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PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt UniProtKB/TrEMBL
B.MOAD DrugBank antibodypedia GoogleScholar

Potassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Karl-Franzens-University

Curated by ChEMBL

BDBM22985(Aralen | CHEMBL76 | CHLOROQUINE PHOSPHATE | Chloro...)

IC50: 2.50E+3nMAssay Description:Inhibition of human ERG expressed in HEK293 cells assessed as reduction in tail current at membrane potential of +20 mVMore data for this Ligand-Target Pair

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CHEMBL DrugBank MCE
KEGG PC cid PC sid PDB Patents Similars

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt UniProtKB/TrEMBL
B.MOAD DrugBank antibodypedia GoogleScholar

Potassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Karl-Franzens-University

Curated by ChEMBL

BDBM50151865(CHEMBL172 | MEFLOQUINE)

IC50: 2.60E+3nMAssay Description:Inhibition of human ERG expressed in HEK293 cells assessed as reduction in tail current at membrane potential of +20 mVMore data for this Ligand-Target Pair

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CHEMBL MCE
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PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD GoogleScholar

Prostaglandin G/H synthase 2(Ovis aries (Sheep))
University Of Graz

Curated by ChEMBL

BDBM50029593(CHEMBL7162 | N-(2-(cyclohexyloxy)-4-nitrophenyl)me...)

IC50: 2.60E+3nMAssay Description:Inhibition of sheep placental cotyledens COX2 assessed as PGE2 level by EIAMore data for this Ligand-Target Pair

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CHEMBL MCE
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Details Article PubMed PDB

3D Structure (crystal)

Potassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Karl-Franzens-University

Curated by ChEMBL

BDBM50065629(CHEMBL3401424)

IC50: 2.63E+3nMAssay Description:Inhibition of human ERG expressed in HEK293 cells assessed as reduction in tail current at membrane potential of +20 mVMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt UniProtKB/TrEMBL
B.MOAD DrugBank antibodypedia GoogleScholar

CHEMBL PC cid PC sid

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank GoogleScholar

Polyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL

BDBM50315285(CHEMBL1089840 | aR-6,7-dihydro-6-(10-hydroxyethyl)...)

IC50: 4.20E+3nMAssay Description:Inhibition of 5-LOX-mediated LTB4 production in stimulated human neutrophile granulocytes after 10 mins by EIAMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank GoogleScholar

Polyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL

BDBM50315286(CHEMBL1088887 | aR-6-(10-iodoethyl)-1,2,3,9,10,11-...)

IC50: 4.50E+3nMAssay Description:Inhibition of 5-LOX-mediated LTB4 production in stimulated human neutrophile granulocytes after 10 mins by EIAMore data for this Ligand-Target Pair

Integrase(Human immunodeficiency virus 1)
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM50484177(CHEMBL1813504)

IC50: 5.00E+3nMAssay Description:Inhibition of wild-type HIV1 integrase strand transfer activity using [32P]-5'-end-labeled 5'-ACTGCTAGAGATTTTCCACAC-3' as substrate after 1 hrMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank GoogleScholar

Polyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
University Of Graz

Curated by ChEMBL

BDBM50000541((+-)-1-(1-Benzo[b]thien-2-ylethyl)-1-hydroxyurea |...)

IC50: 5.00E+3nMAssay Description:Inhibition of 5-LOX-mediated LTB4 production in stimulated human neutrophile granulocytes after 10 mins by EIAMore data for this Ligand-Target Pair

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CHEMBL DrugBank MCE
PC cid PC sid Patents Similars

Details Article PubMed DrugBank

Integrase(Human immunodeficiency virus 1)
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM50484163(CHEMBL1813506)

IC50: 8.00E+3nMAssay Description:Inhibition of wild-type HIV1 integrase strand transfer activity using [32P]-5'-end-labeled 5'-ACTGCTAGAGATTTTCCACAC-3' as substrate after 1 hrMore data for this Ligand-Target Pair

Integrase(Human immunodeficiency virus 1)
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM50484164(CHEMBL1813508)

IC50: 1.10E+4nMAssay Description:Inhibition of wild-type HIV1 integrase strand transfer activity using [32P]-5'-end-labeled 5'-ACTGCTAGAGATTTTCCACAC-3' as substrate after 1 hrMore data for this Ligand-Target Pair

Integrase(Human immunodeficiency virus 1)
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM50484168(CHEMBL1813496)

IC50: 1.20E+4nMAssay Description:Inhibition of wild-type HIV1 integrase strand transfer activity using [32P]-5'-end-labeled 5'-ACTGCTAGAGATTTTCCACAC-3' as substrate after 1 hrMore data for this Ligand-Target Pair

Integrase(Human immunodeficiency virus 1)
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM50484182(CHEMBL1813507)

IC50: 1.30E+4nMAssay Description:Inhibition of wild-type HIV1 integrase strand transfer activity using [32P]-5'-end-labeled 5'-ACTGCTAGAGATTTTCCACAC-3' as substrate after 1 hrMore data for this Ligand-Target Pair

Integrase(Human immunodeficiency virus 1)
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM50484147(CHEMBL1813512)

IC50: 1.40E+4nMAssay Description:Inhibition of wild-type HIV1 integrase strand transfer activity using [32P]-5'-end-labeled 5'-ACTGCTAGAGATTTTCCACAC-3' as substrate after 1 hrMore data for this Ligand-Target Pair

Integrase(Human immunodeficiency virus 1)
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM50484160(CHEMBL1813497)

IC50: 1.50E+4nMAssay Description:Inhibition of wild-type HIV1 integrase strand transfer activity using [32P]-5'-end-labeled 5'-ACTGCTAGAGATTTTCCACAC-3' as substrate after 1 hrMore data for this Ligand-Target Pair

Integrase(Human immunodeficiency virus 1)
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM50484169(CHEMBL1813501)

IC50: 1.80E+4nMAssay Description:Inhibition of wild-type HIV1 integrase strand transfer activity using [32P]-5'-end-labeled 5'-ACTGCTAGAGATTTTCCACAC-3' as substrate after 1 hrMore data for this Ligand-Target Pair

Integrase(Human immunodeficiency virus 1)
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM50484146(CHEMBL1813509)

IC50: 1.90E+4nMAssay Description:Inhibition of wild-type HIV1 integrase strand transfer activity using [32P]-5'-end-labeled 5'-ACTGCTAGAGATTTTCCACAC-3' as substrate after 1 hrMore data for this Ligand-Target Pair

Integrase(Human immunodeficiency virus 1)
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM50484171(CHEMBL1813514)

IC50: 2.00E+4nMAssay Description:Inhibition of wild-type HIV1 integrase strand transfer activity using [32P]-5'-end-labeled 5'-ACTGCTAGAGATTTTCCACAC-3' as substrate after 1 hrMore data for this Ligand-Target Pair

Integrase(Human immunodeficiency virus 1)
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM50484161(CHEMBL1813498)

IC50: 2.10E+4nMAssay Description:Inhibition of wild-type HIV1 integrase strand transfer activity using [32P]-5'-end-labeled 5'-ACTGCTAGAGATTTTCCACAC-3' as substrate after 1 hrMore data for this Ligand-Target Pair

Integrase(Human immunodeficiency virus 1)
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM50484148(CHEMBL1813513)

IC50: 2.20E+4nMAssay Description:Inhibition of wild-type HIV1 integrase strand transfer activity using [32P]-5'-end-labeled 5'-ACTGCTAGAGATTTTCCACAC-3' as substrate after 1 hrMore data for this Ligand-Target Pair

Integrase(Human immunodeficiency virus 1)
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM50484158(CHEMBL1813386)

IC50: 2.30E+4nMAssay Description:Inhibition of wild-type HIV1 integrase strand transfer activity using [32P]-5'-end-labeled 5'-ACTGCTAGAGATTTTCCACAC-3' as substrate after 1 hrMore data for this Ligand-Target Pair

Integrase(Human immunodeficiency virus 1)
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM50484159(CHEMBL1813493)

IC50: 2.40E+4nMAssay Description:Inhibition of wild-type HIV1 integrase strand transfer activity using [32P]-5'-end-labeled 5'-ACTGCTAGAGATTTTCCACAC-3' as substrate after 1 hrMore data for this Ligand-Target Pair

Integrase(Human immunodeficiency virus 1)
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM50484181(CHEMBL1813385)

IC50: 2.60E+4nMAssay Description:Inhibition of wild-type HIV1 integrase strand transfer activity using [32P]-5'-end-labeled 5'-ACTGCTAGAGATTTTCCACAC-3' as substrate after 1 hrMore data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD GoogleScholar

Prostaglandin G/H synthase 2(Ovis aries (Sheep))
University Of Graz

Curated by ChEMBL

BDBM50315284(CHEMBL1089510 | aR-6,7-Dihydro-6-(10-hydroxyethyl)...)

IC50: 3.21E+4nMAssay Description:Inhibition of sheep placental cotyledens COX2 assessed as PGE2 level by EIAMore data for this Ligand-Target Pair

Integrase(Human immunodeficiency virus 1)
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM50484173(CHEMBL1813511)

IC50: 3.40E+4nMAssay Description:Inhibition of wild-type HIV1 integrase strand transfer activity using [32P]-5'-end-labeled 5'-ACTGCTAGAGATTTTCCACAC-3' as substrate after 1 hrMore data for this Ligand-Target Pair

Integrase(Human immunodeficiency virus 1)
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM50477870(CHEMBL252553)

IC50: 3.50E+4nMAssay Description:Inhibition of wild-type HIV1 integrase strand transfer activity using [32P]-5'-end-labeled 5'-ACTGCTAGAGATTTTCCACAC-3' as substrate after 1 hrMore data for this Ligand-Target Pair

Integrase(Human immunodeficiency virus 1)
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM50484183(CHEMBL1813515)

IC50: 3.90E+4nMAssay Description:Inhibition of wild-type HIV1 integrase strand transfer activity using [32P]-5'-end-labeled 5'-ACTGCTAGAGATTTTCCACAC-3' as substrate after 1 hrMore data for this Ligand-Target Pair

Integrase(Human immunodeficiency virus 1)
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM50484165(CHEMBL1813510)

IC50: 4.40E+4nMAssay Description:Inhibition of wild-type HIV1 integrase strand transfer activity using [32P]-5'-end-labeled 5'-ACTGCTAGAGATTTTCCACAC-3' as substrate after 1 hrMore data for this Ligand-Target Pair

Integrase(Human immunodeficiency virus 1)
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM50484145(CHEMBL1813505)

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD GoogleScholar

Prostaglandin G/H synthase 2(Ovis aries (Sheep))
University Of Graz

Curated by ChEMBL

BDBM50116888(CHEMBL3612976)

IC50: 5.00E+4nMAssay Description:Inhibition of sheep placental cotyledons COX-2 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition after 20 mi...More data for this Ligand-Target Pair

Integrase(Human immunodeficiency virus 1)
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM50484146(CHEMBL1813509)

IC50: 5.30E+4nMAssay Description:Inhibition of wild-type HIV1 integrase 3'-processing activity using [32P]-5'-end-labeled 5'-ACTGCTAGAGATTTTCCACAC-3' as substrate after 1 hrMore data for this Ligand-Target Pair

Integrase(Human immunodeficiency virus 1)
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM50484147(CHEMBL1813512)

IC50: 5.50E+4nMAssay Description:Inhibition of wild-type HIV1 integrase 3'-processing activity using [32P]-5'-end-labeled 5'-ACTGCTAGAGATTTTCCACAC-3' as substrate after 1 hrMore data for this Ligand-Target Pair

Integrase(Human immunodeficiency virus 1)
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM50484143(CHEMBL1813502)

IC50: 5.60E+4nMAssay Description:Inhibition of wild-type HIV1 integrase strand transfer activity using [32P]-5'-end-labeled 5'-ACTGCTAGAGATTTTCCACAC-3' as substrate after 1 hrMore data for this Ligand-Target Pair

Integrase(Human immunodeficiency virus 1)
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM50484170(CHEMBL1813495)

IC50: 5.80E+4nMAssay Description:Inhibition of wild-type HIV1 integrase strand transfer activity using [32P]-5'-end-labeled 5'-ACTGCTAGAGATTTTCCACAC-3' as substrate after 1 hrMore data for this Ligand-Target Pair

Integrase(Human immunodeficiency virus 1)
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM50484163(CHEMBL1813506)

IC50: 7.00E+4nMAssay Description:Inhibition of wild-type HIV1 integrase 3'-processing activity using [32P]-5'-end-labeled 5'-ACTGCTAGAGATTTTCCACAC-3' as substrate after 1 hrMore data for this Ligand-Target Pair

Integrase(Human immunodeficiency virus 1)
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM50484148(CHEMBL1813513)

IC50: 7.50E+4nMAssay Description:Inhibition of wild-type HIV1 integrase 3'-processing activity using [32P]-5'-end-labeled 5'-ACTGCTAGAGATTTTCCACAC-3' as substrate after 1 hrMore data for this Ligand-Target Pair

Integrase(Human immunodeficiency virus 1)
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM50484168(CHEMBL1813496)

IC50: 8.30E+4nMAssay Description:Inhibition of wild-type HIV1 integrase 3'-processing activity using [32P]-5'-end-labeled 5'-ACTGCTAGAGATTTTCCACAC-3' as substrate after 1 hrMore data for this Ligand-Target Pair

Integrase(Human immunodeficiency virus 1)
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM50484178(CHEMBL1813382)

IC50: 8.50E+4nMAssay Description:Inhibition of wild-type HIV1 integrase strand transfer activity using [32P]-5'-end-labeled 5'-ACTGCTAGAGATTTTCCACAC-3' as substrate after 1 hrMore data for this Ligand-Target Pair

Integrase(Human immunodeficiency virus 1)
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM50484164(CHEMBL1813508)

IC50: 8.90E+4nMAssay Description:Inhibition of wild-type HIV1 integrase 3'-processing activity using [32P]-5'-end-labeled 5'-ACTGCTAGAGATTTTCCACAC-3' as substrate after 1 hrMore data for this Ligand-Target Pair

Integrase(Human immunodeficiency virus 1)
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM50484160(CHEMBL1813497)

IC50: 9.00E+4nMAssay Description:Inhibition of wild-type HIV1 integrase 3'-processing activity using [32P]-5'-end-labeled 5'-ACTGCTAGAGATTTTCCACAC-3' as substrate after 1 hrMore data for this Ligand-Target Pair

Integrase(Human immunodeficiency virus 1)
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM50484166(CHEMBL1813383)

IC50: 9.70E+4nMAssay Description:Inhibition of wild-type HIV1 integrase strand transfer activity using [32P]-5'-end-labeled 5'-ACTGCTAGAGATTTTCCACAC-3' as substrate after 1 hrMore data for this Ligand-Target Pair

Integrase(Human immunodeficiency virus 1)
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM50484144(CHEMBL1813503)

IC50: 1.00E+5nMAssay Description:Inhibition of wild-type HIV1 integrase strand transfer activity using [32P]-5'-end-labeled 5'-ACTGCTAGAGATTTTCCACAC-3' as substrate after 1 hrMore data for this Ligand-Target Pair

Integrase(Human immunodeficiency virus 1)
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM50484149(CHEMBL1813517)

IC50: >1.00E+5nMAssay Description:Inhibition of wild-type HIV1 integrase strand transfer activity using [32P]-5'-end-labeled 5'-ACTGCTAGAGATTTTCCACAC-3' as substrate after 1 hrMore data for this Ligand-Target Pair

Integrase(Human immunodeficiency virus 1)
Chinese Academy Of Sciences

Curated by ChEMBL

BDBM50484150(CHEMBL1813371)

IC50: >1.00E+5nMAssay Description:Inhibition of wild-type HIV1 integrase 3'-processing activity using [32P]-5'-end-labeled 5'-ACTGCTAGAGATTTTCCACAC-3' as substrate after 1 hrMore data for this Ligand-Target Pair