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Found 7 with Last Name = 'takahashi' and Initial = 'js'
TargetNuclear receptor subfamily 1 group D member 2(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50366239(CHEMBL1961797)
Affinity DataIC50:  560nMAssay Description:Increased REV-ERB-beta LBD dependent repressor activity in HEK293 cell reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50366239(CHEMBL1961797)
Affinity DataIC50:  620nMAssay Description:REV-ERB-alpha mediated transcriptional suppression at Bmal1 promoter in HEK293 cell reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50366238(CHEMBL1961796)
Affinity DataIC50:  670nMAssay Description:Increased REV-ERB-alpha LBD dependent repressor activity in HEK293 cell reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50366238(CHEMBL1961796)
Affinity DataIC50:  710nMAssay Description:REV-ERB-alpha mediated transcriptional suppression at Bmal1 promoter in HEK293 cell reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50366239(CHEMBL1961797)
Affinity DataIC50:  790nMAssay Description:Increased REV-ERB-alpha LBD dependent repressor activity in HEK293 cell reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 2(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50366238(CHEMBL1961796)
Affinity DataIC50:  800nMAssay Description:Increased REV-ERB-beta LBD dependent repressor activity in HEK293 cell reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group D member 1(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50366238(CHEMBL1961796)
Affinity DataKd:  800nMAssay Description:Dissociation constant for binding to REV-ERB-alpha by circular dichroismMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed