicin-induced calcium flux by fluorometric analysisMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Mus musculus)
University Of Utah
Curated by ChEMBL
University Of Utah
Curated by ChEMBL
Affinity DataIC50: 1.32E+6nMAssay Description:Antagonist activity at TRPV1 channel in C57B1 mouse dorsal root ganglion cells assessed as inhibition of capsaicin-induced calcium flux by fluorometr...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Roseman University Of Health Sciences
Curated by ChEMBL
Roseman University Of Health Sciences
Curated by ChEMBL
Affinity DataIC50: 1.32E+6nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cell assessed as inhibition of capsaicin-induced calcium flux by fluorometric analysisMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Mus musculus)
University Of Utah
Curated by ChEMBL
University Of Utah
Curated by ChEMBL
Affinity DataIC50: 1.67E+6nMAssay Description:Antagonist activity at TRPV1 channel in C57B1 mouse dorsal root ganglion cells assessed as inhibition of capsaicin-induced calcium flux by fluorometr...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Roseman University Of Health Sciences
Curated by ChEMBL
Roseman University Of Health Sciences
Curated by ChEMBL
Affinity DataIC50: 1.67E+6nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cell assessed as inhibition of capsaicin-induced calcium flux by fluorometric analysisMore data for this Ligand-Target Pair