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Found 52 with Last Name = 'teixeira' and Initial = 'n'
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50135997(CHEMBL3754471)
Affinity DataKi:  23nMAssay Description:Competitive irreversible inhibition of human placental microsome aromatase using varying levels of [1beta3H]-androstenedione as substrate measured af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50135997(CHEMBL3754471)
Affinity DataKi:  25nMAssay Description:Competitive reversible inhibition of human placental microsome aromatase using varying levels of [1beta3H]-androstenedione as substrate measured afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50398447(Aromasin | EXEMESTANE)
Affinity DataKi:  26nMAssay Description:Competitive inhibition of human placental microsome aromatase using varying levels of [1beta2beta3H]-androstenedione as substrateMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50332805((3R,4S,5R,8R,9S,10R,13S,14S)-10,13-Dimethyl-hexade...)
Affinity DataKi:  38nMAssay Description:Inhibition of aromatase in human microsomes using [1beta-3H]androstenedione as substrate after 5 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50174541((3R,4S,5R,10R,13S)-10,13-Dimethyl-hexadecahydro-20...)
Affinity DataKi:  38nMAssay Description:Inhibition constant against aromatase protein from human placental microsomes using [1-beta-3H]-androstenedione; Competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50332803((5S,8R,9S,10S,13S,14S)-10,13-dimethyl-5,6,7,8,9,10...)
Affinity DataKi:  50nMAssay Description:Inhibition of aromatase in human microsomes using [1beta-3H]androstenedione as substrate after 5 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50174544((5S,10S,13S)-10,13-Dimethyl-1,2,5,6,7,8,9,10,11,12...)
Affinity DataKi:  50nMAssay Description:Inhibition constant against aromatase protein from human placental microsomes using [1-beta-3H]-androstenedione; Competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50388393(CHEMBL2058266)
Affinity DataKi:  86nMAssay Description:Inhibition of aromatase in human microsomes using [1beta-3H]androstenedione as substrate after 5 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50388396(CHEMBL1077603)
Affinity DataKi:  100nMAssay Description:Inhibition of aromatase in human microsomes using [1beta-3H]androstenedione as substrate after 5 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50174543((3R,5R,10R,13S)-3-Hydroxy-10,13-dimethyl-tetradeca...)
Affinity DataKi:  147nMAssay Description:Inhibition constant against aromatase protein from human placental microsomes using [1-beta-3H]-androstenedione; Competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50174542((10aR,12aS)-7-Hydroxy-10a,12a-dimethyl-3,4,4a,5,6,...)
Affinity DataKi:  660nMAssay Description:Inhibition constant against aromatase protein from human placental microsomes using [1-beta-3H]-androstenedione; Competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50388394(CHEMBL2058267)
Affinity DataKi:  9.50E+3nMAssay Description:Inhibition of aromatase in human microsomes using [1beta-3H]androstenedione as substrate after 5 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50240798((8R,9S,10R,13S,14S)-4-Hydroxy-10,13-dimethyl-1,6,7...)
Affinity DataIC50:  42nMAssay Description:Inhibition of aromatase in human placental microsomes using [1beta-3H]androstenedione as substrate after 15 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50240798((8R,9S,10R,13S,14S)-4-Hydroxy-10,13-dimethyl-1,6,7...)
Affinity DataIC50:  42nMAssay Description:Inhibitory concentration against aromatase protein from human placental microsomes using [1-beta-3H]-androstenedione; Competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50398447(Aromasin | EXEMESTANE)
Affinity DataIC50:  50nMAssay Description:Inhibition of human placental microsome aromatase using [1beta-3H] androstenedione as substrate after 15 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50523404(CHEMBL4575994)
Affinity DataIC50:  55nMAssay Description:Inhibition of human placental microsome aromatase using [1beta3H]-androstenedione as substrate measured after 15 mins in presence of NADPH by liquid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50135997(CHEMBL3754471)
Affinity DataIC50:  60nMAssay Description:Inhibition of human placental microsome aromatase using [1beta3H]-androstenedione as substrate measured after 15 mins in presence of NADPH by liquid ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50069753(CHEMBL3407538)
Affinity DataIC50:  100nMAssay Description:Inhibition of human placental microsome aromatase using [1beta-3H] androstenedione as substrate after 15 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50523395(CHEMBL4514728)
Affinity DataIC50:  105nMAssay Description:Inhibition of human placental microsome aromatase using [1beta3H]-androstenedione as substrate measured after 15 mins in presence of NADPH by liquid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50168058(CHEMBL3798461)
Affinity DataIC50:  110nMAssay Description:Inhibition of aromatase in human placental microsomes using [1beta-3H]-androstenedione as substrate assessed as tritiated H2O release after 15 mins b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50523399(CHEMBL4454575)
Affinity DataIC50:  110nMAssay Description:Inhibition of human placental microsome aromatase using [1beta3H]-androstenedione as substrate measured after 15 mins in presence of NADPH by liquid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50332807((8R,9S,10R,13S,14S)-10,13-dimethyl-2,3,7,8,9,10,11...)
Affinity DataIC50:  135nMAssay Description:Inhibition of aromatase in human placental microsomes using [1beta-3H]androstenedione as substrate after 15 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50174541((3R,4S,5R,10R,13S)-10,13-Dimethyl-hexadecahydro-20...)
Affinity DataIC50:  145nMAssay Description:Inhibitory concentration against aromatase protein from human placental microsomes using [1-beta-3H]-androstenedione; Competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50332805((3R,4S,5R,8R,9S,10R,13S,14S)-10,13-Dimethyl-hexade...)
Affinity DataIC50:  145nMAssay Description:Inhibition of aromatase in human placental microsomes using [1beta-3H]androstenedione as substrate after 15 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50135862(CHEMBL3751881)
Affinity DataIC50:  170nMAssay Description:Inhibition of human placental microsome aromatase using [1beta3H]-androstenedione as substrate measured after 15 mins in presence of NADPH by liquid ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50523403(CHEMBL4460869)
Affinity DataIC50:  175nMAssay Description:Inhibition of human placental microsome aromatase using [1beta3H]-androstenedione as substrate measured after 15 mins in presence of NADPH by liquid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50388396(CHEMBL1077603)
Affinity DataIC50:  183nMAssay Description:Inhibition of aromatase in human placental microsomes using [1beta-3H]androstenedione as substrate after 15 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50523400(CHEMBL4520056)
Affinity DataIC50:  210nMAssay Description:Inhibition of human placental microsome aromatase using [1beta3H]-androstenedione as substrate measured after 15 mins in presence of NADPH by liquid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50332803((5S,8R,9S,10S,13S,14S)-10,13-dimethyl-5,6,7,8,9,10...)
Affinity DataIC50:  225nMAssay Description:Inhibition of aromatase in human placental microsomes using [1beta-3H]androstenedione as substrate after 15 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50174544((5S,10S,13S)-10,13-Dimethyl-1,2,5,6,7,8,9,10,11,12...)
Affinity DataIC50:  225nMAssay Description:Inhibitory concentration against aromatase protein from human placental microsomes using [1-beta-3H]-androstenedione; Competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50168056(CHEMBL3799363)
Affinity DataIC50:  250nMAssay Description:Inhibition of aromatase in human placental microsomes using [1beta-3H]-androstenedione as substrate assessed as tritiated H2O release after 15 mins b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50069753(CHEMBL3407538)
Affinity DataIC50:  250nMAssay Description:Inhibition of human placental microsome aromatase expressed in human MCF7 cells using [1beta-3H] androstenedione as substrate after 1 hr by liquid sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50523396(CHEMBL487113)
Affinity DataIC50:  270nMAssay Description:Inhibition of human placental microsome aromatase using [1beta3H]-androstenedione as substrate measured after 15 mins in presence of NADPH by liquid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50523397(CHEMBL4451962)
Affinity DataIC50:  405nMAssay Description:Inhibition of human placental microsome aromatase using [1beta3H]-androstenedione as substrate measured after 15 mins in presence of NADPH by liquid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50123151(CHEMBL3623223)
Affinity DataIC50:  470nMAssay Description:Inhibition of aromatase in human placental microsomes using [1beta-3H]-androstenedione as substrate assessed as tritiated H2O release after 15 mins b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50523402(CHEMBL4468497)
Affinity DataIC50:  520nMAssay Description:Inhibition of human placental microsome aromatase using [1beta3H]-androstenedione as substrate measured after 15 mins in presence of NADPH by liquid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50168057(CHEMBL3800417)
Affinity DataIC50:  530nMAssay Description:Inhibition of aromatase in human placental microsomes using [1beta-3H]-androstenedione as substrate assessed as tritiated H2O release after 15 mins b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50523398(CHEMBL4564333)
Affinity DataIC50:  560nMAssay Description:Inhibition of human placental microsome aromatase using [1beta3H]-androstenedione as substrate measured after 15 mins in presence of NADPH by liquid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50069755(CHEMBL3407536)
Affinity DataIC50:  620nMAssay Description:Inhibition of human placental microsome aromatase using [1beta-3H] androstenedione as substrate after 15 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50174543((3R,5R,10R,13S)-3-Hydroxy-10,13-dimethyl-tetradeca...)
Affinity DataIC50:  670nMAssay Description:Inhibitory concentration against aromatase protein from human placental microsomes using [1-beta-3H]-androstenedione; Competitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50069752(CHEMBL3407539)
Affinity DataIC50:  670nMAssay Description:Inhibition of human placental microsome aromatase using [1beta-3H] androstenedione as substrate after 15 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50069755(CHEMBL3407536)
Affinity DataIC50:  730nMAssay Description:Inhibition of human placental microsome aromatase expressed in human MCF7 cells using [1beta-3H] androstenedione as substrate after 1 hr by liquid sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50069754(CHEMBL3407537)
Affinity DataIC50:  810nMAssay Description:Inhibition of human placental microsome aromatase using [1beta-3H] androstenedione as substrate after 15 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50523401(CHEMBL4515880)
Affinity DataIC50:  840nMAssay Description:Inhibition of human placental microsome aromatase using [1beta3H]-androstenedione as substrate measured after 15 mins in presence of NADPH by liquid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50523405(CHEMBL4520027)
Affinity DataIC50:  880nMAssay Description:Inhibition of human placental microsome aromatase using [1beta3H]-androstenedione as substrate measured after 15 mins in presence of NADPH by liquid ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50398447(Aromasin | EXEMESTANE)
Affinity DataIC50:  900nMAssay Description:Inhibition of human placental microsome aromatase expressed in human MCF7 cells using [1beta-3H] androstenedione as substrate after 1 hr by liquid sc...More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50388393(CHEMBL2058266)
Affinity DataIC50:  970nMAssay Description:Inhibition of aromatase in human placental microsomes using [1beta-3H]androstenedione as substrate after 15 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50069752(CHEMBL3407539)
Affinity DataIC50:  980nMAssay Description:Inhibition of human placental microsome aromatase expressed in human MCF7 cells using [1beta-3H] androstenedione as substrate after 1 hr by liquid sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50388395(CHEMBL2058268)
Affinity DataIC50:  1.15E+3nMAssay Description:Inhibition of aromatase in human placental microsomes using [1beta-3H]androstenedione as substrate after 15 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Coimbra

Curated by ChEMBL
LigandPNGBDBM50069754(CHEMBL3407537)
Affinity DataIC50:  1.18E+3nMAssay Description:Inhibition of human placental microsome aromatase expressed in human MCF7 cells using [1beta-3H] androstenedione as substrate after 1 hr by liquid sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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