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Found 348 with Last Name = 'terebetski' and Initial = 'j'
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50021345(CHEMBL3287928)
Affinity DataKi:  637nMAssay Description:Displacement of [35S]MK-499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50021331(CHEMBL3287930)
Affinity DataKi:  740nMAssay Description:Displacement of [35S]MK-499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50350538(CHEMBL1812717)
Affinity DataKi:  1.25E+3nMAssay Description:Displacement of [35S]MK-499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50021346(CHEMBL3287926)
Affinity DataKi:  1.54E+3nMAssay Description:Displacement of [35S]MK-499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50021329(CHEMBL3287932)
Affinity DataKi:  2.50E+3nMAssay Description:Displacement of [35S]MK-499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50021344(CHEMBL3287929)
Affinity DataKi:  5.21E+3nMAssay Description:Displacement of [35S]MK-499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50021334(CHEMBL3287931)
Affinity DataKi:  2.85E+4nMAssay Description:Displacement of [35S]MK-499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50021330(CHEMBL3287927)
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [35S]MK-499 from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Mus musculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50362418(CHEMBL1938418)
Affinity DataIC50:  0.180nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Mus musculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50362419(CHEMBL1940544)
Affinity DataIC50:  0.200nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434318(CHEMBL2386566)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of human FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Mus musculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50362420(CHEMBL1940540)
Affinity DataIC50:  0.330nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434329(CHEMBL2386554)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of rat FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Mus musculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50362417(CHEMBL1940545)
Affinity DataIC50:  0.420nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Mus musculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50362409(CHEMBL1940543)
Affinity DataIC50:  0.430nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434329(CHEMBL2386554)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of human FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434316(CHEMBL2386568)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of human FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434318(CHEMBL2386566)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of rat FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Mus musculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50362417(CHEMBL1940545)
Affinity DataIC50:  0.660nMAssay Description:Antagonist activity at mouse NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Mus musculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50362414(CHEMBL1940537)
Affinity DataIC50:  0.690nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434317(CHEMBL2386567)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of human FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Mus musculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50362419(CHEMBL1940544)
Affinity DataIC50:  0.860nMAssay Description:Antagonist activity at mouse NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434313(CHEMBL2386571)
Affinity DataIC50:  1nMAssay Description:Inhibition of human FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434315(CHEMBL2386569)
Affinity DataIC50:  1nMAssay Description:Inhibition of human FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Mus musculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50362412(CHEMBL1940539)
Affinity DataIC50:  1.10nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434322(CHEMBL2386562)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of human FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434314(CHEMBL2386570)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of human FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434314(CHEMBL2386570)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of rat FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Mus musculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50362418(CHEMBL1938418)
Affinity DataIC50:  1.30nMAssay Description:Antagonist activity at mouse NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434316(CHEMBL2386568)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of rat FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434315(CHEMBL2386569)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of rat FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434320(CHEMBL2386564)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of human FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434317(CHEMBL2386567)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of rat FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434313(CHEMBL2386571)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of rat FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Mus musculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50362420(CHEMBL1940540)
Affinity DataIC50:  1.80nMAssay Description:Antagonist activity at mouse NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Mus musculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50362415(CHEMBL1940536)
Affinity DataIC50:  1.90nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Mus musculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50362411(CHEMBL1940541)
Affinity DataIC50:  2.20nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Mus musculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50362413(CHEMBL1940538)
Affinity DataIC50:  2.40nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Mus musculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50362410(CHEMBL1940542)
Affinity DataIC50:  2.60nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Mus musculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50362437(CHEMBL1940367)
Affinity DataIC50:  2.80nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434319(CHEMBL2386565)
Affinity DataIC50:  3nMAssay Description:Inhibition of rat FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434319(CHEMBL2386565)
Affinity DataIC50:  3nMAssay Description:Inhibition of human FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Mus musculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50362412(CHEMBL1940539)
Affinity DataIC50:  3nMAssay Description:Antagonist activity at mouse NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Mus musculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50362430(CHEMBL1940526)
Affinity DataIC50:  3.10nMAssay Description:Displacement of [125]-hNPW23 from mouse NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434321(CHEMBL2386563)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of human FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434323(CHEMBL2386561)
Affinity DataIC50:  3.30nMAssay Description:Inhibition of human FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Mus musculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50362409(CHEMBL1940543)
Affinity DataIC50:  3.90nMAssay Description:Antagonist activity at mouse NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434328(CHEMBL2386555)
Affinity DataIC50:  4.20nMAssay Description:Inhibition of rat FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptides B/W receptor type 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50362414(CHEMBL1940537)
Affinity DataIC50:  4.20nMAssay Description:Displacement of [125]-hNPW23 from human NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434320(CHEMBL2386564)
Affinity DataIC50:  4.20nMAssay Description:Inhibition of rat FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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