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Found 173 with Last Name = 'sahu' and Initial = 'pk'
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50252829((2S,3S,4R,5R)-5-(6-(3-iodobenzylamino)-9H-purin-9-...)
Affinity DataKi:  0.25nMAssay Description:Displacement of [125I]I-AB-MECA from human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50237784(CHEMBL4088081)
Affinity DataKi:  0.570nMAssay Description:Displacement of [125I]I-AB-MECA from human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50237775(CHEMBL4068467)
Affinity DataKi:  0.900nMAssay Description:Displacement of [125I]I-AB-MECA from human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50237788(CHEMBL4087331)
Affinity DataKi:  1nMAssay Description:Displacement of [125I]I-AB-MECA from human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50237770(CHEMBL4067750)
Affinity DataKi:  1.40nMAssay Description:Binding affinity to human sphingosine 1-phosphate receptor 5 expressed in CHO cells was determined by using [33P]-S1P as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM21221((2S,3S,4R,5R)-5-(2-chloro-6-{[(3-iodophenyl)methyl...)
Affinity DataKi:  1.40nMAssay Description:Displacement of [125I]I-AB-MECA from human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50237782(CHEMBL4059977)
Affinity DataKi:  1.5nMAssay Description:Displacement of [125I]I-AB-MECA from human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50237789(CHEMBL4103146)
Affinity DataKi:  1.80nMAssay Description:Displacement of [125I]I-AB-MECA from human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50118812((2S,3S,4R,5R)-3,4-Dihydroxy-5-[6-(3-iodo-benzylami...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [125I]I-AB-MECA from human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50237778(CHEMBL4103705)
Affinity DataKi:  1.90nMAssay Description:Displacement of [125I]I-AB-MECA from human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50237786(CHEMBL4068634)
Affinity DataKi:  2nMAssay Description:Displacement of [125I]I-AB-MECA from human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50237780(CHEMBL4102379)
Affinity DataKi:  2nMAssay Description:Displacement of [125I]I-AB-MECA from human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50237777(CHEMBL4078444)
Affinity DataKi:  2.30nMAssay Description:Displacement of [125I]I-AB-MECA from human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50237771(CHEMBL4090519)
Affinity DataKi:  2.5nMAssay Description:Displacement of [125I]I-AB-MECA from human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50237781(CHEMBL4084951)
Affinity DataKi:  3.40nMAssay Description:Displacement of [125I]I-AB-MECA from human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50237776(CHEMBL4095809)
Affinity DataKi:  3.5nMAssay Description:Displacement of [125I]I-AB-MECA from human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50237785(CHEMBL4065920)
Affinity DataKi:  3.60nMAssay Description:Displacement of [125I]I-AB-MECA from human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50237774(CHEMBL4059807)
Affinity DataKi:  3.80nMAssay Description:Displacement of [125I]I-AB-MECA from human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50237772(CHEMBL4069499)
Affinity DataKi:  3.90nMAssay Description:Displacement of [125I]I-AB-MECA from human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50237779(CHEMBL4079448)
Affinity DataKi:  4.20nMAssay Description:Displacement of [125I]I-AB-MECA from human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50237773(CHEMBL4080205)
Affinity DataKi:  4.40nMAssay Description:Displacement of [125I]I-AB-MECA from human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496304(CHEMBL3125712)
Affinity DataKi:  4.90nMAssay Description:Displacement of [125I]-I-AB-MECA from recombinant human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496310(CHEMBL3125713)
Affinity DataKi:  6.70nMAssay Description:Displacement of [125I]-I-AB-MECA from recombinant human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50237783(CHEMBL4094418)
Affinity DataKi:  7.10nMAssay Description:Displacement of [125I]I-AB-MECA from human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496311(CHEMBL3125718)
Affinity DataKi:  7.80nMAssay Description:Displacement of [125I]-I-AB-MECA from recombinant human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496307(CHEMBL3125717)
Affinity DataKi:  8.60nMAssay Description:Displacement of [125I]-I-AB-MECA from recombinant human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496308(CHEMBL3125714)
Affinity DataKi:  9.20nMAssay Description:Displacement of [125I]-I-AB-MECA from recombinant human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496311(CHEMBL3125718)
Affinity DataKi:  11nMAssay Description:Displacement of [125I]-I-AB-MECA from rat adenosine A3 receptor expressed in RBL-2H3 cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496305(CHEMBL3125716)
Affinity DataKi:  12nMAssay Description:Displacement of [125I]-I-AB-MECA from recombinant human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496306(CHEMBL3125711)
Affinity DataKi:  16nMAssay Description:Displacement of [125I]-I-AB-MECA from recombinant human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496309(CHEMBL3125719)
Affinity DataKi:  16nMAssay Description:Displacement of [125I]-I-AB-MECA from recombinant human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50252829((2S,3S,4R,5R)-5-(6-(3-iodobenzylamino)-9H-purin-9-...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]R-PLA from human adenosine A1 receptor expressed in CHO cells after 60 mins by liquid scintillation analyzerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50237783(CHEMBL4094418)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]R-PLA from human adenosine A1 receptor expressed in CHO cells after 60 mins by liquid scintillation analyzerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496305(CHEMBL3125716)
Affinity DataKi:  26nMAssay Description:Displacement of [125I]-I-AB-MECA from rat adenosine A3 receptor expressed in RBL-2H3 cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50237770(CHEMBL4067750)
Affinity DataKi:  38nMAssay Description:Compound was tested for binding affinity against Fucosyltransferase 6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496308(CHEMBL3125714)
Affinity DataKi:  39nMAssay Description:Displacement of [125I]-I-AB-MECA from rat adenosine A3 receptor expressed in RBL-2H3 cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496309(CHEMBL3125719)
Affinity DataKi:  43nMAssay Description:Displacement of [125I]-I-AB-MECA from rat adenosine A3 receptor expressed in RBL-2H3 cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496303(CHEMBL3125715)
Affinity DataKi:  58nMAssay Description:Displacement of [125I]-I-AB-MECA from rat adenosine A3 receptor expressed in RBL-2H3 cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50237785(CHEMBL4065920)
Affinity DataKi:  59nMAssay Description:Displacement of [3H]R-PLA from human adenosine A1 receptor expressed in CHO cells after 60 mins by liquid scintillation analyzerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496307(CHEMBL3125717)
Affinity DataKi:  59nMAssay Description:Displacement of [125I]-I-AB-MECA from rat adenosine A3 receptor expressed in RBL-2H3 cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50237788(CHEMBL4087331)
Affinity DataKi:  62nMAssay Description:Displacement of [3H]R-PLA from human adenosine A1 receptor expressed in CHO cells after 60 mins by liquid scintillation analyzerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496306(CHEMBL3125711)
Affinity DataKi:  65nMAssay Description:Displacement of [125I]-I-AB-MECA from rat adenosine A3 receptor expressed in RBL-2H3 cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50237771(CHEMBL4090519)
Affinity DataKi:  84nMAssay Description:Compound was tested for binding affinity against Fucosyltransferase 6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496306(CHEMBL3125711)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]-CGS21680 from human adenosine A2A receptor expressed in HEK293 cells after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50237780(CHEMBL4102379)
Affinity DataKi:  156nMAssay Description:Displacement of [3H]R-PLA from human adenosine A1 receptor expressed in CHO cells after 60 mins by liquid scintillation analyzerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496303(CHEMBL3125715)
Affinity DataKi:  160nMAssay Description:Displacement of [125I]-I-AB-MECA from recombinant human adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50496310(CHEMBL3125713)
Affinity DataKi:  176nMAssay Description:Displacement of [125I]-I-AB-MECA from rat adenosine A3 receptor expressed in RBL-2H3 cells after 60 mins by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50237778(CHEMBL4103705)
Affinity DataKi:  186nMAssay Description:Displacement of [3H]-citalopram from serotonin transporter of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50237789(CHEMBL4103146)
Affinity DataKi:  195nMAssay Description:Displacement of [3H]CGS21680 from human adenosine A2A receptor expressed in HEK293 cells after 60 mins by liquid scintillation analyzerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50237775(CHEMBL4068467)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]R-PLA from human adenosine A1 receptor expressed in CHO cells after 60 mins by liquid scintillation analyzerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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