TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Academic Hospital Vrije Universiteit
Curated by ChEMBL
Academic Hospital Vrije Universiteit
Curated by ChEMBL
Affinity DataKi: 950nMAssay Description:TP_TRANSPORTER: inhibition of DNP-SG uptake in membrane vesicles from GLC4/ADR cellsMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family C member 5(Homo sapiens (Human))
The Netherlands Cancer Institute
Curated by ChEMBL
The Netherlands Cancer Institute
Curated by ChEMBL
Affinity DataIC50: <1.00E+5nMAssay Description:TP_TRANSPORTER: inhibition of PMEA efflux (PMEA: 1 uM) in MRP5-expressing MDCKII cellsMore data for this Ligand-Target Pair