TargetTrypanothione reductase(Trypanosoma cruzi)
Pontificia Universidad Catolica Del Peru
Curated by ChEMBL
Pontificia Universidad Catolica Del Peru
Curated by ChEMBL
Affinity DataKi: 1.70E+3nMAssay Description:Inhibition of Trypanosoma cruzi recombinant trypanothione reductaseMore data for this Ligand-Target Pair
TargetTrypanothione reductase(Crithidia fasciculata)
Pontificia Universidad Catolica Del Peru
Curated by ChEMBL
Pontificia Universidad Catolica Del Peru
Curated by ChEMBL
Affinity DataKi: 1.80E+3nMAssay Description:Inhibition of Crithidia fasciculata free trypanothione reductaseMore data for this Ligand-Target Pair
TargetTrypanothione reductase(Trypanosoma cruzi)
Pontificia Universidad Catolica Del Peru
Curated by ChEMBL
Pontificia Universidad Catolica Del Peru
Curated by ChEMBL
Affinity DataKi: 2.00E+3nMAssay Description:Inhibition of Trypanosoma cruzi recombinant trypanothione reductaseMore data for this Ligand-Target Pair
TargetTrypanothione reductase(Trypanosoma cruzi)
Pontificia Universidad Catolica Del Peru
Curated by ChEMBL
Pontificia Universidad Catolica Del Peru
Curated by ChEMBL
Affinity DataKi: 3.20E+3nMAssay Description:Inhibition of Trypanosoma cruzi recombinant trypanothione reductaseMore data for this Ligand-Target Pair
TargetTrypanothione reductase(Trypanosoma cruzi)
Pontificia Universidad Catolica Del Peru
Curated by ChEMBL
Pontificia Universidad Catolica Del Peru
Curated by ChEMBL
Affinity DataKi: 7.00E+3nMAssay Description:Inhibition of Trypanosoma cruzi recombinant trypanothione reductaseMore data for this Ligand-Target Pair
TargetTrypanothione reductase(Trypanosoma cruzi)
Pontificia Universidad Catolica Del Peru
Curated by ChEMBL
Pontificia Universidad Catolica Del Peru
Curated by ChEMBL
Affinity DataKi: 7.00E+3nMAssay Description:Inhibition of Trypanosoma cruzi recombinant trypanothione reductaseMore data for this Ligand-Target Pair
TargetTrypanothione reductase(Trypanosoma cruzi)
Pontificia Universidad Catolica Del Peru
Curated by ChEMBL
Pontificia Universidad Catolica Del Peru
Curated by ChEMBL
Affinity DataKi: 7.60E+3nMAssay Description:Inhibition of Trypanosoma cruzi recombinant trypanothione reductaseMore data for this Ligand-Target Pair
TargetTrypanothione reductase(Trypanosoma cruzi)
Pontificia Universidad Catolica Del Peru
Curated by ChEMBL
Pontificia Universidad Catolica Del Peru
Curated by ChEMBL
Affinity DataKi: 1.20E+4nMAssay Description:Inhibition of Trypanosoma cruzi recombinant trypanothione reductaseMore data for this Ligand-Target Pair
TargetTrypanothione reductase(Crithidia fasciculata)
Pontificia Universidad Catolica Del Peru
Curated by ChEMBL
Pontificia Universidad Catolica Del Peru
Curated by ChEMBL
Affinity DataKi: 1.30E+4nMAssay Description:Inhibition of Crithidia fasciculata trypanothione reductase-substrate complexMore data for this Ligand-Target Pair
TargetTrypanothione reductase(Trypanosoma cruzi)
Pontificia Universidad Catolica Del Peru
Curated by ChEMBL
Pontificia Universidad Catolica Del Peru
Curated by ChEMBL
Affinity DataKi: 2.69E+4nMAssay Description:Inhibition of Trypanosoma cruzi recombinant trypanothione reductaseMore data for this Ligand-Target Pair
TargetTrypanothione reductase(Trypanosoma cruzi)
Pontificia Universidad Catolica Del Peru
Curated by ChEMBL
Pontificia Universidad Catolica Del Peru
Curated by ChEMBL
Affinity DataKi: 3.51E+4nMAssay Description:Inhibition of Trypanosoma cruzi recombinant trypanothione reductaseMore data for this Ligand-Target Pair
TargetTrypanothione reductase(Trypanosoma cruzi)
Pontificia Universidad Catolica Del Peru
Curated by ChEMBL
Pontificia Universidad Catolica Del Peru
Curated by ChEMBL
Affinity DataKi: 5.16E+4nMAssay Description:Inhibition of Trypanosoma cruzi recombinant trypanothione reductase-substrate complexMore data for this Ligand-Target Pair
TargetTrypanothione reductase(Trypanosoma cruzi)
Pontificia Universidad Catolica Del Peru
Curated by ChEMBL
Pontificia Universidad Catolica Del Peru
Curated by ChEMBL
Affinity DataKi: 6.46E+4nMAssay Description:Inhibition of Trypanosoma cruzi recombinant trypanothione reductaseMore data for this Ligand-Target Pair
TargetTrypanothione reductase(Trypanosoma cruzi)
Pontificia Universidad Catolica Del Peru
Curated by ChEMBL
Pontificia Universidad Catolica Del Peru
Curated by ChEMBL
Affinity DataKi: 1.44E+5nMAssay Description:Inhibition of Trypanosoma cruzi recombinant trypanothione reductaseMore data for this Ligand-Target Pair
Affinity DataIC50: 2.29E+3nMAssay Description:Antagonist activity against VDR-LBD (unknown origin) expressed in Escherichia coli assessed as inhibition of VDR agonist LG190178-induced SRC2-3 coac...More data for this Ligand-Target Pair
Affinity DataIC50: 2.86E+3nMAssay Description:Antagonist activity against VDR-LBD (unknown origin) expressed in Escherichia coli assessed as inhibition of VDR agonist LG190178-induced SRC2-3 coac...More data for this Ligand-Target Pair
TargetTrypanothione reductase(Trypanosoma cruzi)
Pontificia Universidad Catolica Del Peru
Curated by ChEMBL
Pontificia Universidad Catolica Del Peru
Curated by ChEMBL
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of Trypanosoma cruzi recombinant trypanothione reductaseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+4nMAssay Description:Agonist activity at VDR-LBD (unknown origin) expressed in Escherichia coli assessed as SRC2-3 coactivator peptide recruitment after 30 mins by fluore...More data for this Ligand-Target Pair
Affinity DataIC50: 1.36E+4nMAssay Description:Agonist activity at VDR-LBD (unknown origin) expressed in Escherichia coli assessed as SRC2-3 coactivator peptide recruitment after 30 mins by fluore...More data for this Ligand-Target Pair
Affinity DataIC50: 1.45E+4nMAssay Description:Antagonist activity against VDR-LBD (unknown origin) expressed in Escherichia coli assessed as inhibition of VDR agonist LG190178-induced SRC2-3 coac...More data for this Ligand-Target Pair
Affinity DataIC50: 1.51E+4nMAssay Description:Agonist activity at VP16 tagged-VDR-LBD (unknown origin) expressed in HEK293T cells assessed as SRC1 coactivator peptide recruitment after 16 hrs by ...More data for this Ligand-Target Pair
Affinity DataIC50: 2.33E+4nMAssay Description:Antagonist activity against VDR-LBD (unknown origin) expressed in Escherichia coli assessed as inhibition of VDR agonist LG190178-induced SRC2-3 coac...More data for this Ligand-Target Pair
Affinity DataIC50: 3.15E+4nMAssay Description:Antagonist activity against VDR-LBD (unknown origin) expressed in Escherichia coli assessed as inhibition of VDR agonist LG190178-induced SRC2-3 coac...More data for this Ligand-Target Pair
Affinity DataIC50: 4.01E+4nMAssay Description:Antagonist activity against VDR-LBD (unknown origin) expressed in Escherichia coli assessed as inhibition of VDR agonist LG190178-induced SRC2-3 coac...More data for this Ligand-Target Pair
Affinity DataIC50: 4.67E+4nMAssay Description:Antagonist activity against VDR-LBD (unknown origin) expressed in Escherichia coli assessed as inhibition of VDR agonist LG190178-induced SRC2-3 coac...More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Antagonist activity against VP16 tagged-VDR-LBD (unknown origin) expressed in HEK293T cells assessed as inhibition of 1,25-dihydroxyvitamin D3-induce...More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Antagonist activity against VP16 tagged-VDR-LBD (unknown origin) expressed in HEK293T cells assessed as inhibition of 1,25-dihydroxyvitamin D3-induce...More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Antagonist activity against VP16 tagged-VDR-LBD (unknown origin) expressed in HEK293T cells assessed as inhibition of 1,25-dihydroxyvitamin D3-induce...More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Antagonist activity against VP16 tagged-VDR-LBD (unknown origin) expressed in HEK293T cells assessed as inhibition of 1,25-dihydroxyvitamin D3-induce...More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Agonist activity at VP16 tagged-VDR-LBD (unknown origin) expressed in HEK293T cells assessed as SRC1 coactivator peptide recruitment after 16 hrs by ...More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Agonist activity at human VP16 tagged-VDR-LBD after 16 hrs by luciferase reporter gene based transcription assayMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Agonist activity at VP16 tagged-VDR-LBD (unknown origin) expressed in HEK293T cells assessed as SRC1 coactivator peptide recruitment after 16 hrs by ...More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Antagonist activity against VP16 tagged-VDR-LBD (unknown origin) expressed in HEK293T cells assessed as inhibition of 1,25-dihydroxyvitamin D3-induce...More data for this Ligand-Target Pair
TargetTrypanothione reductase(Trypanosoma cruzi)
Pontificia Universidad Catolica Del Peru
Curated by ChEMBL
Pontificia Universidad Catolica Del Peru
Curated by ChEMBL
Affinity DataIC50: 9.04E+4nMAssay Description:Inhibition of Trypanosoma cruzi recombinant trypanothione reductaseMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity against VDR-LBD (unknown origin) expressed in Escherichia coli assessed as inhibition of VDR agonist LG190178-induced SRC2-3 coac...More data for this Ligand-Target Pair
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity against VP16 tagged-VDR-LBD (unknown origin) expressed in HEK293T cells assessed as inhibition of 1,25-dihydroxyvitamin D3-induce...More data for this Ligand-Target Pair
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity against VP16 tagged-VDR-LBD (unknown origin) expressed in HEK293T cells assessed as inhibition of 1,25-dihydroxyvitamin D3-induce...More data for this Ligand-Target Pair
Affinity DataIC50: >1.50E+5nMAssay Description:Agonist activity at human VP16 tagged-VDR-LBD after 16 hrs by luciferase reporter gene based transcription assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.50E+5nMAssay Description:Agonist activity at VP16 tagged-VDR-LBD (unknown origin) expressed in HEK293T cells assessed as SRC1 coactivator peptide recruitment after 16 hrs by ...More data for this Ligand-Target Pair
Affinity DataIC50: >1.50E+5nMAssay Description:Agonist activity at VDR-LBD (unknown origin) expressed in Escherichia coli assessed as SRC2-3 coactivator peptide recruitment after 30 mins by fluore...More data for this Ligand-Target Pair
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity against VP16 tagged-VDR-LBD (unknown origin) expressed in HEK293T cells assessed as inhibition of 1,25-dihydroxyvitamin D3-induce...More data for this Ligand-Target Pair
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity against VP16 tagged-VDR-LBD (unknown origin) expressed in HEK293T cells assessed as inhibition of 1,25-dihydroxyvitamin D3-induce...More data for this Ligand-Target Pair
Affinity DataIC50: >1.50E+5nMAssay Description:Agonist activity at VDR-LBD (unknown origin) expressed in Escherichia coli assessed as SRC2-3 coactivator peptide recruitment after 30 mins by fluore...More data for this Ligand-Target Pair
Affinity DataIC50: >1.50E+5nMAssay Description:Agonist activity at VDR-LBD (unknown origin) expressed in Escherichia coli assessed as SRC2-3 coactivator peptide recruitment after 30 mins by fluore...More data for this Ligand-Target Pair
Affinity DataEC50: 1.49E+3nMAssay Description:Agonist activity at VP16 tagged-VDR-LBD (unknown origin) expressed in HEK293T cells assessed as SRC1 coactivator peptide recruitment after 16 hrs by ...More data for this Ligand-Target Pair
Affinity DataEC50: >1.50E+5nMAssay Description:Agonist activity at VP16 tagged-VDR-LBD (unknown origin) expressed in HEK293T cells assessed as SRC1 coactivator peptide recruitment after 16 hrs by ...More data for this Ligand-Target Pair
Affinity DataEC50: >1.50E+5nMAssay Description:Agonist activity at VP16 tagged-VDR-LBD (unknown origin) expressed in HEK293T cells assessed as SRC1 coactivator peptide recruitment after 16 hrs by ...More data for this Ligand-Target Pair
Affinity DataEC50: >1.50E+5nMAssay Description:Antagonist activity against VDR-LBD (unknown origin) expressed in Escherichia coli assessed as inhibition of VDR agonist LG190178-induced SRC2-3 coac...More data for this Ligand-Target Pair
Affinity DataEC50: 2.05E+4nMAssay Description:Antagonist activity against VDR-LBD (unknown origin) expressed in Escherichia coli assessed as inhibition of VDR agonist LG190178-induced SRC2-3 coac...More data for this Ligand-Target Pair
Affinity DataEC50: >1.50E+5nMAssay Description:Antagonist activity against VDR-LBD (unknown origin) expressed in Escherichia coli assessed as inhibition of VDR agonist LG190178-induced SRC2-3 coac...More data for this Ligand-Target Pair