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Found 215 with Last Name = 'reister' and Initial = 'sm'
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173960((2S,4S)-1-((R)-2-amino-3-methyl-3-(pyridin-2-ylmet...)
Affinity DataKi:  12nMAssay Description:Inhibitory activity against human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173976((2S,4S)-1-((R)-2-amino-3-methyl-3-(pyridin-3-ylmet...)
Affinity DataKi:  18nMAssay Description:Inhibitory activity against human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173983((2S,4S)-1-((R)-2-amino-3-methyl-3-(3-phenylpropylt...)
Affinity DataKi:  24nMAssay Description:Inhibitory activity against human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173981((2S,4S)-1-((R)-3-(4-methoxybenzylthio)-2-amino-3-m...)
Affinity DataKi:  29nMAssay Description:Inhibitory activity against human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173958((2S,4S)-1-((R)-2-amino-3-methyl-3-(pyridin-4-ylmet...)
Affinity DataKi:  33nMAssay Description:Inhibitory activity against human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173967((2S,4S)-1-((R)-2-amino-3-((5-chlorobenzo[b]thiophe...)
Affinity DataKi:  40nMAssay Description:Inhibitory activity against human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173977((2S,4S)-1-((R)-2-amino-3-(3-(4-fluorophenyl)propyl...)
Affinity DataKi:  45nMAssay Description:Inhibitory activity against human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173971(CHEMBL427193 | N-(((R)-3-amino-4-((2S,4S)-2-cyano-...)
Affinity DataKi:  46nMAssay Description:Inhibitory activity against human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173963((2S,4S)-1-((R)-2-amino-3-(4-methoxybenzylsulfonyl)...)
Affinity DataKi:  53nMAssay Description:Inhibitory activity against human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173979((2S,4S)-1-((R)-2-amino-3-methyl-3-(phenethylthio)b...)
Affinity DataKi:  56nMAssay Description:Inhibitory activity against human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173972((2S,4S)-1-((R)-3-(4-(trifluoromethyl)benzylthio)-2...)
Affinity DataKi:  63nMAssay Description:Inhibitory activity against human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173961((2S,4S)-1-((R)-3-(3-phenoxybenzylthio)-2-amino-3-m...)
Affinity DataKi:  65nMAssay Description:Inhibitory activity against human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173978((2S,4S)-1-((R)-3-(4-cyanobenzylsulfonyl)-2-amino-3...)
Affinity DataKi:  68nMAssay Description:Inhibitory activity against human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173965((2S,4S)-1-((R)-3-(4-(methylsulfonyl)benzylsulfonyl...)
Affinity DataKi:  76nMAssay Description:Inhibitory activity against human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173957((2S,4S)-1-((R)-3-(4-methoxybenzylsulfinyl)-2-amino...)
Affinity DataKi:  112nMAssay Description:Inhibitory activity against human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173959((S)-1-((R)-3-(4-methoxybenzylsulfonyl)-2-amino-3-m...)
Affinity DataKi:  115nMAssay Description:Inhibitory activity against human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173968((R)-3-amino-4-((2S,4S)-2-cyano-4-fluoropyrrolidin-...)
Affinity DataKi:  154nMAssay Description:Inhibitory activity against human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173973(CHEMBL201053 | N-(4-(((R)-3-amino-4-((2S,4S)-2-cya...)
Affinity DataKi:  225nMAssay Description:Inhibitory activity against human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173964((2S,4S)-1-((R)-3-(4-fluorobenzylsulfonyl)-2-amino-...)
Affinity DataKi:  281nMAssay Description:Inhibitory activity against human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173962((2S,4S)-1-((R)-2-amino-3-methyl-3-(3-phenylpropyls...)
Affinity DataKi:  302nMAssay Description:Inhibitory activity against human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173975((2S,4S)-1-((R)-3-(2-methoxybenzylsulfonyl)-2-amino...)
Affinity DataKi:  309nMAssay Description:Inhibitory activity against human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173984((2S,4S)-1-((R)-3-(3-phenoxybenzylsulfonyl)-2-amino...)
Affinity DataKi:  310nMAssay Description:Inhibitory activity against human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173970((2S,4S)-1-((R)-3-(3-methoxybenzylsulfonyl)-2-amino...)
Affinity DataKi:  316nMAssay Description:Inhibitory activity against human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173966((2S,4S)-1-((R)-2-amino-3-(benzylsulfonyl)-3-methyl...)
Affinity DataKi:  324nMAssay Description:Inhibitory activity against human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173969((2S,4S)-1-((R)-3-(4-(benzyloxy)benzylsulfonyl)-2-a...)
Affinity DataKi:  428nMAssay Description:Inhibitory activity against human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173983((2S,4S)-1-((R)-2-amino-3-methyl-3-(3-phenylpropylt...)
Affinity DataKi:  523nMAssay Description:Inhibitory activity against recombinant DPP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173974((2S,4S)-1-((R)-2-amino-3-methyl-3-p-tolylmethanesu...)
Affinity DataKi:  530nMAssay Description:Inhibitory activity against human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173980((2S,4S)-1-[(R)-2-amino-3-(biphenyl-4-ylmethanesulf...)
Affinity DataKi:  579nMAssay Description:Inhibitory activity against human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173977((2S,4S)-1-((R)-2-amino-3-(3-(4-fluorophenyl)propyl...)
Affinity DataKi:  701nMAssay Description:Inhibitory activity against recombinant DPP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173961((2S,4S)-1-((R)-3-(3-phenoxybenzylthio)-2-amino-3-m...)
Affinity DataKi:  1.07E+3nMAssay Description:Inhibitory activity against recombinant DPP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173972((2S,4S)-1-((R)-3-(4-(trifluoromethyl)benzylthio)-2...)
Affinity DataKi:  1.13E+3nMAssay Description:Inhibitory activity against recombinant DPP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173971(CHEMBL427193 | N-(((R)-3-amino-4-((2S,4S)-2-cyano-...)
Affinity DataKi:  1.28E+3nMAssay Description:Inhibitory activity against recombinant sepraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173982((2S,4S)-1-((R)-2-amino-3-methyl-3-(pyridin-4-ylmet...)
Affinity DataKi:  1.28E+3nMAssay Description:Inhibitory activity against human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173981((2S,4S)-1-((R)-3-(4-methoxybenzylthio)-2-amino-3-m...)
Affinity DataKi:  3.95E+3nMAssay Description:Inhibitory activity against recombinant DPP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173967((2S,4S)-1-((R)-2-amino-3-((5-chlorobenzo[b]thiophe...)
Affinity DataKi:  5.16E+3nMAssay Description:Inhibitory activity against recombinant sepraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173984((2S,4S)-1-((R)-3-(3-phenoxybenzylsulfonyl)-2-amino...)
Affinity DataKi:  6.86E+3nMAssay Description:Inhibitory activity against recombinant sepraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173973(CHEMBL201053 | N-(4-(((R)-3-amino-4-((2S,4S)-2-cya...)
Affinity DataKi:  7.93E+3nMAssay Description:Inhibitory activity against recombinant sepraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173978((2S,4S)-1-((R)-3-(4-cyanobenzylsulfonyl)-2-amino-3...)
Affinity DataKi:  9.45E+3nMAssay Description:Inhibitory activity against recombinant sepraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173980((2S,4S)-1-[(R)-2-amino-3-(biphenyl-4-ylmethanesulf...)
Affinity DataKi:  9.66E+3nMAssay Description:Inhibitory activity against recombinant sepraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173958((2S,4S)-1-((R)-2-amino-3-methyl-3-(pyridin-4-ylmet...)
Affinity DataKi:  9.66E+3nMAssay Description:Inhibitory activity against recombinant sepraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173983((2S,4S)-1-((R)-2-amino-3-methyl-3-(3-phenylpropylt...)
Affinity DataKi:  1.22E+4nMAssay Description:Inhibitory activity against recombinant sepraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173975((2S,4S)-1-((R)-3-(2-methoxybenzylsulfonyl)-2-amino...)
Affinity DataKi:  1.24E+4nMAssay Description:Inhibitory activity against recombinant sepraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173961((2S,4S)-1-((R)-3-(3-phenoxybenzylthio)-2-amino-3-m...)
Affinity DataKi:  1.28E+4nMAssay Description:Inhibitory activity against recombinant sepraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173979((2S,4S)-1-((R)-2-amino-3-methyl-3-(phenethylthio)b...)
Affinity DataKi:  1.44E+4nMAssay Description:Inhibitory activity against recombinant DPP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173968((R)-3-amino-4-((2S,4S)-2-cyano-4-fluoropyrrolidin-...)
Affinity DataKi:  1.46E+4nMAssay Description:Inhibitory activity against recombinant sepraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173977((2S,4S)-1-((R)-2-amino-3-(3-(4-fluorophenyl)propyl...)
Affinity DataKi:  1.58E+4nMAssay Description:Inhibitory activity against recombinant sepraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173970((2S,4S)-1-((R)-3-(3-methoxybenzylsulfonyl)-2-amino...)
Affinity DataKi:  1.70E+4nMAssay Description:Inhibitory activity against recombinant sepraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173965((2S,4S)-1-((R)-3-(4-(methylsulfonyl)benzylsulfonyl...)
Affinity DataKi:  1.73E+4nMAssay Description:Inhibitory activity against recombinant DPP2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173960((2S,4S)-1-((R)-2-amino-3-methyl-3-(pyridin-2-ylmet...)
Affinity DataKi:  1.91E+4nMAssay Description:Inhibitory activity against recombinant sepraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50173969((2S,4S)-1-((R)-3-(4-(benzyloxy)benzylsulfonyl)-2-a...)
Affinity DataKi:  2.04E+4nMAssay Description:Inhibitory activity against recombinant sepraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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