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Found 14 with Last Name = 'taketa' and Initial = 'k'
TargetNeuromedin-U receptor 2(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50049421(CHEMBL3315349)
Affinity DataEC50:  2.5nMAssay Description:Agonist activity at human NMUR2 expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-U receptor 2(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50049422(CHEMBL3315335)
Affinity DataEC50:  6.40nMAssay Description:Agonist activity at human NMUR2 expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50049421(CHEMBL3315349)
Affinity DataEC50:  0.430nMAssay Description:Agonist activity at human NMUR1 expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-U receptor 2(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50049423(CHEMBL3315278)
Affinity DataEC50:  8.40nMAssay Description:Partial agonist activity at human NMUR2 expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50049424(CHEMBL3315348)
Affinity DataEC50:  2.20nMAssay Description:Partial agonist activity at human NMUR1 expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50049423(CHEMBL3315278)
Affinity DataEC50:  9nMAssay Description:Partial agonist activity at human NMUR1 expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50085928(CHEMBL3425593)
Affinity DataEC50:  0.0830nMAssay Description:Agonist activity at human NMUR1 expressed in CHO cells assessed as intracellular calcium flux at by Fluo-4 AM dye based fluorometric imaging methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-U receptor 1(Mus musculus)
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50049425(CHEMBL3356083)
Affinity DataEC50:  9.5nMAssay Description:Agonist activity at mouse NMUR1 expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-U receptor 1(Mus musculus)
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50049426(CHEMBL3356082)
Affinity DataEC50:  2.41E+3nMAssay Description:Agonist activity at mouse NMUR1 expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-U receptor 2(Mus musculus)
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50049426(CHEMBL3356082)
Affinity DataEC50:  156nMAssay Description:Agonist activity at mouse NMUR2 expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-U receptor 2(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50049421(CHEMBL3315349)
Affinity DataEC50:  0.920nMAssay Description:Agonist activity at human NMUR2 expressed in CHO cells assessed as intracellular calcium flux at by Fluo-4 AM dye based fluorometric imaging methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-U receptor 2(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50085928(CHEMBL3425593)
Affinity DataEC50:  2.60nMAssay Description:Agonist activity at human NMUR2 expressed in CHO cells assessed as intracellular calcium flux at by Fluo-4 AM dye based fluorometric imaging methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50049421(CHEMBL3315349)
Affinity DataEC50:  0.140nMAssay Description:Agonist activity at human NMUR1 expressed in CHO cells assessed as intracellular calcium flux at by Fluo-4 AM dye based fluorometric imaging methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-U receptor 2(Mus musculus)
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50049425(CHEMBL3356083)
Affinity DataEC50:  3nMAssay Description:Agonist activity at mouse NMUR2 expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed