Compile Data Set for Download or QSAR
maximum 50k data
Found 30 with Last Name = 'schipper' and Initial = 'j'
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Duphar

Curated by PDSP Ki Database
LigandPNGBDBM50035057((eltoprazine)1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)...)
Affinity DataKi:  40nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Duphar

Curated by PDSP Ki Database
LigandPNGBDBM50035057((eltoprazine)1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)...)
Affinity DataKi:  52nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50035057((eltoprazine)1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)...)
Affinity DataKi:  81nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine 1D receptor(Bos taurus (Bovine))
Duphar

Curated by PDSP Ki Database
LigandPNGBDBM50035057((eltoprazine)1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)...)
Affinity DataKi:  390nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Duphar

Curated by PDSP Ki Database
LigandPNGBDBM50035057((eltoprazine)1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)...)
Affinity DataKi:  420nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Duphar

Curated by PDSP Ki Database
LigandPNGBDBM50035057((eltoprazine)1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)...)
Affinity DataKi:  790nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Duphar

Curated by PDSP Ki Database
LigandPNGBDBM50035057((eltoprazine)1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)...)
Affinity DataKi:  1.10E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Mus musculus (house mouse))
Duphar

Curated by PDSP Ki Database
LigandPNGBDBM50035057((eltoprazine)1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)...)
Affinity DataKi:  1.30E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Duphar

Curated by PDSP Ki Database
LigandPNGBDBM50035057((eltoprazine)1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)...)
Affinity DataKi:  1.70E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50035057((eltoprazine)1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)...)
Affinity DataKi:  3.10E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(RAT)
Duphar

Curated by PDSP Ki Database
LigandPNGBDBM50035057((eltoprazine)1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)...)
Affinity DataKi:  3.90E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50035057((eltoprazine)1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)...)
Affinity DataKi:  9.30E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50035057((eltoprazine)1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Duphar

Curated by PDSP Ki Database
LigandPNGBDBM50035057((eltoprazine)1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Duphar

Curated by PDSP Ki Database
LigandPNGBDBM50035057((eltoprazine)1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Duphar

Curated by PDSP Ki Database
LigandPNGBDBM50035057((eltoprazine)1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtachykinin-1(RAT)
Duphar

Curated by PDSP Ki Database
LigandPNGBDBM50035057((eltoprazine)1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Duphar

Curated by PDSP Ki Database
LigandPNGBDBM50035057((eltoprazine)1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50035057((eltoprazine)1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
Duphar

Curated by PDSP Ki Database
LigandPNGBDBM50035057((eltoprazine)1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Duphar

Curated by PDSP Ki Database
LigandPNGBDBM50035057((eltoprazine)1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50035057((eltoprazine)1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50035057((eltoprazine)1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50035057((eltoprazine)1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50035057((eltoprazine)1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50035057((eltoprazine)1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcium release-activated calcium channel protein 1(Homo sapiens (Human))
Duphar

Curated by PDSP Ki Database
LigandPNGBDBM50035057((eltoprazine)1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent calcium channel gamma-1 subunit(Homo sapiens (Human))
Duphar

Curated by PDSP Ki Database
LigandPNGBDBM50035057((eltoprazine)1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
Duphar

Curated by PDSP Ki Database
LigandPNGBDBM50035057((eltoprazine)1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50035057((eltoprazine)1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed