Affinity DataKi: 12nMAssay Description:The compound was tested in vivo for inhibition of gastric proton-pump enzyme H+/K+ ATPaseMore data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:Inhibitory activity against dog gastric proton-pump enzyme H+/K+ ATPaseMore data for this Ligand-Target Pair
Affinity DataKi: 290nM ΔG°: -37.6kJ/molepH: 6.8 T: 2°CAssay Description:The assay was performed as previously described with slight modifications [Chen et al., J. Agric. Food Chem., 50:4108-12]. The reaction medium was 1 ...More data for this Ligand-Target Pair
Affinity DataKi: 640nM ΔG°: -35.6kJ/molepH: 6.8 T: 2°CAssay Description:The assay was performed as previously described with slight modifications [Chen et al., J. Agric. Food Chem., 50:4108-12]. The reaction medium was 1 ...More data for this Ligand-Target Pair
Affinity DataKi: 950nM ΔG°: -35.8kJ/molepH: 6.8 T: 2°CAssay Description:The assay was performed as previously described with slight modifications [Chen et al., J. Agric. Food Chem., 50:4108-12]. The reaction medium was 1 ...More data for this Ligand-Target Pair
Affinity DataKi: 1.05E+3nM ΔG°: -35.5kJ/molepH: 6.8 T: 2°CAssay Description:The assay was performed as previously described with slight modifications [Chen et al., J. Agric. Food Chem., 50:4108-12]. The reaction medium was 1 ...More data for this Ligand-Target Pair
Affinity DataKi: 5.70E+3nM ΔG°: -31.1kJ/molepH: 6.8 T: 2°CAssay Description:The assay was performed as previously described with slight modifications [Chen et al., J. Agric. Food Chem., 50:4108-12]. The reaction medium was 1 ...More data for this Ligand-Target Pair
Affinity DataKi: 5.90E+3nM ΔG°: -31.0kJ/molepH: 6.8 T: 2°CAssay Description:The assay was performed as previously described with slight modifications [Chen et al., J. Agric. Food Chem., 50:4108-12]. The reaction medium was 1 ...More data for this Ligand-Target Pair
Affinity DataKi: 6.10E+3nM ΔG°: -29.3kJ/molepH: 6.8 T: 2°CAssay Description:Kinetic assay of catecholase and cresolase activities was carried out through depletion of MeBACat and MePAPh for 1 or 2 min with enzyme concentratio...More data for this Ligand-Target Pair
Affinity DataKi: 7.20E+3nM ΔG°: -28.9kJ/molepH: 6.8 T: 2°CAssay Description:Kinetic assay of catecholase and cresolase activities was carried out through depletion of MeBACat and MePAPh for 1 or 2 min with enzyme concentratio...More data for this Ligand-Target Pair
Affinity DataKi: 9.40E+3nM ΔG°: -28.9kJ/molepH: 6.8 T: 2°CAssay Description:The assay was performed as previously described with slight modifications [Chen et al., J. Agric. Food Chem., 50:4108-12]. The reaction medium was 1 ...More data for this Ligand-Target Pair
Affinity DataKi: 9.80E+3nM ΔG°: -28.1kJ/molepH: 6.8 T: 2°CAssay Description:Kinetic assay of catecholase and cresolase activities was carried out through depletion of MeBACat and MePAPh for 1 or 2 min with enzyme concentratio...More data for this Ligand-Target Pair
Affinity DataKi: 1.29E+4nM ΔG°: -27.4kJ/molepH: 6.8 T: 2°CAssay Description:Kinetic assay of catecholase and cresolase activities was carried out through depletion of MeBACat and MePAPh for 1 or 2 min with enzyme concentratio...More data for this Ligand-Target Pair
Affinity DataKi: 1.41E+4nM ΔG°: -27.9kJ/molepH: 6.8 T: 2°CAssay Description:The assay was performed as previously described with slight modifications [Chen et al., J. Agric. Food Chem., 50:4108-12]. The reaction medium was 1 ...More data for this Ligand-Target Pair
Affinity DataKi: 2.18E+4nM ΔG°: -26.2kJ/molepH: 6.8 T: 2°CAssay Description:Kinetic assay of catecholase and cresolase activities was carried out through depletion of MeBACat and MePAPh for 1 or 2 min with enzyme concentratio...More data for this Ligand-Target Pair
Affinity DataKi: 4.22E+4nM ΔG°: -24.6kJ/molepH: 6.8 T: 2°CAssay Description:Kinetic assay of catecholase and cresolase activities was carried out through depletion of MeBACat and MePAPh for 1 or 2 min with enzyme concentratio...More data for this Ligand-Target Pair
Affinity DataKi: 5.75E+4nMAssay Description:Inhibitory activity against dog gastric proton-pump enzyme H+/K+ ATPaseMore data for this Ligand-Target Pair
Affinity DataKi: 5.78E+4nMAssay Description:Inhibitory activity against dog gastric proton-pump enzyme H+/K+ ATPaseMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Inhibitory activity against dog gastric proton-pump enzyme H+/K+ ATPaseMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Inhibitory activity against dog gastric proton-pump enzyme H+/K+ ATPaseMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Inhibitory activity of gastric proton-pump enzyme H+/K+ ATPase was determined at 50 uMMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Inhibitory activity against dog gastric proton-pump enzyme H+/K+ ATPaseMore data for this Ligand-Target Pair