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Found 83 with Last Name = 'sartor' and Initial = 'm'
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50359481(CHEMBL1926899)
Affinity DataIC50:  0.0900nMAssay Description:Antagonist activity against human CCR5 assessed as inhibition of HIV1 gp120-induced cell-cell fusion between human HeLa P4/R5 cells and CHO-tat10 cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50359487(CHEMBL1926893)
Affinity DataIC50:  0.200nMAssay Description:Antagonist activity against human CCR5 assessed as inhibition of HIV1 gp120-induced cell-cell fusion between human HeLa P4/R5 cells and CHO-tat10 cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50359482(CHEMBL1926898)
Affinity DataIC50:  0.300nMAssay Description:Antagonist activity against human CCR5 assessed as inhibition of HIV1 gp120-induced cell-cell fusion between human HeLa P4/R5 cells and CHO-tat10 cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50359478(CHEMBL1927009)
Affinity DataIC50:  0.300nMAssay Description:Antagonist activity against human CCR5 assessed as inhibition of HIV1 gp120-induced cell-cell fusion between human HeLa P4/R5 cells and CHO-tat10 cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50359459(CHEMBL1927008)
Affinity DataIC50:  0.300nMAssay Description:Antagonist activity against human CCR5 assessed as inhibition of HIV1 gp120-induced cell-cell fusion between human HeLa P4/R5 cells and CHO-tat10 cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50359485(CHEMBL1926896)
Affinity DataIC50:  0.300nMAssay Description:Antagonist activity against human CCR5 assessed as inhibition of HIV1 gp120-induced cell-cell fusion between human HeLa P4/R5 cells and CHO-tat10 cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50359480(CHEMBL1926900)
Affinity DataIC50:  0.600nMAssay Description:Antagonist activity against human CCR5 assessed as inhibition of HIV1 gp120-induced cell-cell fusion between human HeLa P4/R5 cells and CHO-tat10 cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50359479(CHEMBL1927010)
Affinity DataIC50:  0.700nMAssay Description:Antagonist activity against human CCR5 assessed as inhibition of HIV1 gp120-induced cell-cell fusion between human HeLa P4/R5 cells and CHO-tat10 cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50359489(CHEMBL1926891)
Affinity DataIC50:  0.700nMAssay Description:Antagonist activity against human CCR5 assessed as inhibition of HIV1 gp120-induced cell-cell fusion between human HeLa P4/R5 cells and CHO-tat10 cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50359464(CHEMBL1926901)
Affinity DataIC50:  0.800nMAssay Description:Antagonist activity against human CCR5 assessed as inhibition of HIV1 gp120-induced cell-cell fusion between human HeLa P4/R5 cells and CHO-tat10 cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50359461(CHEMBL1926904)
Affinity DataIC50:  0.980nMAssay Description:Antagonist activity against human CCR5 assessed as inhibition of HIV1 gp120-induced cell-cell fusion between human HeLa P4/R5 cells and CHO-tat10 cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50359463(CHEMBL1926902)
Affinity DataIC50:  1.30nMAssay Description:Antagonist activity against human CCR5 assessed as inhibition of HIV1 gp120-induced cell-cell fusion between human HeLa P4/R5 cells and CHO-tat10 cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50359486(CHEMBL1926894)
Affinity DataIC50:  1.5nMAssay Description:Antagonist activity against human CCR5 assessed as inhibition of HIV1 gp120-induced cell-cell fusion between human HeLa P4/R5 cells and CHO-tat10 cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50359483(CHEMBL1926897)
Affinity DataIC50:  1.60nMAssay Description:Antagonist activity against human CCR5 assessed as inhibition of HIV1 gp120-induced cell-cell fusion between human HeLa P4/R5 cells and CHO-tat10 cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50359466(CHEMBL1926885)
Affinity DataIC50:  2nMAssay Description:Antagonist activity against human CCR5 assessed as inhibition of HIV1 gp120-induced cell-cell fusion between human HeLa P4/R5 cells and CHO-tat10 cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50359490(CHEMBL1926890)
Affinity DataIC50:  2.40nMAssay Description:Antagonist activity against human CCR5 assessed as inhibition of HIV1 gp120-induced cell-cell fusion between human HeLa P4/R5 cells and CHO-tat10 cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50359467(CHEMBL1926884)
Affinity DataIC50:  3nMAssay Description:Antagonist activity against human CCR5 assessed as inhibition of HIV1 gp120-induced cell-cell fusion between human HeLa P4/R5 cells and CHO-tat10 cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50359465(CHEMBL1926886)
Affinity DataIC50:  3nMAssay Description:Antagonist activity against human CCR5 assessed as inhibition of HIV1 gp120-induced cell-cell fusion between human HeLa P4/R5 cells and CHO-tat10 cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50359460(CHEMBL1926905)
Affinity DataIC50:  7nMAssay Description:Antagonist activity against human CCR5 assessed as inhibition of HIV1 gp120-induced cell-cell fusion between human HeLa P4/R5 cells and CHO-tat10 cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50359491(CHEMBL1926889)
Affinity DataIC50:  7nMAssay Description:Antagonist activity against human CCR5 assessed as inhibition of HIV1 gp120-induced cell-cell fusion between human HeLa P4/R5 cells and CHO-tat10 cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50337581(CHEMBL1682993 | rac-N1-(1-(4-Methylpyridin-2-yl)et...)
Affinity DataIC50:  8nMAssay Description:Antagonist activity at CXCR4 in human CEM-CCRF cells assessed as inhibition of SDF-1-induced calcium signalingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50359468(CHEMBL1926883)
Affinity DataIC50:  8nMAssay Description:Antagonist activity against human CCR5 assessed as inhibition of HIV1 gp120-induced cell-cell fusion between human HeLa P4/R5 cells and CHO-tat10 cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50337584((S)-N1-((3-aminopyridin-2-yl)methyl)-N1-(5,6,7,8-t...)
Affinity DataIC50:  10.9nMAssay Description:Displacement of [125I]SDF-1alpha from CXCR4 in human CEM-CCRF cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50359492(CHEMBL1926888)
Affinity DataIC50:  10.9nMAssay Description:Antagonist activity against human CCR5 assessed as inhibition of HIV1 gp120-induced cell-cell fusion between human HeLa P4/R5 cells and CHO-tat10 cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50359471(CHEMBL1926878)
Affinity DataIC50:  11nMAssay Description:Antagonist activity against human CCR5 assessed as inhibition of HIV1 gp120-induced cell-cell fusion between human HeLa P4/R5 cells and CHO-tat10 cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50359493(CHEMBL1926887)
Affinity DataIC50:  12nMAssay Description:Antagonist activity against human CCR5 assessed as inhibition of HIV1 gp120-induced cell-cell fusion between human HeLa P4/R5 cells and CHO-tat10 cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50359488(CHEMBL1926892)
Affinity DataIC50:  12.3nMAssay Description:Antagonist activity against human CCR5 assessed as inhibition of HIV1 gp120-induced cell-cell fusion between human HeLa P4/R5 cells and CHO-tat10 cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50337585((S)-N1-((1H-benzo[d]imidazol-2-yl)methyl)-N1-(1-(p...)
Affinity DataIC50:  16.6nMAssay Description:Displacement of [125I]SDF-1alpha from CXCR4 in human CEM-CCRF cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50337577(CHEMBL1682989 | rac-N1-(3-iso-Butylpyridin-2-ylmet...)
Affinity DataIC50:  18nMAssay Description:Antagonist activity at CXCR4 in human CEM-CCRF cells assessed as inhibition of SDF-1-induced calcium signalingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50337561(CHEMBL1682854 | rac-N1-(3-methylpyridin-2-ylmethyl...)
Affinity DataIC50:  18nMAssay Description:Antagonist activity at CXCR4 in human CEM-CCRF cells assessed as inhibition of SDF-1-induced calcium signalingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50359474(CHEMBL1926875)
Affinity DataIC50:  19nMAssay Description:Antagonist activity against human CCR5 assessed as inhibition of HIV1 gp120-induced cell-cell fusion between human HeLa P4/R5 cells and CHO-tat10 cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50337566(CHEMBL1682859 | rac-N'-(3,5-Dimethylpyridin-2-ylme...)
Affinity DataIC50:  19nMAssay Description:Antagonist activity at CXCR4 in human CEM-CCRF cells assessed as inhibition of SDF-1-induced calcium signalingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50337580(CHEMBL1682992 | rac-N1-(3,5-dimethylpyridin-2-ylme...)
Affinity DataIC50:  20nMAssay Description:Antagonist activity at CXCR4 in human CEM-CCRF cells assessed as inhibition of SDF-1-induced calcium signalingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50337574(CHEMBL1682986 | racN1-(3-Methylpyridin-2-ylmethyl)...)
Affinity DataIC50:  23nMAssay Description:Antagonist activity at CXCR4 in human CEM-CCRF cells assessed as inhibition of SDF-1-induced calcium signalingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50359475(CHEMBL1926874)
Affinity DataIC50:  26nMAssay Description:Antagonist activity against human CCR5 assessed as inhibition of HIV1 gp120-induced cell-cell fusion between human HeLa P4/R5 cells and CHO-tat10 cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50337570(CHEMBL1682863 | rac-N1-(3-Aminopyridin-2-ylmethyl)...)
Affinity DataIC50:  27nMAssay Description:Antagonist activity at CXCR4 in human CEM-CCRF cells assessed as inhibition of SDF-1-induced calcium signalingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50359470(CHEMBL1926880)
Affinity DataIC50:  30nMAssay Description:Antagonist activity against human CCR5 assessed as inhibition of HIV1 gp120-induced cell-cell fusion between human HeLa P4/R5 cells and CHO-tat10 cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50359477(CHEMBL1926872)
Affinity DataIC50:  34nMAssay Description:Antagonist activity against human CCR5 assessed as inhibition of HIV1 gp120-induced cell-cell fusion between human HeLa P4/R5 cells and CHO-tat10 cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50337563(CHEMBL1682856 | rac-N1-(4-Methylpyridin-2-ylmethyl...)
Affinity DataIC50:  35nMAssay Description:Antagonist activity at CXCR4 in human CEM-CCRF cells assessed as inhibition of SDF-1-induced calcium signalingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50337586((S)-N1-((3-methylpyridin-2-yl)methyl)-N1-(1-(pyrid...)
Affinity DataIC50:  35.8nMAssay Description:Displacement of [125I]SDF-1alpha from CXCR4 in human CEM-CCRF cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50337565(CHEMBL1682858 | rac-N1-((4,6-dimethylpyridin-2-yl)...)
Affinity DataIC50:  38nMAssay Description:Antagonist activity at CXCR4 in human CEM-CCRF cells assessed as inhibition of SDF-1-induced calcium signalingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50359484(CHEMBL1926895)
Affinity DataIC50:  40nMAssay Description:Antagonist activity against human CCR5 assessed as inhibition of HIV1 gp120-induced cell-cell fusion between human HeLa P4/R5 cells and CHO-tat10 cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50337573(CHEMBL1682866 | racN1-(3-chloropyridin-2-ylmethyl)...)
Affinity DataIC50:  44nMAssay Description:Antagonist activity at CXCR4 in human CEM-CCRF cells assessed as inhibition of SDF-1-induced calcium signalingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50337567(CHEMBL1682860 | rac-N1-(6-aminopyridin-2-ylmethyl)...)
Affinity DataIC50:  49nMAssay Description:Antagonist activity at CXCR4 in human CEM-CCRF cells assessed as inhibition of SDF-1-induced calcium signalingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50339967(CHEMBL1762313 | N-(3-(4-(benzyl(4-bromophenyl)amin...)
Affinity DataIC50:  49nMAssay Description:Antagonist activity against human CCR5 assessed as inhibition of HIV1 gp120-induced cell-cell fusion between human HeLa P4/R5 cells and CHO-tat10 cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50359476(CHEMBL1926873)
Affinity DataIC50:  50nMAssay Description:Antagonist activity against human CCR5 assessed as inhibition of HIV1 gp120-induced cell-cell fusion between human HeLa P4/R5 cells and CHO-tat10 cel...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50337564(CHEMBL1682857 | rac-N1-(6-Methylpyridin-2-ylmethyl...)
Affinity DataIC50:  53nMAssay Description:Antagonist activity at CXCR4 in human CEM-CCRF cells assessed as inhibition of SDF-1-induced calcium signalingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50337583((S)-N1-((3,5-dimethylpyridin-2-yl)methyl)-N1-(5,6,...)
Affinity DataIC50:  62.9nMAssay Description:Displacement of [125I]SDF-1alpha from CXCR4 in human CEM-CCRF cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50337571(CHEMBL1682864 | rac-N1-(3-isopropylpyridin-2-ylmet...)
Affinity DataIC50:  63nMAssay Description:Antagonist activity at CXCR4 in human CEM-CCRF cells assessed as inhibition of SDF-1-induced calcium signalingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50337578(CHEMBL1682990 | rac-N1-((5-methylpyridin-2-yl)meth...)
Affinity DataIC50:  66nMAssay Description:Antagonist activity at CXCR4 in human CEM-CCRF cells assessed as inhibition of SDF-1-induced calcium signalingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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