Compile Data Set for Download or QSAR
maximum 50k data
Found 53 with Last Name = 'sadler' and Initial = 'tm'
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319739(3,3-dimethyl-N-(4-(2-(4-sulfamoylphenylamino)pyrim...)
Affinity DataIC50:  10nMAssay Description:Inhibition of FLAG-tagged IKKbeta after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50303035(4-(4-(5-methylthiophen-2-yl)pyrimidin-2-ylamino)be...)
Affinity DataIC50:  19nMAssay Description:Inhibition of FLAG-tagged IKKbeta after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319743(CHEMBL1085122 | N-(4-(2-(4-sulfamoylphenylamino)py...)
Affinity DataIC50:  20nMAssay Description:Inhibition of FLAG-tagged IKKbeta after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319737(4-(4-(4-methoxyphenyl)pyrimidin-2-ylamino)benzenes...)
Affinity DataIC50:  40nMAssay Description:Inhibition of FLAG-tagged IKKbeta after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319741(2-phenyl-N-(4-(2-(4-sulfamoylphenylamino)pyrimidin...)
Affinity DataIC50:  50nMAssay Description:Inhibition of FLAG-tagged IKKbeta after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319759(CHEMBL1085309 | N-(2-hydroxyethyl)-4-(4-(thiophen-...)
Affinity DataIC50:  130nMAssay Description:Inhibition of FLAG-tagged IKKbeta after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319757(CHEMBL1085710 | N-(3-(dimethylamino)propyl)-4-(4-(...)
Affinity DataIC50:  170nMAssay Description:Inhibition of FLAG-tagged IKKbeta after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319753(4-(4-(thiophen-3-yl)pyrimidin-2-ylamino)benzenesul...)
Affinity DataIC50:  180nMAssay Description:Inhibition of FLAG-tagged IKKbeta after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319755(CHEMBL1085880 | N-(2-(dimethylamino)ethyl)-4-(4-(t...)
Affinity DataIC50:  230nMAssay Description:Inhibition of FLAG-tagged IKKbeta after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319751(CHEMBL1083483 | methyl 3-oxo-3-(2-(4-sulfamoylphen...)
Affinity DataIC50:  280nMAssay Description:Inhibition of FLAG-tagged IKKbeta after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319745(CHEMBL1084628 | N-(2-(4-sulfamoylphenylamino)-5,6-...)
Affinity DataIC50:  310nMAssay Description:Inhibition of FLAG-tagged IKKbeta after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319738(4-(8-methoxy-5,6-dihydrobenzo[h]quinazolin-2-ylami...)
Affinity DataIC50:  420nMAssay Description:Inhibition of IKKbeta expressed in human HeLa cells transfected with pNFkappaB-luciferase assessed inhibition of TNFalpha-induced NF-kappaB expressio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319744(CHEMBL1084361 | N-(2-(4-sulfamoylphenylamino)-5,6-...)
Affinity DataIC50:  510nMAssay Description:Inhibition of FLAG-tagged IKKbeta after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319756(4-(5,6-dihydrothieno[2,3-h]quinazolin-2-ylamino)-N...)
Affinity DataIC50:  510nMAssay Description:Inhibition of IKKbeta expressed in human HeLa cells transfected with pNFkappaB-luciferase assessed inhibition of TNFalpha-induced NF-kappaB expressio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319738(4-(8-methoxy-5,6-dihydrobenzo[h]quinazolin-2-ylami...)
Affinity DataIC50:  550nMAssay Description:Inhibition of FLAG-tagged IKKbeta after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319758(4-(5,6-dihydrothieno[2,3-h]quinazolin-2-ylamino)-N...)
Affinity DataIC50:  620nMAssay Description:Inhibition of IKKbeta expressed in human HeLa cells transfected with pNFkappaB-luciferase assessed inhibition of TNFalpha-induced NF-kappaB expressio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319737(4-(4-(4-methoxyphenyl)pyrimidin-2-ylamino)benzenes...)
Affinity DataIC50:  640nMAssay Description:Inhibition of IKKbeta expressed in human HeLa cells transfected with pNFkappaB-luciferase assessed inhibition of TNFalpha-induced NF-kappaB expressio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319756(4-(5,6-dihydrothieno[2,3-h]quinazolin-2-ylamino)-N...)
Affinity DataIC50:  770nMAssay Description:Inhibition of FLAG-tagged IKKbeta after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319755(CHEMBL1085880 | N-(2-(dimethylamino)ethyl)-4-(4-(t...)
Affinity DataIC50:  770nMAssay Description:Inhibition of IKKbeta expressed in human HeLa cells transfected with pNFkappaB-luciferase assessed inhibition of TNFalpha-induced NF-kappaB expressio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319758(4-(5,6-dihydrothieno[2,3-h]quinazolin-2-ylamino)-N...)
Affinity DataIC50:  780nMAssay Description:Inhibition of FLAG-tagged IKKbeta after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319754(4-(5,6-dihydrothieno[2,3-h]quinazolin-2-ylamino)be...)
Affinity DataIC50:  790nMAssay Description:Inhibition of FLAG-tagged IKKbeta after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319754(4-(5,6-dihydrothieno[2,3-h]quinazolin-2-ylamino)be...)
Affinity DataIC50:  800nMAssay Description:Inhibition of IKKbeta expressed in human HeLa cells transfected with pNFkappaB-luciferase assessed inhibition of TNFalpha-induced NF-kappaB expressio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319740(3,3-dimethyl-N-(2-(4-sulfamoylphenylamino)-5,6-dih...)
Affinity DataIC50:  820nMAssay Description:Inhibition of FLAG-tagged IKKbeta after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319744(CHEMBL1084361 | N-(2-(4-sulfamoylphenylamino)-5,6-...)
Affinity DataIC50:  830nMAssay Description:Inhibition of IKKbeta expressed in human HeLa cells transfected with pNFkappaB-luciferase assessed inhibition of TNFalpha-induced NF-kappaB expressio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319745(CHEMBL1084628 | N-(2-(4-sulfamoylphenylamino)-5,6-...)
Affinity DataIC50:  970nMAssay Description:Inhibition of IKKbeta expressed in human HeLa cells transfected with pNFkappaB-luciferase assessed inhibition of TNFalpha-induced NF-kappaB expressio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319757(CHEMBL1085710 | N-(3-(dimethylamino)propyl)-4-(4-(...)
Affinity DataIC50:  1.06E+3nMAssay Description:Inhibition of IKKbeta expressed in human HeLa cells transfected with pNFkappaB-luciferase assessed inhibition of TNFalpha-induced NF-kappaB expressio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319750(CHEMBL1083482 | N-(2-(4-sulfamoylphenylamino)-5,6-...)
Affinity DataIC50:  1.11E+3nMAssay Description:Inhibition of FLAG-tagged IKKbeta after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319760(4-(5,6-dihydrothieno[2,3-h]quinazolin-2-ylamino)-N...)
Affinity DataIC50:  1.22E+3nMAssay Description:Inhibition of FLAG-tagged IKKbeta after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319740(3,3-dimethyl-N-(2-(4-sulfamoylphenylamino)-5,6-dih...)
Affinity DataIC50:  1.36E+3nMAssay Description:Inhibition of IKKbeta expressed in human HeLa cells transfected with pNFkappaB-luciferase assessed inhibition of TNFalpha-induced NF-kappaB expressio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319735(4-(5,6-dihydrobenzo[h]quinazolin-2-ylamino)benzene...)
Affinity DataIC50:  1.43E+3nMAssay Description:Inhibition of IKKbeta expressed in human HeLa cells transfected with pNFkappaB-luciferase assessed inhibition of TNFalpha-induced NF-kappaB expressio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319750(CHEMBL1083482 | N-(2-(4-sulfamoylphenylamino)-5,6-...)
Affinity DataIC50:  1.46E+3nMAssay Description:Inhibition of IKKbeta expressed in human HeLa cells transfected with pNFkappaB-luciferase assessed inhibition of TNFalpha-induced NF-kappaB expressio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319749(CHEMBL1083176 | N-(2-(4-sulfamoylphenylamino)-5,6-...)
Affinity DataIC50:  1.57E+3nMAssay Description:Inhibition of IKKbeta expressed in human HeLa cells transfected with pNFkappaB-luciferase assessed inhibition of TNFalpha-induced NF-kappaB expressio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319748(3-methyl-N-(2-(4-sulfamoylphenylamino)-5,6-dihydro...)
Affinity DataIC50:  1.59E+3nMAssay Description:Inhibition of FLAG-tagged IKKbeta after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319746(2-(4-methoxyphenyl)-N-(2-(4-sulfamoylphenylamino)-...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of IKKbeta expressed in human HeLa cells transfected with pNFkappaB-luciferase assessed inhibition of TNFalpha-induced NF-kappaB expressio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319753(4-(4-(thiophen-3-yl)pyrimidin-2-ylamino)benzenesul...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of IKKbeta expressed in human HeLa cells transfected with pNFkappaB-luciferase assessed inhibition of TNFalpha-induced NF-kappaB expressio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50303035(4-(4-(5-methylthiophen-2-yl)pyrimidin-2-ylamino)be...)
Affinity DataIC50:  1.71E+3nMAssay Description:Inhibition of IKKbeta expressed in human HeLa cells transfected with pNFkappaB-luciferase assessed inhibition of TNFalpha-induced NF-kappaB expressio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319742(2-phenyl-N-(2-(4-sulfamoylphenylamino)-5,6-dihydro...)
Affinity DataIC50:  1.79E+3nMAssay Description:Inhibition of IKKbeta expressed in human HeLa cells transfected with pNFkappaB-luciferase assessed inhibition of TNFalpha-induced NF-kappaB expressio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319735(4-(5,6-dihydrobenzo[h]quinazolin-2-ylamino)benzene...)
Affinity DataIC50:  1.83E+3nMAssay Description:Inhibition of FLAG-tagged IKKbeta after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319746(2-(4-methoxyphenyl)-N-(2-(4-sulfamoylphenylamino)-...)
Affinity DataIC50:  1.83E+3nMAssay Description:Inhibition of FLAG-tagged IKKbeta after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319747(3-methyl-N-(2-(4-sulfamoylphenylamino)-5,6-dihydro...)
Affinity DataIC50:  1.94E+3nMAssay Description:Inhibition of FLAG-tagged IKKbeta after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319760(4-(5,6-dihydrothieno[2,3-h]quinazolin-2-ylamino)-N...)
Affinity DataIC50:  1.96E+3nMAssay Description:Inhibition of IKKbeta expressed in human HeLa cells transfected with pNFkappaB-luciferase assessed inhibition of TNFalpha-induced NF-kappaB expressio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319749(CHEMBL1083176 | N-(2-(4-sulfamoylphenylamino)-5,6-...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of FLAG-tagged IKKbeta after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319752(CHEMBL1086357 | N-(2-(4-sulfamoylphenylamino)-5,6-...)
Affinity DataIC50:  2.23E+3nMAssay Description:Inhibition of FLAG-tagged IKKbeta after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319742(2-phenyl-N-(2-(4-sulfamoylphenylamino)-5,6-dihydro...)
Affinity DataIC50:  2.38E+3nMAssay Description:Inhibition of FLAG-tagged IKKbeta after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319739(3,3-dimethyl-N-(4-(2-(4-sulfamoylphenylamino)pyrim...)
Affinity DataIC50:  2.46E+3nMAssay Description:Inhibition of IKKbeta expressed in human HeLa cells transfected with pNFkappaB-luciferase assessed inhibition of TNFalpha-induced NF-kappaB expressio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319759(CHEMBL1085309 | N-(2-hydroxyethyl)-4-(4-(thiophen-...)
Affinity DataIC50:  3.39E+3nMAssay Description:Inhibition of IKKbeta expressed in human HeLa cells transfected with pNFkappaB-luciferase assessed inhibition of TNFalpha-induced NF-kappaB expressio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319736(4-(6,7-Dihydro-5H-benzo[6,7]cyclohepta[1,2-d]pyrim...)
Affinity DataIC50:  4.06E+3nMAssay Description:Inhibition of IKKbeta expressed in human HeLa cells transfected with pNFkappaB-luciferase assessed inhibition of TNFalpha-induced NF-kappaB expressio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319741(2-phenyl-N-(4-(2-(4-sulfamoylphenylamino)pyrimidin...)
Affinity DataIC50:  4.47E+3nMAssay Description:Inhibition of IKKbeta expressed in human HeLa cells transfected with pNFkappaB-luciferase assessed inhibition of TNFalpha-induced NF-kappaB expressio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319747(3-methyl-N-(2-(4-sulfamoylphenylamino)-5,6-dihydro...)
Affinity DataIC50:  6.40E+3nMAssay Description:Inhibition of IKKbeta expressed in human HeLa cells transfected with pNFkappaB-luciferase assessed inhibition of TNFalpha-induced NF-kappaB expressio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50319743(CHEMBL1085122 | N-(4-(2-(4-sulfamoylphenylamino)py...)
Affinity DataIC50:  6.91E+3nMAssay Description:Inhibition of IKKbeta expressed in human HeLa cells transfected with pNFkappaB-luciferase assessed inhibition of TNFalpha-induced NF-kappaB expressio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 53 total ) | Next | Last >>
Jump to: