TargetAdenosine receptor A3(Homo sapiens (Human))
Merck Research Laboratories
Curated by PDSP Ki Database
Merck Research Laboratories
Curated by PDSP Ki Database
TargetAdenosine receptor A3(Homo sapiens (Human))
Merck Research Laboratories
Curated by PDSP Ki Database
Merck Research Laboratories
Curated by PDSP Ki Database
TargetAdenosine receptor A3(Homo sapiens (Human))
Merck Research Laboratories
Curated by PDSP Ki Database
Merck Research Laboratories
Curated by PDSP Ki Database
TargetAdenosine receptor A3(Homo sapiens (Human))
Merck Research Laboratories
Curated by PDSP Ki Database
Merck Research Laboratories
Curated by PDSP Ki Database
TargetAdenosine receptor A3(Homo sapiens (Human))
Merck Research Laboratories
Curated by PDSP Ki Database
Merck Research Laboratories
Curated by PDSP Ki Database
TargetAdenosine receptor A3(Homo sapiens (Human))
Merck Research Laboratories
Curated by PDSP Ki Database
Merck Research Laboratories
Curated by PDSP Ki Database
TargetAdenosine receptor A3(Homo sapiens (Human))
Merck Research Laboratories
Curated by PDSP Ki Database
Merck Research Laboratories
Curated by PDSP Ki Database
TargetAdenosine receptor A3(Homo sapiens (Human))
Merck Research Laboratories
Curated by PDSP Ki Database
Merck Research Laboratories
Curated by PDSP Ki Database
Affinity DataIC50: 1nMAssay Description:Inhibition of influenza A sialidase (neuraminidase)More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of influenza A sialidase (neuraminidase)More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of influenza A sialidase (neuraminidase)More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of influenza A sialidase (neuraminidase)More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of influenza A sialidase (neuraminidase)More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of influenza A sialidase (neuraminidase)More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of influenza B sialidase (neuraminidase)More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of influenza A sialidase (neuraminidase)More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of influenza A sialidase (neuraminidase)More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of influenza A sialidase (neuraminidase)More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of influenza A sialidase (neuraminidase)More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of influenza A sialidase (neuraminidase)More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of influenza A sialidase (neuraminidase)More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Oxford
Curated by ChEMBL
University Of Oxford
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of rapid delayed inward rectifying potassium current (IKr) measured using manual patch clamp assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Oxford
Curated by ChEMBL
University Of Oxford
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of transient outward potassium current (Ito) current in Chinese Hamster Ovary (CHO) K1 cells expressing human Kv4.3 measured using IonWork...More data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibition of influenza A sialidase (neuraminidase)More data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibition of influenza A sialidase (neuraminidase)More data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Inhibition of influenza A sialidase (neuraminidase)More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Oxford
Curated by ChEMBL
University Of Oxford
Curated by ChEMBL
Affinity DataIC50: 79nMAssay Description:Inhibition of transient outward potassium current (Ito) current in Chinese Hamster Ovary (CHO) K1 cells expressing human Kv4.3 measured using IonWork...More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Oxford
Curated by ChEMBL
University Of Oxford
Curated by ChEMBL
Affinity DataIC50: 126nMAssay Description:Inhibition of rapid delayed inward rectifying potassium current (IKr) in Chinese hamster ovary (CHO) K1 cells stably expressing hERG measured using I...More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Oxford
Curated by ChEMBL
University Of Oxford
Curated by ChEMBL
Affinity DataIC50: 126nMAssay Description:Inhibition of slow delayed inward rectifying potassium current (Iks) in Chinese Hamster Ovary (CHO) cells expressing hKvLQT1/hminK measured using Ion...More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Oxford
Curated by ChEMBL
University Of Oxford
Curated by ChEMBL
Affinity DataIC50: 126nMAssay Description:Inhibition of rapid delayed inward rectifying potassium current (IKr) in Chinese hamster ovary (CHO) K1 cells stably expressing hERG measured using I...More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Oxford
Curated by ChEMBL
University Of Oxford
Curated by ChEMBL
Affinity DataIC50: 158nMAssay Description:Inhibition of slow delayed inward rectifying potassium current (Iks) in Chinese Hamster Ovary (CHO) cells expressing hKvLQT1/hminK measured using Ion...More data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Inhibition of influenza A sialidase (neuraminidase)More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Oxford
Curated by ChEMBL
University Of Oxford
Curated by ChEMBL
Affinity DataIC50: 251nMAssay Description:Inhibition of transient outward potassium current (Ito) current in Chinese Hamster Ovary (CHO) K1 cells expressing human Kv4.3 measured using IonWork...More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Oxford
Curated by ChEMBL
University Of Oxford
Curated by ChEMBL
Affinity DataIC50: 251nMAssay Description:Inhibition of slow delayed inward rectifying potassium current (Iks) in Chinese Hamster Ovary (CHO) cells expressing hKvLQT1/hminK measured using Ion...More data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of influenza A sialidase (neuraminidase)More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Oxford
Curated by ChEMBL
University Of Oxford
Curated by ChEMBL
Affinity DataIC50: 316nMAssay Description:Inhibition of rapid delayed inward rectifying potassium current (IKr) measured using manual patch clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: 320nMAssay Description:Inhibition of influenza A sialidase (neuraminidase)More data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibition of influenza B sialidase (neuraminidase)More data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibition of influenza B sialidase (neuraminidase)More data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibition of influenza B sialidase (neuraminidase)More data for this Ligand-Target Pair
Affinity DataIC50: 450nMAssay Description:Inhibition of influenza A sialidase (neuraminidase)More data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition of influenza B sialidase (neuraminidase)More data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition of influenza B sialidase (neuraminidase)More data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition of influenza A sialidase (neuraminidase)More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Oxford
Curated by ChEMBL
University Of Oxford
Curated by ChEMBL
Affinity DataIC50: 631nMAssay Description:Inhibition of rapid delayed inward rectifying potassium current (IKr) in Chinese hamster ovary (CHO) cells stable expressing hERG measured using IonW...More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Oxford
Curated by ChEMBL
University Of Oxford
Curated by ChEMBL
Affinity DataIC50: 631nMAssay Description:Inhibition of transient outward potassium current (Ito) current in Chinese Hamster Ovary (CHO) K1 cells expressing human Kv4.3 measured using IonWork...More data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Inhibition of influenza B sialidase (neuraminidase)More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of influenza B sialidase (neuraminidase)More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Oxford
Curated by ChEMBL
University Of Oxford
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rapid delayed inward rectifying potassium current (IKr) in Chinese hamster ovary (CHO) K1 cells stably expressing hERG measured using I...More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Oxford
Curated by ChEMBL
University Of Oxford
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of fast sodium current (INa) in HEK293 cells transfected with human Nav1.5 measured using IonWorks Quattro automated patch clamp platformMore data for this Ligand-Target Pair