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Found 12 with Last Name = 'savinov' and Initial = 'sn'
TargetProtein Mdm4(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50327206((2S,5S,8S,11S,14S,17S,20S,23S,26S,29S)-11-((1H-ind...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of GST-tagged p53 binding to MDMX by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50327206((2S,5S,8S,11S,14S,17S,20S,23S,26S,29S)-11-((1H-ind...)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of GST-tagged p53 binding to Hdm2 by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50327208(CHEMBL1256053 | tert-butyl (S)-1-((S)-1-((S)-3-(1H...)
Affinity DataIC50:  1.92E+5nMAssay Description:Inhibition of GST-tagged p53 binding to MDMX by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50327213((3S,6S,9S,12S,15S,18S)-3-benzyl-6-sec-butyl-15,18-...)
Affinity DataIC50:  2.09E+5nMAssay Description:Inhibition of GST-tagged p53 binding to Hdm2 by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50327210(CHEMBL1256067 | isobutyl (6S,9S,12S)-9-((1H-indol-...)
Affinity DataIC50:  3.00E+5nMAssay Description:Inhibition of GST-tagged p53 binding to MDMX by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50327209((4S,7S,10S)-7-((1H-indol-3-yl)methyl)-15-amino-4-b...)
Affinity DataIC50:  3.07E+5nMAssay Description:Inhibition of GST-tagged p53 binding to MDMX by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50327211(CHEMBL1256064 | tert-butyl (6S,9S,12S)-9-((1H-indo...)
Affinity DataIC50:  3.39E+5nMAssay Description:Inhibition of GST-tagged p53 binding to MDMX by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50327212(CHEMBL1256044 | benzyl (6S,9S,12S)-9-((1H-indol-3-...)
Affinity DataIC50:  3.48E+5nMAssay Description:Inhibition of GST-tagged p53 binding to MDMX by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50327207(((S)-5-((S)-3-(1H-indol-3-yl)-1-oxo-1-((S)-1-oxo-3...)
Affinity DataIC50:  4.63E+5nMAssay Description:Inhibition of GST-tagged p53 binding to MDMX by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50327206((2S,5S,8S,11S,14S,17S,20S,23S,26S,29S)-11-((1H-ind...)
Affinity DataKd:  75nMAssay Description:Binding affinity to Hdm2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Mdm4(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50327206((2S,5S,8S,11S,14S,17S,20S,23S,26S,29S)-11-((1H-ind...)
Affinity DataKd:  390nMAssay Description:Binding affinity to MDMXMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50327206((2S,5S,8S,11S,14S,17S,20S,23S,26S,29S)-11-((1H-ind...)
Affinity DataKd:  75nMAssay Description:Binding affinity to Hdm2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed