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Found 26 with Last Name = 'ritschel' and Initial = 't'
TargetQueuine tRNA-ribosyltransferase(Zymomonas mobilis)
Philipps-UniversitÄT Marburg

LigandPNGBDBM84658(lin-benzoguanine scaffold, 7)
Affinity DataKi:  3.5nMpH: 7.3Assay Description:Inhibition assay using tRNA-guanine transglycosylase (TGT).More data for this Ligand-Target Pair
TargetQueuine tRNA-ribosyltransferase(Zymomonas mobilis)
Philipps-UniversitÄT Marburg

LigandPNGBDBM84659(lin-benzoguanine scaffold, 8)
Affinity DataKi:  5.5nMpH: 7.3Assay Description:Inhibition assay using tRNA-guanine transglycosylase (TGT).More data for this Ligand-Target Pair
Ligand InfoMMDBPC cidPC sid
In DepthDetails ArticlePubMedMMDB

TargetQueuine tRNA-ribosyltransferase(Zymomonas mobilis)
Philipps-UniversitÄT Marburg

LigandPNGBDBM84657(lin-benzoguanine scaffold, 6)
Affinity DataKi:  5.80nMpH: 7.3Assay Description:Inhibition assay using tRNA-guanine transglycosylase (TGT).More data for this Ligand-Target Pair
TargetQueuine tRNA-ribosyltransferase(Zymomonas mobilis)
Philipps-UniversitÄT Marburg

LigandPNGBDBM84660(lin-benzoguanine scaffold, 9)
Affinity DataKi:  6nMpH: 7.3Assay Description:Inhibition assay using tRNA-guanine transglycosylase (TGT).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetQueuine tRNA-ribosyltransferase(Zymomonas mobilis)
Philipps-UniversitÄT Marburg

LigandPNGBDBM84661(lin-benzoguanine scaffold, 10)
Affinity DataKi:  10nMpH: 7.3Assay Description:Inhibition assay using tRNA-guanine transglycosylase (TGT).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetQueuine tRNA-ribosyltransferase(Zymomonas mobilis)
Philipps-UniversitÄT Marburg

LigandPNGBDBM84656(lin-benzoguanine scaffold, 5)
Affinity DataKi:  77nMpH: 7.3Assay Description:Inhibition assay using tRNA-guanine transglycosylase (TGT).More data for this Ligand-Target Pair
TargetQueuine tRNA-ribosyltransferase(Zymomonas mobilis)
Philipps-UniversitÄT Marburg

LigandPNGBDBM84655(lin-benzoguanine scaffold, 4)
Affinity DataKi:  1.50E+3nMpH: 7.3Assay Description:Inhibition assay using tRNA-guanine transglycosylase (TGT).More data for this Ligand-Target Pair
TargetQueuine tRNA-ribosyltransferase(Zymomonas mobilis)
Philipps-UniversitÄT Marburg

LigandPNGBDBM84654(lin-benzoguanine scaffold, 3)
Affinity DataKi:  4.10E+3nMpH: 7.3Assay Description:Inhibition assay using tRNA-guanine transglycosylase (TGT).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetQueuine tRNA-ribosyltransferase(Zymomonas mobilis)
Philipps-UniversitÄT Marburg

LigandPNGBDBM84653(Quinazolinone scaffold, 2)
Affinity DataKi:  7.60E+3nMpH: 7.3Assay Description:Inhibition assay using tRNA-guanine transglycosylase (TGT).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetQueuine tRNA-ribosyltransferase(Zymomonas mobilis)
Philipps-UniversitÄT Marburg

LigandPNGBDBM84652(Quinazolinone scaffold, 1)
Affinity DataKi:  3.10E+4nMpH: 7.3Assay Description:Inhibition assay using tRNA-guanine transglycosylase (TGT).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPapain(Carica papaya)
Radboud University Nijmegen

Curated by ChEMBL
LigandPNGBDBM20120((2S)-N-(cyanomethyl)-3-phenyl-2-[(4-phenylphenyl)f...)
Affinity DataIC50:  220nMAssay Description:Inhibition of papaya papain using Z-Phe-Arg-pNA substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPapain(Carica papaya)
Radboud University Nijmegen

Curated by ChEMBL
LigandPNGBDBM50048077(CHEMBL3357470)
Affinity DataIC50:  270nMAssay Description:Inhibition of papaya papain using Z-Phe-Arg-pNA substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPapain(Carica papaya)
Radboud University Nijmegen

Curated by ChEMBL
LigandPNGBDBM50048079(CHEMBL3357955)
Affinity DataIC50:  280nMAssay Description:Inhibition of papaya papain using Z-Phe-Arg-pNA substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPapain(Carica papaya)
Radboud University Nijmegen

Curated by ChEMBL
LigandPNGBDBM50048070(CHEMBL3357964)
Affinity DataIC50:  350nMAssay Description:Inhibition of papaya papain using Z-Phe-Arg-pNA substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPapain(Carica papaya)
Radboud University Nijmegen

Curated by ChEMBL
LigandPNGBDBM20119((2S)-N-(cyanomethyl)-3-phenyl-2-(phenylformamido)p...)
Affinity DataIC50:  360nMAssay Description:Inhibition of papaya papain using Z-Phe-Arg-pNA substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPapain(Carica papaya)
Radboud University Nijmegen

Curated by ChEMBL
LigandPNGBDBM50048080(CHEMBL3357956)
Affinity DataIC50:  710nMAssay Description:Inhibition of papaya papain using Z-Phe-Arg-pNA substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPapain(Carica papaya)
Radboud University Nijmegen

Curated by ChEMBL
LigandPNGBDBM50048081(CHEMBL3357957)
Affinity DataIC50:  980nMAssay Description:Inhibition of papaya papain using Z-Phe-Arg-pNA substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPapain(Carica papaya)
Radboud University Nijmegen

Curated by ChEMBL
LigandPNGBDBM50048082(CHEMBL3357958)
Affinity DataIC50:  1.58E+3nMAssay Description:Inhibition of papaya papain using Z-Phe-Arg-pNA substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPapain(Carica papaya)
Radboud University Nijmegen

Curated by ChEMBL
LigandPNGBDBM50048072(CHEMBL3357962)
Affinity DataIC50:  2.25E+3nMAssay Description:Inhibition of papaya papain using Z-Phe-Arg-pNA substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPapain(Carica papaya)
Radboud University Nijmegen

Curated by ChEMBL
LigandPNGBDBM50048074(CHEMBL3357468)
Affinity DataIC50:  2.27E+3nMAssay Description:Inhibition of papaya papain using Z-Phe-Arg-pNA substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPapain(Carica papaya)
Radboud University Nijmegen

Curated by ChEMBL
LigandPNGBDBM50048068(CHEMBL3357961)
Affinity DataIC50:  2.71E+3nMAssay Description:Inhibition of papaya papain using Z-Phe-Arg-pNA substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPapain(Carica papaya)
Radboud University Nijmegen

Curated by ChEMBL
LigandPNGBDBM50048073(CHEMBL3357963)
Affinity DataIC50:  3.97E+3nMAssay Description:Inhibition of papaya papain using Z-Phe-Arg-pNA substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPapain(Carica papaya)
Radboud University Nijmegen

Curated by ChEMBL
LigandPNGBDBM50048071(CHEMBL3357965)
Affinity DataIC50:  5.98E+3nMAssay Description:Inhibition of papaya papain using Z-Phe-Arg-pNA substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPapain(Carica papaya)
Radboud University Nijmegen

Curated by ChEMBL
LigandPNGBDBM50048075(CHEMBL3357469)
Affinity DataIC50:  7.10E+3nMAssay Description:Inhibition of papaya papain using Z-Phe-Arg-pNA substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPapain(Carica papaya)
Radboud University Nijmegen

Curated by ChEMBL
LigandPNGBDBM50048083(CHEMBL3357959)
Affinity DataIC50:  1.39E+4nMAssay Description:Inhibition of papaya papain using Z-Phe-Arg-pNA substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPapain(Carica papaya)
Radboud University Nijmegen

Curated by ChEMBL
LigandPNGBDBM50048067(CHEMBL3357960)
Affinity DataIC50:  5.12E+4nMAssay Description:Inhibition of papaya papain using Z-Phe-Arg-pNA substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed