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Found 100 with Last Name = 'terauchi' and Initial = 'h'
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50138191((1S,5S,6R,7R)-7-Chloro-5-methyl-2-aza-bicyclo[4.1....)
Affinity DataIC50:  3nMAssay Description:Inhibition of inducible nitric oxide synthase (iNOS) in miceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50161394((4R,5R)-5-Ethyl-4-methyl-selenazolidin-(2Z)-yliden...)
Affinity DataIC50:  9.30nMAssay Description:Inhibitory concentration against inducible nitric acid synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50161393((4R,5R)-4-Ethyl-5-methyl-selenazolidin-(2Z)-yliden...)
Affinity DataIC50:  9.40nMAssay Description:Inhibitory concentration against inducible nitric acid synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Mus musculus)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50138191((1S,5S,6R,7R)-7-Chloro-5-methyl-2-aza-bicyclo[4.1....)
Affinity DataIC50:  15nMAssay Description:Inhibition of neuronal nitric oxide synthase (nNOS) in miceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50161388((4S,5S)-4-Ethyl-5-methyl-selenazolidin-(2Z)-yliden...)
Affinity DataIC50:  21nMAssay Description:Inhibitory concentration against inducible nitric acid synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50161389((4R,5S)-4-Ethyl-5-methyl-selenazolidin-(2Z)-yliden...)
Affinity DataIC50:  21nMAssay Description:Inhibitory concentration against inducible nitric acid synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50161392((4S,5S)-5-Ethyl-4-methyl-selenazolidin-(2Z)-yliden...)
Affinity DataIC50:  34nMAssay Description:Inhibitory concentration against inducible nitric acid synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50138189((4S,5R)-5-Methyl-4-propyl-oxazolidin-(2Z)-ylidenea...)
Affinity DataIC50:  41nMAssay Description:Inhibition of inducible nitric oxide synthase (iNOS) in miceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50138195((4S,5S)-4,5-Diethyl-oxazolidin-(2Z)-ylideneamine |...)
Affinity DataIC50:  56nMAssay Description:Inhibition of inducible nitric oxide synthase (iNOS) in miceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50161395((4R,5S)-5-Ethyl-4-methyl-selenazolidin-(2Z)-yliden...)
Affinity DataIC50:  66nMAssay Description:Inhibitory concentration against inducible nitric acid synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50138201(5-Methyl-oxazolidin-(2Z)-ylideneamine | CHEMBL1074...)
Affinity DataIC50:  74nMAssay Description:Inhibition of inducible nitric oxide synthase (iNOS) in miceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50161390((4S,5R)-4-Ethyl-5-methyl-selenazolidin-(2Z)-yliden...)
Affinity DataIC50:  80nMAssay Description:Inhibitory concentration against inducible nitric acid synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50161393((4R,5R)-4-Ethyl-5-methyl-selenazolidin-(2Z)-yliden...)
Affinity DataIC50:  92nMAssay Description:Inhibitory concentration against neuronal nitric acid synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50138190((4S,5S)-5-Methyl-4-propyl-oxazolidin-(2Z)-ylidenea...)
Affinity DataIC50:  120nMAssay Description:Inhibition of inducible nitric oxide synthase (iNOS) in miceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50138192((4S,5R)-4-Ethyl-5-methyl-oxazolidin-(2Z)-ylideneam...)
Affinity DataIC50:  120nMAssay Description:Inhibition of inducible nitric oxide synthase (iNOS) in miceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50138194((4S,5S)-5-Ethyl-4-methyl-oxazolidin-(2Z)-ylideneam...)
Affinity DataIC50:  120nMAssay Description:Inhibition of inducible nitric oxide synthase (iNOS) in miceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50138198((4S,5R)-4,5-Diethyl-oxazolidin-(2Z)-ylideneamine |...)
Affinity DataIC50:  130nMAssay Description:Inhibition of inducible nitric oxide synthase (iNOS) in miceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50138184((4S,5R)-4,5-Dimethyl-oxazolidin-(2Z)-ylideneamine ...)
Affinity DataIC50:  150nMAssay Description:Inhibition of inducible nitric oxide synthase (iNOS) in miceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50138185((4S,5R)-5-Ethyl-4-methyl-oxazolidin-(2Z)-ylideneam...)
Affinity DataIC50:  160nMAssay Description:Inhibition of inducible nitric oxide synthase (iNOS) in miceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50138187((4S,5S)-4-Ethyl-5-methyl-oxazolidin-(2Z)-ylideneam...)
Affinity DataIC50:  170nMAssay Description:Inhibition of inducible nitric oxide synthase (iNOS) in miceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Sus scrofa (Pig))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50037078(2-(Phenyl)-isothiazolo[5,4-b]pyridin-3(2H)-one | 2...)
Affinity DataIC50:  190nMAssay Description:Inhibition of porcine gastric H+/K+ ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Sus scrofa (Pig))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50056046(2-Pyridin-4-yl-isothiazolo[5,4-b]pyridin-3-one | C...)
Affinity DataIC50:  220nMAssay Description:Inhibition of porcine gastric H+/K+ ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50138196((4S,5R)-5-Methyl-4-pentyl-oxazolidin-(2Z)-ylidenea...)
Affinity DataIC50:  230nMAssay Description:Inhibition of inducible nitric oxide synthase (iNOS) in miceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50138193(5-Ethyl-oxazolidin-(2Z)-ylideneamine | CHEMBL10835...)
Affinity DataIC50:  280nMAssay Description:Inhibition of inducible nitric oxide synthase (iNOS) in miceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50161389((4R,5S)-4-Ethyl-5-methyl-selenazolidin-(2Z)-yliden...)
Affinity DataIC50:  280nMAssay Description:Inhibitory concentration against neuronal nitric acid synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50161388((4S,5S)-4-Ethyl-5-methyl-selenazolidin-(2Z)-yliden...)
Affinity DataIC50:  280nMAssay Description:Inhibitory concentration against neuronal nitric acid synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50161391((4S,5R)-5-Ethyl-4-methyl-selenazolidin-(2Z)-yliden...)
Affinity DataIC50:  340nMAssay Description:Inhibitory concentration against inducible nitric acid synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50161392((4S,5S)-5-Ethyl-4-methyl-selenazolidin-(2Z)-yliden...)
Affinity DataIC50:  350nMAssay Description:Inhibitory concentration against neuronal nitric acid synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Homo sapiens (Human))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50241343((RS)-6-methoxy-2-((4-methoxy-3,5-dimethylpyridin-2...)
Affinity DataIC50:  370nMAssay Description:Inhibition of [14C]-aminopyrine (AP) accumulation stimulated by dibutyryl cyclic AMP in isolated rabbit parietal cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Homo sapiens (Human))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50056043(2-(2,4-Diethoxy-phenylmethanesulfinyl)-N-pyridin-4...)
Affinity DataIC50:  400nMAssay Description:Inhibition of [14C]-aminopyrine (AP) accumulation stimulated by dibutyryl cyclic AMP in isolated rabbit parietal cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Mus musculus)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50138186(5-Bromomethyl-oxazolidin-(2Z)-ylideneamine | CHEMB...)
Affinity DataIC50:  400nMAssay Description:Inhibition of neuronal nitric oxide synthase (nNOS) in miceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50226181((3R,4S,5R,6R)-5-hydroxy-6-(4-hydroxy-3-(4-hydroxy-...)
Affinity DataIC50:  408nMAssay Description:Iinhibitory activity against Escherichia coli DNA gyraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Homo sapiens (Human))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50056045(2-(2-Ethoxy-4-methoxy-phenylmethanesulfinyl)-N-pyr...)
Affinity DataIC50:  450nMAssay Description:Inhibition of [14C]-aminopyrine (AP) accumulation stimulated by dibutyryl cyclic AMP in isolated rabbit parietal cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Homo sapiens (Human))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50056041(2-(2,4-Dimethoxy-6-methyl-phenylmethanesulfinyl)-N...)
Affinity DataIC50:  460nMAssay Description:Inhibition of [14C]-aminopyrine (AP) accumulation stimulated by dibutyryl cyclic AMP in isolated rabbit parietal cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50138186(5-Bromomethyl-oxazolidin-(2Z)-ylideneamine | CHEMB...)
Affinity DataIC50:  500nMAssay Description:Inhibition of inducible nitric oxide synthase (iNOS) in miceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Mus musculus)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50225106((2S)-2-amino-5-{[(E)-amino(nitroimino)methyl]amino...)
Affinity DataIC50:  500nMAssay Description:Inhibition of neuronal nitric oxide synthase (nNOS) in miceMore data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50138200((4S,5S)-5-Methyl-4-pentyl-oxazolidin-(2Z)-ylidenea...)
Affinity DataIC50:  500nMAssay Description:Inhibition of inducible nitric oxide synthase (iNOS) in miceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Sus scrofa (Pig))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50056049(2-Isobutyl-isothiazolo[5,4-b]pyridin-3-one | CHEMB...)
Affinity DataIC50:  530nMAssay Description:Inhibition of porcine gastric H+/K+ ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Mus musculus)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50138190((4S,5S)-5-Methyl-4-propyl-oxazolidin-(2Z)-ylidenea...)
Affinity DataIC50:  570nMAssay Description:Inhibition of neuronal nitric oxide synthase (nNOS) in miceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Homo sapiens (Human))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50056056(2-(2,4-Dimethoxy-phenylmethanesulfinyl)-N-pyridin-...)
Affinity DataIC50:  590nMAssay Description:Inhibition of [14C]-aminopyrine (AP) accumulation stimulated by dibutyryl cyclic AMP in isolated rabbit parietal cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50366822(AT-4140 | CI-978 | SPARFLOXACIN | Spara)
Affinity DataIC50:  637nMAssay Description:Iinhibitory activity against Escherichia coli DNA gyraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Mus musculus)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50138192((4S,5R)-4-Ethyl-5-methyl-oxazolidin-(2Z)-ylideneam...)
Affinity DataIC50:  680nMAssay Description:Inhibition of neuronal nitric oxide synthase (nNOS) in miceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50161390((4S,5R)-4-Ethyl-5-methyl-selenazolidin-(2Z)-yliden...)
Affinity DataIC50:  740nMAssay Description:Inhibitory concentration against neuronal nitric acid synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Mus musculus)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50138200((4S,5S)-5-Methyl-4-pentyl-oxazolidin-(2Z)-ylidenea...)
Affinity DataIC50:  790nMAssay Description:Inhibition of neuronal nitric oxide synthase (nNOS) in miceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50161394((4R,5R)-5-Ethyl-4-methyl-selenazolidin-(2Z)-yliden...)
Affinity DataIC50:  790nMAssay Description:Inhibitory concentration against neuronal nitric acid synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Mus musculus)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50138185((4S,5R)-5-Ethyl-4-methyl-oxazolidin-(2Z)-ylideneam...)
Affinity DataIC50:  850nMAssay Description:Inhibition of neuronal nitric oxide synthase (nNOS) in miceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Mus musculus)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50138189((4S,5R)-5-Methyl-4-propyl-oxazolidin-(2Z)-ylidenea...)
Affinity DataIC50:  920nMAssay Description:Inhibition of neuronal nitric oxide synthase (nNOS) in miceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium-transporting ATPase alpha chain 1/subunit beta(Homo sapiens (Human))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50056042(CHEMBL108285 | N-Pyridin-4-yl-2-(2,4,6-trimethoxy-...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of [14C]-aminopyrine (AP) accumulation stimulated by dibutyryl cyclic AMP in isolated rabbit parietal cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Mus musculus)
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50138198((4S,5R)-4,5-Diethyl-oxazolidin-(2Z)-ylideneamine |...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of neuronal nitric oxide synthase (nNOS) in miceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, brain(Homo sapiens (Human))
Dainippon Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50161395((4R,5S)-5-Ethyl-4-methyl-selenazolidin-(2Z)-yliden...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibitory concentration against neuronal nitric acid synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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