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Found 1243 with Last Name = 'takahashi' and Initial = 'm'
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50149389(1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-p...)
Affinity DataKi:  0.110nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50149381(1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-p...)
Affinity DataKi:  0.120nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50149398(1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-p...)
Affinity DataKi:  0.130nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50149384((S)-1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)
Affinity DataKi:  0.150nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50149396(1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-p...)
Affinity DataKi:  0.170nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50149375(1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-p...)
Affinity DataKi:  0.190nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50149374(1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-p...)
Affinity DataKi:  0.220nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50149394(1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-p...)
Affinity DataKi:  0.290nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50149386(1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-p...)
Affinity DataKi:  0.330nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50149378(1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-p...)
Affinity DataKi:  0.360nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50149382(1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-p...)
Affinity DataKi:  0.490nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50149385((S)-1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)
Affinity DataKi:  0.510nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50149376(1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-p...)
Affinity DataKi:  0.520nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)
Affinity DataKi:  0.690nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50149391(1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-p...)
Affinity DataKi:  1.10nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50149377(1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyr...)
Affinity DataKi:  2.40nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50127501(3-(4-Carbamimidoyl-2-{2-[4-(pyrrolidine-1-carbonyl...)
Affinity DataKi:  3nMAssay Description:Inhibitory activity against Coagulation factor X (fXa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50149402(1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyr...)
Affinity DataKi:  4.10nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50149397(1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyr...)
Affinity DataKi:  5.80nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50149379(1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyr...)
Affinity DataKi:  6.60nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50127492(4-[5-Carbamimidoyl-2-(2-carboxy-2-oxo-ethyl)-pheno...)
Affinity DataKi:  11nMAssay Description:Inhibitory activity against Coagulation factor X (fXa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50149399((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)
Affinity DataKi:  13nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50149376(1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-p...)
Affinity DataKi:  14nMAssay Description:Binding affinity against rat brain opioid receptor delta 1 using [3H]-DPDPE radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50149385((S)-1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)
Affinity DataKi:  18nMAssay Description:Binding affinity against rat brain opioid receptor delta 1 using [3H]-DPDPE radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50127502(4-[5-Carbamimidoyl-2-(2-carboxy-2-oxo-ethyl)-pheno...)
Affinity DataKi:  18nMAssay Description:Inhibitory activity against Coagulation factor X (fXa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50149394(1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-p...)
Affinity DataKi:  20nMAssay Description:Binding affinity against rat brain opioid receptor delta 1 using [3H]-DPDPE radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50127495(3-[4-Carbamimidoyl-2-(2-{4-[1-(1-imino-ethyl)-pipe...)
Affinity DataKi:  20nMAssay Description:Inhibitory activity against Coagulation factor X (fXa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50127504(CHEMBL55770 | N-[2-(3-Carbamimidoyl-phenoxy)-ethyl...)
Affinity DataKi:  20nMAssay Description:Inhibitory activity against Coagulation factor X (fXa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50149383(1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyr...)
Affinity DataKi:  20nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50149391(1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-p...)
Affinity DataKi:  21nMAssay Description:Binding affinity against rat brain opioid receptor delta 1 using [3H]-DPDPE radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50127494(3-(4-Carbamimidoyl-2-{2-[(3,4,5,6-tetrahydro-2H-[1...)
Affinity DataKi:  21nMAssay Description:Inhibitory activity against Coagulation factor X (fXa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50149404(1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyr...)
Affinity DataKi:  22nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50149400((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)
Affinity DataKi:  24nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50127498(3-{4-Carbamimidoyl-2-[2-(4-carbamimidoyl-benzoylam...)
Affinity DataKi:  26nMAssay Description:Inhibitory activity against Coagulation factor X (fXa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50149388(1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyr...)
Affinity DataKi:  27nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50127503(3-(4-Carbamimidoyl-benzoylamino)-4-(3-carbamimidoy...)
Affinity DataKi:  28nMAssay Description:Inhibitory activity against Coagulation factor X (fXa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50149384((S)-1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)
Affinity DataKi:  28nMAssay Description:Binding affinity against rat brain opioid receptor delta 1 using [3H]-DPDPE radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50149389(1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-p...)
Affinity DataKi:  30nMAssay Description:Binding affinity against rat brain opioid receptor delta 1 using [3H]-DPDPE radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50149382(1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-p...)
Affinity DataKi:  33nMAssay Description:Binding affinity against rat brain opioid receptor delta 1 using [3H]-DPDPE radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50149403(1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyr...)
Affinity DataKi:  34nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50127493(3-(4-Carbamimidoyl-2-{2-[(3,4,5,6-tetrahydro-2H-[1...)
Affinity DataKi:  43nMAssay Description:Inhibitory activity against Coagulation factor X (fXa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50149380(1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyr...)
Affinity DataKi:  46nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50149374(1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-p...)
Affinity DataKi:  47nMAssay Description:Binding affinity against rat brain opioid receptor delta 1 using [3H]-DPDPE radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50149390(1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyr...)
Affinity DataKi:  48nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50149401(1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyr...)
Affinity DataKi:  49nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50149381(1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-p...)
Affinity DataKi:  53nMAssay Description:Binding affinity against rat brain opioid receptor delta 1 using [3H]-DPDPE radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50149378(1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-p...)
Affinity DataKi:  53nMAssay Description:Binding affinity against rat brain opioid receptor delta 1 using [3H]-DPDPE radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50149387(1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyr...)
Affinity DataKi:  56nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50149395(1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyr...)
Affinity DataKi:  61nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50149393(1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyr...)
Affinity DataKi:  73nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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