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Found 139 with Last Name = 'salim' and Initial = 'a'
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029896(4'-(2-Butyl-6-oxo-6H-pyrimidin-1-ylmethyl)-bipheny...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50241491(2-{4-Butyl-2-methyl-6-oxo-5-[2'-(1H-tetrazol-5-yl)...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029903(3-Benzyl-6-butyl-2-methyl-5-[2'-(1H-tetrazol-5-yl)...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029911(2-{4-Butyl-2-methyl-6-oxo-5-[2'-(1H-tetrazol-5-yl)...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029910(4'-(4-Butyl-6-oxo-1,6-dihydro-pyrimidin-5-ylmethyl...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029907(4'-(1-Benzyl-4-butyl-6-oxo-1,6-dihydro-pyrimidin-5...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029909(4'-[4-Butyl-1-(2-carboxy-benzyl)-6-oxo-1,6-dihydro...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029906(2-[4-Butyl-5-(2'-carboxy-biphenyl-4-ylmethyl)-2-me...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029893(2-[4-Butyl-5-(2'-carboxy-biphenyl-4-ylmethyl)-2-me...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029908(4'-(4-Butyl-6-oxo-1-thiophen-2-ylmethyl-1,6-dihydr...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029899(3-{4-Butyl-2-methyl-6-oxo-5-[2'-(1H-tetrazol-5-yl)...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029905(4'-(2-Butyl-4-methyl-6-oxo-6H-pyrimidin-1-ylmethyl...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029895(2-{4-Butyl-2-methyl-6-oxo-5-[2'-(1H-tetrazol-5-yl)...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029894(4'-(4-Butyl-2-methyl-6-oxo-1,6-dihydro-pyrimidin-5...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029904(4'-[4-Butyl-1-(2-carboxy-benzyl)-2-methyl-6-oxo-1,...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029902(6-Butyl-2-methyl-5-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50241501(6-Butyl-2-methyl-5-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029892(2-{4-Butyl-2-methyl-6-oxo-5-[2'-(1H-tetrazol-5-yl)...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029901(2-{4-Butyl-2-methyl-6-oxo-5-[2'-(1H-tetrazol-5-yl)...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Istituto Lusofarmaco

Curated by ChEMBL
LigandPNGBDBM50029897(4'-[4-Butyl-1-(4-carboxy-benzyl)-6-oxo-1,6-dihydro...)
Affinity DataKi: >4nMAssay Description:Binding affinity towards Angiotensin II type 2 receptor in bovine cerebellar cortical membranes; InactiveMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50003399(4'-(2-Butyl-4-chloro-5-hydroxymethyl-imidazol-1-yl...)
Affinity DataKi:  350nMAssay Description:Tested for the binding affinity using radioligand [125I]-Sar1 Ile8-AII in the rat adrenal capsular membranes (adrenal cortex)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50470054(CHEMBL129225)
Affinity DataKi:  3.30E+3nMAssay Description:Tested for the binding affinity using radioligand [125I]-Sar1 Ile8-AII in the rat adrenal capsular membranes (adrenal cortex)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50470049(CHEMBL340682)
Affinity DataKi:  6.70E+3nMAssay Description:Tested for the binding affinity using radioligand [125I]-Sar1 Ile8-AII in the rat adrenal capsular membranes (adrenal cortex)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50470051(CHEMBL339044)
Affinity DataKi:  9.70E+3nMAssay Description:Tested for the binding affinity using radioligand [125I]-Sar1 Ile8-AII in the rat adrenal capsular membranes (adrenal cortex)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50470050(CHEMBL129170)
Affinity DataKi:  9.80E+3nMAssay Description:Tested for the binding affinity using radioligand [125I]-Sar1 Ile8-AII in the rat adrenal capsular membranes (adrenal cortex)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50470052(CHEMBL127108)
Affinity DataKi: >1.00E+4nMAssay Description:Tested for the binding affinity using radioligand [125I]-Sar1 Ile8-AII in the rat adrenal capsular membranes (adrenal cortex)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50470060(CHEMBL125789)
Affinity DataKi: >1.00E+4nMAssay Description:Tested for the binding affinity using radioligand [125I]-Sar1 Ile8-AII in the rat adrenal capsular membranes (adrenal cortex)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50470055(CHEMBL125790)
Affinity DataKi: >1.00E+4nMAssay Description:Tested for the binding affinity using radioligand [125I]-Sar1 Ile8-AII in the rat adrenal capsular membranes (adrenal cortex)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50470057(CHEMBL129336)
Affinity DataKi: >1.00E+4nMAssay Description:Tested for the binding affinity using radioligand [125I]-Sar1 Ile8-AII in the rat adrenal capsular membranes (adrenal cortex)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50470048(CHEMBL128291)
Affinity DataKi: >1.00E+4nMAssay Description:Tested for the binding affinity using radioligand [125I]-Sar1 Ile8-AII in the rat adrenal capsular membranes (adrenal cortex)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50470047(CHEMBL50135)
Affinity DataKi: >1.00E+4nMAssay Description:Tested for the binding affinity using radioligand [125I]-Sar1 Ile8-AII in the rat adrenal capsular membranes (adrenal cortex)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50470059(CHEMBL338840)
Affinity DataKi: >1.00E+4nMAssay Description:Tested for the binding affinity using radioligand [125I]-Sar1 Ile8-AII in the rat adrenal capsular membranes (adrenal cortex)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50470058(CHEMBL129005)
Affinity DataKi: >1.00E+4nMAssay Description:Tested for the binding affinity using radioligand [125I]-Sar1 Ile8-AII in the rat adrenal capsular membranes (adrenal cortex)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50470053(CHEMBL125621)
Affinity DataKi:  1.16E+4nMAssay Description:Tested for the binding affinity using radioligand [125I]-Sar1 Ile8-AII in the rat adrenal capsular membranes (adrenal cortex)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50470056(CHEMBL129006)
Affinity DataKi:  1.45E+4nMAssay Description:Tested for the binding affinity using radioligand [125I]-Sar1 Ile8-AII in the rat adrenal capsular membranes (adrenal cortex)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290019((3S,6S,9aS)-6-(3-Methyl-1,2,3,4-tetrahydro-quinoli...)
Affinity DataIC50:  18nMAssay Description:In vitro ability to inhibit the activity of human alpha ThrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine protease 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50060000((S)-1-((R)-2-Methylamino-2-phenyl-acetyl)-pyrrolid...)
Affinity DataIC50:  20nMAssay Description:In vitro ability to inhibit the activity of TrypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50060000((S)-1-((R)-2-Methylamino-2-phenyl-acetyl)-pyrrolid...)
Affinity DataIC50:  26nMAssay Description:In vitro ability to inhibit the activity of human alpha ThrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50038001((2R,4R)-1-((S)-5-(diaminomethyleneamino)-2-(3-meth...)
Affinity DataIC50:  39nMAssay Description:In vitro ability to inhibit the activity of human alpha ThrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine protease 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50290019((3S,6S,9aS)-6-(3-Methyl-1,2,3,4-tetrahydro-quinoli...)
Affinity DataIC50:  100nMAssay Description:In vitro ability to inhibit the activity of TrypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290022((3S,6S,9aS)-5-Oxo-6-phenylmethanesulfonylamino-oct...)
Affinity DataIC50:  110nMAssay Description:In vitro ability to inhibit the activity of human alpha ThrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290021((3S,6S,9aS)-6-(Naphthalene-1-sulfonylamino)-5-oxo-...)
Affinity DataIC50:  110nMAssay Description:In vitro ability to inhibit the activity of human alpha ThrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50537903(CHEMBL4639635)
Affinity DataIC50:  350nMAssay Description:Reversal of P-gp mediated multidrug resistance in human SW620/AD300 cells assessed as potentiation of doxorubicin-induced antiproliferative activity ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholesterol side-chain cleavage enzyme, mitochondrial(Rattus norvegicus)
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50600678(CHEMBL5176174)
Affinity DataIC50:  500nMAssay Description:Antibacterial activity against Enterococcus faecalis incubated for 16 to 24 hrs by broth microdilution based spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPlasminogen(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50060000((S)-1-((R)-2-Methylamino-2-phenyl-acetyl)-pyrrolid...)
Affinity DataIC50:  500nMAssay Description:In vitro ability to inhibit the activity of PlasminMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSeed linoleate 13S-lipoxygenase-1(Glycine max (soybean))
Ferdowsi University Of Mashhad

LigandPNGBDBM192765(1,3-Dimethoxy-5-methyl-2-((2E,6E)-3,7,11-trimethyl...)
Affinity DataIC50:  520nMpH: 7.0 T: 2°CAssay Description:Solution A was 50 mm DMAB in an 100 mm phosphate buffer (pH 7.0). Solution B was a mixture of 10 mm MBTH (3 mL) and hemoglobin (5 mg/mL, 3 mL) in 50 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM81939(CAS_52-53-9 | NSC_62969 | VERAPAMIL)
Affinity DataIC50:  710nMAssay Description:Inhibition of P-gp mediated doxorubicin resistance in human SW620/AD300 cells overexpressing P-gp in presence of doxorubicin measured after 52 hrs by...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM81939(CAS_52-53-9 | NSC_62969 | VERAPAMIL)
Affinity DataIC50:  810nMAssay Description:Reversal of P-gp mediated multidrug resistance in human SW620/AD300 cells assessed as potentiation of doxorubicin-induced antiproliferative activity ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50537908(CHEMBL4641108)
Affinity DataIC50:  820nMAssay Description:Reversal of P-gp mediated multidrug resistance in human SW620/AD300 cells assessed as potentiation of doxorubicin-induced antiproliferative activity ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
The University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50537904(CHEMBL4646781)
Affinity DataIC50:  880nMAssay Description:Reversal of P-gp mediated multidrug resistance in human SW620/AD300 cells assessed as potentiation of doxorubicin-induced antiproliferative activity ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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