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Found 429 with Last Name = 'sundell' and Initial = 's'
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50035320((+/-)-8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[...)
Affinity DataKi:  0.200nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT as radioligand in CHO-cells (sc)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50035305((S)-8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[e]...)
Affinity DataKi:  0.200nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Mus musculus (Mouse))
University Of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50044238(CHEMBL63449 | S-(-)-1-(8-Dipropylamino-6,7,8,9-tet...)
Affinity DataKi:  0.200nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT as radioligand in CHO-cells (sc)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Mus musculus (Mouse))
University Of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50044237(CHEMBL65274 | R-(+)-1-(8-Dipropylamino-6,7,8,9-tet...)
Affinity DataKi:  0.200nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT as radioligand in CHO-cells (sc)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50035320((+/-)-8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[...)
Affinity DataKi:  0.200nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50035303((R)-8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[e]...)
Affinity DataKi:  0.200nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
University Centre For Pharmacy

Curated by ChEMBL
LigandPNGBDBM50020217((4aR,10bR)-4-propyl-3,4,4a,5,6,10b-hexahydro-2H-na...)
Affinity DataKi:  0.210nMAssay Description:Tested for antagonist binding affinity by measuring displacement of [3H]spiperone from Human Dopamine receptor D3 expressed in CHO K-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50035335((R)-8-Dipropylamino-4-fluoro-6,7,8,9-tetrahydro-3H...)
Affinity DataKi:  0.300nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50035326(8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[e]indo...)
Affinity DataKi:  0.400nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50036286((R)-(-)-10-methyl-11-hydroxyaporphine | (R)-6,10-d...)
Affinity DataKi:  0.450nMAssay Description:Ability to displace [3H]-8-OH-DPAT binding to rat hippocampal 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50035324((S)-8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[e]...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg

Curated by ChEMBL
LigandPNGBDBM21393(7-(dipropylamino)-5,6,7,8-tetrahydronaphthalen-1-o...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50035319(8-Dipropylamino-4-fluoro-6,7,8,9-tetrahydro-3H-ben...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50035328((R)-8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[e]...)
Affinity DataKi:  0.800nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50035315((S)-8-Dipropylamino-4-fluoro-6,7,8,9-tetrahydro-3H...)
Affinity DataKi:  0.800nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Centre For Pharmacy

Curated by ChEMBL
LigandPNGBDBM50090828((-)-1-Propyl-2,3,10,10a-tetrahydro-1H,4aH-4-oxa-9-...)
Affinity DataKi:  1.10nMAssay Description:Tested for agonist binding affinity by measuring displacement of [3H]NPA from Human Dopamine receptor D2L expressed in CHO K-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50035320((+/-)-8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[...)
Affinity DataKi:  1.30nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
University Centre For Pharmacy

Curated by ChEMBL
LigandPNGBDBM50010586((+)-1-Propyl-2,3,10,10a-tetrahydro-1H,4aH-4,9-diox...)
Affinity DataKi:  1.40nMAssay Description:Tested for antagonist binding affinity by measuring displacement of [3H]spiperone from Human Dopamine receptor D3 expressed in CHO K-1 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50035307(CHEMBL302171 | Dipropyl-(S)-6,7,8,9-tetrahydro-3H-...)
Affinity DataKi:  1.40nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
University Centre For Pharmacy

Curated by ChEMBL
LigandPNGBDBM50010586((+)-1-Propyl-2,3,10,10a-tetrahydro-1H,4aH-4,9-diox...)
Affinity DataKi:  1.40nMAssay Description:Tested for antagonist binding affinity by measuring displacement of [3H]spiperone from Human Dopamine receptor D3 expressed in CHO K-1 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50035304((4-Fluoro-6,7,8,9-tetrahydro-3H-benzo[e]indol-8-yl...)
Affinity DataKi:  1.40nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50044237(CHEMBL65274 | R-(+)-1-(8-Dipropylamino-6,7,8,9-tet...)
Affinity DataKi:  1.40nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50035317(((R)-4-Fluoro-6,7,8,9-tetrahydro-3H-benzo[e]indol-...)
Affinity DataKi:  1.5nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035304((4-Fluoro-6,7,8,9-tetrahydro-3H-benzo[e]indol-8-yl...)
Affinity DataKi:  1.60nMAssay Description:Binding affinity against Dopamine receptor D3 from CHO-K1 cells, using [3H]-spiperone as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
University Centre For Pharmacy

Curated by ChEMBL
LigandPNGBDBM50090829((trans)1-Propyl-2,3,10,10a-tetrahydro-1H,4aH-4-oxa...)
Affinity DataKi:  1.60nMAssay Description:Tested for antagonist binding affinity by measuring displacement of [3H]spiperone from Human Dopamine receptor D3 expressed in CHO K-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50035306((1-Chloro-6,7,8,9-tetrahydro-3H-benzo[e]indol-8-yl...)
Affinity DataKi:  2nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50044238(CHEMBL63449 | S-(-)-1-(8-Dipropylamino-6,7,8,9-tet...)
Affinity DataKi:  2nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50035313(8-Dipropylamino-4-fluoro-6,7,8,9-tetrahydro-3H-ben...)
Affinity DataKi:  2.30nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035304((4-Fluoro-6,7,8,9-tetrahydro-3H-benzo[e]indol-8-yl...)
Affinity DataKi:  2.80nMAssay Description:Binding affinity against Dopamine receptor D2 from CHO-K1 cells, using [3H]-U-86,170 as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
University Centre For Pharmacy

Curated by ChEMBL
LigandPNGBDBM50090828((-)-1-Propyl-2,3,10,10a-tetrahydro-1H,4aH-4-oxa-9-...)
Affinity DataKi:  2.90nMAssay Description:Tested for antagonist binding affinity by measuring displacement of [3H]spiperone from Human Dopamine receptor D3 expressed in CHO K-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50016777(((R)-8-Hydroxy-1,2,3,4-tetrahydro-naphthalen-2-yl)...)
Affinity DataKi:  3.10nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT (agonist) as radioligand (sc)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50035329((+/-)-Dipropyl-(6,7,8,9-tetrahydro-3H-benzo[e]indo...)
Affinity DataKi:  3.30nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
University Centre For Pharmacy

Curated by ChEMBL
LigandPNGBDBM50090832((cis)1-Propyl-2,3,10,10a-tetrahydro-1H,4aH-4-oxa-9...)
Affinity DataKi:  3.60nMAssay Description:Tested for antagonist binding affinity by measuring displacement of [3H]spiperone from Human Dopamine receptor D3 expressed in CHO K-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50035299(((S)-4-Fluoro-6,7,8,9-tetrahydro-3H-benzo[e]indol-...)
Affinity DataKi:  3.70nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035299(((S)-4-Fluoro-6,7,8,9-tetrahydro-3H-benzo[e]indol-...)
Affinity DataKi:  4.10nMAssay Description:Binding affinity against Dopamine receptor D3 from CHO-K1 cells, using [3H]-spiperone as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035299(((S)-4-Fluoro-6,7,8,9-tetrahydro-3H-benzo[e]indol-...)
Affinity DataKi:  4.40nMAssay Description:Binding affinity against Dopamine receptor D2 from CHO-K1 cells, using [3H]-U-86,170 as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035335((R)-8-Dipropylamino-4-fluoro-6,7,8,9-tetrahydro-3H...)
Affinity DataKi:  4.40nMAssay Description:Binding affinity against 5-hydroxytryptamine 1D receptor alpha expressed in CHO-K1 cells, using [3H]-5-HT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035319(8-Dipropylamino-4-fluoro-6,7,8,9-tetrahydro-3H-ben...)
Affinity DataKi:  4.60nMAssay Description:Binding affinity against 5-hydroxytryptamine 1D receptor alpha expressed in CHO-K1 cells, using [3H]-5-HT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50035330(CHEMBL302172 | Dipropyl-(R)-6,7,8,9-tetrahydro-3H-...)
Affinity DataKi:  5.20nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035325((4-Fluoro-1-propyl-6,7,8,9-tetrahydro-3H-benzo[e]i...)
Affinity DataKi:  5.90nMAssay Description:Binding affinity against Dopamine receptor D2 from CHO-K1 cells, using [3H]-U-86,170 as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Centre For Pharmacy

Curated by ChEMBL
LigandPNGBDBM50020217((4aR,10bR)-4-propyl-3,4,4a,5,6,10b-hexahydro-2H-na...)
Affinity DataKi:  6.20nMAssay Description:Human Dopamine receptor D2L affinities to determine agonist activity, using [3H]spip as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035328((R)-8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[e]...)
Affinity DataKi:  6.70nMAssay Description:Binding affinity against 5-hydroxytryptamine 1D receptor alpha expressed in CHO-K1 cells, using [3H]-5-HT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50035330(CHEMBL302172 | Dipropyl-(R)-6,7,8,9-tetrahydro-3H-...)
Affinity DataKi:  7nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50035300(1-(8-Dipropylamino-4-fluoro-6,7,8,9-tetrahydro-3H-...)
Affinity DataKi:  7.10nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50035322(2-(8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[e]i...)
Affinity DataKi:  7.30nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035330(CHEMBL302172 | Dipropyl-(R)-6,7,8,9-tetrahydro-3H-...)
Affinity DataKi:  7.40nMAssay Description:Binding affinity against Dopamine receptor D2 expressed in CHO-K1 cells, using [3H]-U-86,170 as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035326(8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[e]indo...)
Affinity DataKi:  7.5nMAssay Description:Binding affinity against 5-hydroxytryptamine 1D receptor alpha expressed in CHO-K1 cells, using [3H]-5-HT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035317(((R)-4-Fluoro-6,7,8,9-tetrahydro-3H-benzo[e]indol-...)
Affinity DataKi:  7.80nMAssay Description:Binding affinity against Dopamine receptor D2 from CHO-K1 cells, using [3H]-U-86,170 as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50011247(7-Dipropylamino-5,6,7,8-tetrahydro-naphthalen-1-ol...)
Affinity DataKi:  8.40nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035325((4-Fluoro-1-propyl-6,7,8,9-tetrahydro-3H-benzo[e]i...)
Affinity DataKi:  8.40nMAssay Description:Binding affinity against 5-hydroxytryptamine 1D receptor alpha expressed in CHO-K1 cells, using [3H]-5-HT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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