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Found 245 with Last Name = 'russo' and Initial = 'a'
TargetAcylamino-acid-releasing enzyme(Sus scrofa)
Istituto Di Biostrutture E Bioimmagini

Curated by ChEMBL
LigandPNGBDBM50382729(CHEMBL2023560)
Affinity DataKi:  2.40E+4nMAssay Description:Inhibition of pig APEH using acetyl-Ala-pNA as substrate incubated for 2 mins prior to substrate addition by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50005305((SCRIP)3-[2-(2-tert-Butoxycarbonylamino-3-phenyl-p...)
Affinity DataIC50:  8nMAssay Description:Inhibition of human recombinant reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50005305((SCRIP)3-[2-(2-tert-Butoxycarbonylamino-3-phenyl-p...)
Affinity DataIC50:  8nMAssay Description:Inhibition of human recombinant reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50005306(4-Cyclohexyl-2-hydroxy-3-{2-[2-(1-oxo-1,3-dihydro-...)
Affinity DataIC50:  8.90nMAssay Description:Inhibition of human recombinant reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50005301(4-Cyclohexyl-2-hydroxy-3-{2-[2-(1-oxo-1,3-dihydro-...)
Affinity DataIC50:  16nMAssay Description:Inhibition of human recombinant reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 9(Homo sapiens (Human))
Universita` Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)
Affinity DataIC50:  20nMAssay Description:Inhibition of human HDAC9 using ArgHisLysLys(Ac) fluorogenic peptide as a substrate by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50005311(4-Cyclohexyl-2-hydroxy-3-{4-methyl-2-[2-(1-oxo-1,3...)
Affinity DataIC50:  23nMAssay Description:Inhibition of human recombinant reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50005309(4-Cyclohexyl-2-hydroxy-3-{4-methyl-2-[2-(1-oxo-1,3...)
Affinity DataIC50:  36nMAssay Description:Inhibition of human recombinant reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Universita` Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)
Affinity DataIC50:  61nMAssay Description:Inhibition of human HDAC1 using ArgHisLysLys(Ac) fluorogenic peptide as a substrate by fluorimetric assayMore data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50005308(4-Cyclohexyl-2-hydroxy-3-{4-methyl-2-[2-(1-oxo-1H,...)
Affinity DataIC50:  80nMAssay Description:Inhibition of human recombinant reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 11(Homo sapiens (Human))
Universita` Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)
Affinity DataIC50:  100nMAssay Description:Inhibition of human HDAC11 using ArgHisLysLys(Ac) fluorogenic peptide as a substrate by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Universita` Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)
Affinity DataIC50:  100nMAssay Description:Inhibition of human HDAC6 using ArgHisLysLys(Ac) fluorogenic peptide as a substrate by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetRenin(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50005303(4-Cyclohexyl-2-hydroxy-3-{4-methyl-2-[2-(5-oxo-7H-...)
Affinity DataIC50:  100nMAssay Description:Inhibition of human recombinant reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50005302(4-Cyclohexyl-2-hydroxy-3-{4-methyl-2-[2-(3-oxo-tet...)
Affinity DataIC50:  141nMAssay Description:Inhibition of human recombinant reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyamine deacetylase HDAC10(Homo sapiens (Human))
Universita` Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)
Affinity DataIC50:  150nMAssay Description:Inhibition of human HDAC10 using ArgHisLysLys(Ac) fluorogenic peptide as a substrate by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 5(Homo sapiens (Human))
Universita` Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)
Affinity DataIC50:  150nMAssay Description:Inhibition of human HDAC5 using ArgHisLysLys(Ac) fluorogenic peptide as a substrate by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50005307(4-Cyclohexyl-2-hydroxy-3-{4-methyl-2-[2-(2-oxo-pyr...)
Affinity DataIC50:  157nMAssay Description:Inhibition of human recombinant reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Universita` Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)
Affinity DataIC50:  180nMAssay Description:Inhibition of human HDAC8 using ArgHisLysLys(Ac) fluorogenic peptide as a substrate by fluorimetric assayMore data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50005300(4-Cyclohexyl-2-hydroxy-3-{3-(1H-imidazol-4-yl)-2-[...)
Affinity DataIC50:  186nMAssay Description:Inhibition of human recombinant reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50005304(4-Cyclohexyl-2-hydroxy-3-{4-methyl-2-[2-(5-oxo-5,7...)
Affinity DataIC50:  207nMAssay Description:Inhibition of human recombinant reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Universita` Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)
Affinity DataIC50:  210nMAssay Description:Inhibition of human HDAC4 using ArgHisLysLys(Ac) fluorogenic peptide as a substrate by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Universita` Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)
Affinity DataIC50:  240nMAssay Description:Inhibition of human HDAC2 using ArgHisLysLys(Ac) fluorogenic peptide as a substrate by fluorimetric assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 3(Homo sapiens (Human))
Universita` Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)
Affinity DataIC50:  250nMAssay Description:Inhibition of human HDAC3 using ArgHisLysLys(Ac) fluorogenic peptide as a substrate by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetRenin(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50005310(4-Cyclohexyl-3-{2-[2-(1,3-dioxo-1H,3H-benzo[de]iso...)
Affinity DataIC50:  391nMAssay Description:Inhibition of human recombinant reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 6B(Homo sapiens (Human))
Institute Of Biomolecular Chemistry (Icb)

Curated by ChEMBL
LigandPNGBDBM50535443(CHEMBL4591907)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of recombinant human JMJD3 expressed in baculovirus infected Sf9 cells using biotinylated histone H3 peptide as substrate incubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Universita` Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50341839(5-(3-Aminophenyl)-N-(7-(hydroxyimino)-8-(methylami...)
Affinity DataIC50:  1.88E+3nMAssay Description:Inhibition of human HDAC3 using ArgHisLysLys(Ac) fluorogenic peptide as a substrate by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Universita` Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50341854(CHEMBL1767039 | N9-(3-(6-Chloropyridin-3-yl)phenyl...)
Affinity DataIC50:  1.99E+3nMAssay Description:Inhibition of human HDAC3 using ArgHisLysLys(Ac) fluorogenic peptide as a substrate by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 7(Homo sapiens (Human))
Universita` Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)
Affinity DataIC50:  2.48E+3nMAssay Description:Inhibition of human HDAC7 using ArgHisLysLys(Ac) fluorogenic peptide as a substrate by fluorimetric assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 9(Homo sapiens (Human))
Universita` Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50341839(5-(3-Aminophenyl)-N-(7-(hydroxyimino)-8-(methylami...)
Affinity DataIC50:  2.55E+3nMAssay Description:Inhibition of human HDAC9 using ArgHisLysLys(Ac) fluorogenic peptide as a substrate by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Universita` Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50341840(5-(4-Aminophenyl)-N-(7-(hydroxyimino)-8-(methylami...)
Affinity DataIC50:  4.44E+3nMAssay Description:Inhibition of human HDAC3 using ArgHisLysLys(Ac) fluorogenic peptide as a substrate by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 7(Homo sapiens (Human))
Universita` Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50341839(5-(3-Aminophenyl)-N-(7-(hydroxyimino)-8-(methylami...)
Affinity DataIC50:  5.25E+3nMAssay Description:Inhibition of human HDAC7 using ArgHisLysLys(Ac) fluorogenic peptide as a substrate by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 9(Homo sapiens (Human))
Universita` Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50341840(5-(4-Aminophenyl)-N-(7-(hydroxyimino)-8-(methylami...)
Affinity DataIC50:  6.50E+3nMAssay Description:Inhibition of human HDAC9 using ArgHisLysLys(Ac) fluorogenic peptide as a substrate by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Universita` Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50341839(5-(3-Aminophenyl)-N-(7-(hydroxyimino)-8-(methylami...)
Affinity DataIC50:  8.12E+3nMAssay Description:Inhibition of human HDAC1 using ArgHisLysLys(Ac) fluorogenic peptide as a substrate by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Universita` Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50341851(CHEMBL1767036 | N9-([1,1'-Biphenyl]-3-yl)-2-(hydro...)
Affinity DataIC50:  9.60E+3nMAssay Description:Inhibition of human HDAC3 using ArgHisLysLys(Ac) fluorogenic peptide as a substrate by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Universita` Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50341842((S)-2-(Hydroxyimino)-8-((4-methoxybenzyl)amino)-N1...)
Affinity DataIC50:  1.06E+4nMAssay Description:Inhibition of human HDAC3 using ArgHisLysLys(Ac) fluorogenic peptide as a substrate by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Universita` Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50341840(5-(4-Aminophenyl)-N-(7-(hydroxyimino)-8-(methylami...)
Affinity DataIC50:  1.16E+4nMAssay Description:Inhibition of human HDAC1 using ArgHisLysLys(Ac) fluorogenic peptide as a substrate by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 5(Homo sapiens (Human))
Universita` Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50341839(5-(3-Aminophenyl)-N-(7-(hydroxyimino)-8-(methylami...)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of human HDAC5 using ArgHisLysLys(Ac) fluorogenic peptide as a substrate by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 9(Homo sapiens (Human))
Universita` Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50341854(CHEMBL1767039 | N9-(3-(6-Chloropyridin-3-yl)phenyl...)
Affinity DataIC50:  1.33E+4nMAssay Description:Inhibition of human HDAC9 using ArgHisLysLys(Ac) fluorogenic peptide as a substrate by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 5(Homo sapiens (Human))
Universita` Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50341840(5-(4-Aminophenyl)-N-(7-(hydroxyimino)-8-(methylami...)
Affinity DataIC50:  1.53E+4nMAssay Description:Inhibition of human HDAC5 using ArgHisLysLys(Ac) fluorogenic peptide as a substrate by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyamine deacetylase HDAC10(Homo sapiens (Human))
Universita` Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50341839(5-(3-Aminophenyl)-N-(7-(hydroxyimino)-8-(methylami...)
Affinity DataIC50:  1.54E+4nMAssay Description:Inhibition of human HDAC10 using ArgHisLysLys(Ac) fluorogenic peptide as a substrate by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 7(Homo sapiens (Human))
Universita` Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50341840(5-(4-Aminophenyl)-N-(7-(hydroxyimino)-8-(methylami...)
Affinity DataIC50:  1.65E+4nMAssay Description:Inhibition of human HDAC7 using ArgHisLysLys(Ac) fluorogenic peptide as a substrate by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 11(Homo sapiens (Human))
Universita` Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50341839(5-(3-Aminophenyl)-N-(7-(hydroxyimino)-8-(methylami...)
Affinity DataIC50:  1.68E+4nMAssay Description:Inhibition of human HDAC11 using ArgHisLysLys(Ac) fluorogenic peptide as a substrate by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Universita` Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50341842((S)-2-(Hydroxyimino)-8-((4-methoxybenzyl)amino)-N1...)
Affinity DataIC50:  1.75E+4nMAssay Description:Inhibition of human HDAC1 using ArgHisLysLys(Ac) fluorogenic peptide as a substrate by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Universita` Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50341853(2-(Hydroxyimino)-N1-methyl-N9-(3-(pyridine-3-yl)ph...)
Affinity DataIC50:  1.84E+4nMAssay Description:Inhibition of human HDAC3 using ArgHisLysLys(Ac) fluorogenic peptide as a substrate by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Universita` Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50341844(2-(Hydroxyimino)-N1-methyl-N9-phenylnonanediamide ...)
Affinity DataIC50:  1.86E+4nMAssay Description:Inhibition of human HDAC3 using ArgHisLysLys(Ac) fluorogenic peptide as a substrate by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Universita` Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50341854(CHEMBL1767039 | N9-(3-(6-Chloropyridin-3-yl)phenyl...)
Affinity DataIC50:  1.93E+4nMAssay Description:Inhibition of human HDAC1 using ArgHisLysLys(Ac) fluorogenic peptide as a substrate by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 9(Homo sapiens (Human))
Universita` Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50341851(CHEMBL1767036 | N9-([1,1'-Biphenyl]-3-yl)-2-(hydro...)
Affinity DataIC50:  1.94E+4nMAssay Description:Inhibition of human HDAC9 using ArgHisLysLys(Ac) fluorogenic peptide as a substrate by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 5(Homo sapiens (Human))
Universita` Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50341854(CHEMBL1767039 | N9-(3-(6-Chloropyridin-3-yl)phenyl...)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of human HDAC5 using ArgHisLysLys(Ac) fluorogenic peptide as a substrate by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Universita` Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50341852(3'-(8-(Hydroxyimino)-9-(methylamino)-9-oxononanami...)
Affinity DataIC50:  2.11E+4nMAssay Description:Inhibition of human HDAC3 using ArgHisLysLys(Ac) fluorogenic peptide as a substrate by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyamine deacetylase HDAC10(Homo sapiens (Human))
Universita` Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50341840(5-(4-Aminophenyl)-N-(7-(hydroxyimino)-8-(methylami...)
Affinity DataIC50:  2.18E+4nMAssay Description:Inhibition of human HDAC10 using ArgHisLysLys(Ac) fluorogenic peptide as a substrate by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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