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Found 47 with Last Name = 'terenius' and Initial = 'l'
TargetSubstance-P receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataIC50:  1.5nMAssay Description:Affinity for rat Tachykinin receptor 1 determined in displacement screening by using radioligand 3,4-[3H]-(L-Pro e2) SP.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM21015((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...)
Affinity DataIC50:  3.5nMAssay Description:The compound was tested for binding affinity towards rat Opioid receptor mu 1 by displacing [3H]DAMGO.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50059841((S)-1-[(S)-2-[2-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hy...)
Affinity DataIC50:  6.20nMAssay Description:The compound was tested for binding affinity towards [3H]DAMGO, in rat Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataIC50:  8.5nMAssay Description:Binding to mu opioid receptor by using [3H]-DAMGO as radioligand in guinea pig brain minus cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50081923((S)-1-[(S)-2-{[5-((S)-1-{(R)-2-[(S)-2-Amino-3-(4-h...)
Affinity DataIC50:  12nMAssay Description:The compound was tested for binding affinity towards rat Opioid receptor mu 1 by displacing [3H]DAMGO.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50081924((S)-1-[(S)-2-[5-((S)-1-{(R)-2-[(S)-2-Amino-3-(4-hy...)
Affinity DataIC50:  17nMAssay Description:The compound was tested for binding affinity towards rat Opioid receptor mu 1 by displacing [3H]DAMGO.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50081925((S)-1-[(S)-2-[5-((S)-1-{(R)-2-[(S)-2-Amino-3-(4-hy...)
Affinity DataIC50:  20nMAssay Description:The compound was tested for binding affinity towards rat Opioid receptor mu 1 by displacing [3H]DAMGO.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50081929((S)-1-[(S)-2-{[5-((S)-1-{(R)-2-[(S)-2-Amino-3-(4-h...)
Affinity DataIC50:  21nMAssay Description:The compound was tested for binding affinity towards rat Opioid receptor mu 1 by displacing [3H]DAMGO.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50081927((S)-1-[(S)-2-{[5-((S)-1-{(R)-2-[(S)-2-Amino-3-(4-h...)
Affinity DataIC50:  31nMAssay Description:The compound was tested for binding affinity towards rat Opioid receptor mu 1 by displacing [3H]DAMGO.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataIC50:  130nMAssay Description:Binding to kappa opioid receptor by using [3H]-U-69,593 as radioligand in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50283517(10-(3-furyl)-4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4...)
Affinity DataIC50:  200nMAssay Description:Binding to mu opioid receptor by using [3H]-DAMGO as radioligand in guinea pig brain minus cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50081935((alpha)-H-Arg-Pro-Lys-pro-Gln-Gln-Phe-{2-[5-((S)-1...)
Affinity DataIC50:  307nMAssay Description:Affinity for rat Tachykinin receptor 1 determined in displacement screening by using radioligand 3,4-[3H]-(L-Pro e2) SP.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataIC50:  430nMAssay Description:Binding to delta opioid receptor by using [3H]-DPDPE as radioligand in guinea pig brain minus cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticleDrugBank

TargetMu-type opioid receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50081926((S)-1-[(S)-2-[5-((S)-1-{(R)-2-[(S)-2-Amino-3-(4-hy...)
Affinity DataIC50:  490nMAssay Description:The compound was tested for binding affinity towards rat Opioid receptor mu 1 by displacing [3H]DAMGO.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50283522(4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-azapentacycl...)
Affinity DataIC50:  530nMAssay Description:Binding to mu opioid receptor by using [3H]-DAMGO as radioligand in guinea pig brain minus cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50283516(1-[14-hydroxy-4-methyl-(1S,5R,13R,14S,17R)-12-oxa-...)
Affinity DataIC50:  640nMAssay Description:Binding to mu opioid receptor by using [3H]-DAMGO as radioligand in guinea pig brain minus cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50283517(10-(3-furyl)-4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4...)
Affinity DataIC50:  910nMAssay Description:Binding to kappa opioid receptor by using [3H]-U-69,593 as radioligand in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50081936(CHEMBL263584 | H-Arg-Pro-Lys-pro-Gln-Gln-Phe-{5-[(...)
Affinity DataIC50: >1.00E+3nMAssay Description:Affinity for rat Tachykinin receptor 1 determined in displacement screening by using radioligand 3,4-[3H]-(L-Pro e2) SP.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50081924((S)-1-[(S)-2-[5-((S)-1-{(R)-2-[(S)-2-Amino-3-(4-hy...)
Affinity DataIC50: >1.00E+3nMAssay Description:Affinity for rat Tachykinin receptor 1 determined in displacement screening by using radioligand 3,4-[3H]-(L-Pro e2) SP.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM21015((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...)
Affinity DataIC50: >1.00E+3nMAssay Description:Affinity for rat Tachykinin receptor 1 determined in displacement screening by using radioligand 3,4-[3H]-(L-Pro e2) SP.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50081927((S)-1-[(S)-2-{[5-((S)-1-{(R)-2-[(S)-2-Amino-3-(4-h...)
Affinity DataIC50: >1.00E+3nMAssay Description:Affinity for rat Tachykinin receptor 1 determined in displacement screening by using radioligand 3,4-[3H]-(L-Pro e2) SP.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50081935((alpha)-H-Arg-Pro-Lys-pro-Gln-Gln-Phe-{2-[5-((S)-1...)
Affinity DataIC50: >1.00E+3nMAssay Description:Affinity for rat Tachykinin receptor 1 determined in displacement screening by using radioligand 3,4-[3H]-(L-Pro e2) SP.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50081933(CHEMBL138013 | {(S)-1-[3-(2-Hydroxy-ethyl)-[1,2,4]...)
Affinity DataIC50: >1.00E+3nMAssay Description:Affinity for rat Tachykinin receptor 1 determined in displacement screening by using radioligand 3,4-[3H]-(L-Pro e2) SP.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50081926((S)-1-[(S)-2-[5-((S)-1-{(R)-2-[(S)-2-Amino-3-(4-hy...)
Affinity DataIC50: >1.00E+3nMAssay Description:Affinity for rat Tachykinin receptor 1 determined in displacement screening by using radioligand 3,4-[3H]-(L-Pro e2) SP.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50081932(CHEMBL410170 | H-Arg-Pro-Lys-pro-Gln-Gln-Phe-{5-[(...)
Affinity DataIC50: >1.00E+3nMAssay Description:Affinity for rat Tachykinin receptor 1 determined in displacement screening by using radioligand 3,4-[3H]-(L-Pro e2) SP.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50081931(CHEMBL402884 | H-Arg-Pro-Lys-pro-Gln-Gln-Phe-{2-[5...)
Affinity DataIC50: >1.00E+3nMAssay Description:Affinity for rat Tachykinin receptor 1 determined in displacement screening by using radioligand 3,4-[3H]-(L-Pro e2) SP.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50081930(CHEMBL268138 | H-Arg-Pro-Lys-pro-Gln-Gln-Phe-{5-[(...)
Affinity DataIC50: >1.00E+3nMAssay Description:Affinity for rat Tachykinin receptor 1 determined in displacement screening by using radioligand 3,4-[3H]-(L-Pro e2) SP.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50081929((S)-1-[(S)-2-{[5-((S)-1-{(R)-2-[(S)-2-Amino-3-(4-h...)
Affinity DataIC50: >1.00E+3nMAssay Description:Affinity for rat Tachykinin receptor 1 determined in displacement screening by using radioligand 3,4-[3H]-(L-Pro e2) SP.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50081928(CHEMBL136875 | [5-((S)-1-tert-Butoxycarbonylamino-...)
Affinity DataIC50: >1.00E+3nMAssay Description:Affinity for rat Tachykinin receptor 1 determined in displacement screening by using radioligand 3,4-[3H]-(L-Pro e2) SP.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50081925((S)-1-[(S)-2-[5-((S)-1-{(R)-2-[(S)-2-Amino-3-(4-hy...)
Affinity DataIC50: >1.00E+3nMAssay Description:Affinity for rat Tachykinin receptor 1 determined in displacement screening by using radioligand 3,4-[3H]-(L-Pro e2) SP.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50059841((S)-1-[(S)-2-[2-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hy...)
Affinity DataIC50: >1.00E+3nMAssay Description:Affinity for rat Tachykinin receptor 1 determined in displacement screening by using radioligand 3,4-[3H]-(L-Pro e2) SP.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50081923((S)-1-[(S)-2-{[5-((S)-1-{(R)-2-[(S)-2-Amino-3-(4-h...)
Affinity DataIC50: >1.00E+3nMAssay Description:Affinity for rat Tachykinin receptor 1 determined in displacement screening by using radioligand 3,4-[3H]-(L-Pro e2) SP.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50283521(10-(2-furyl)-4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4...)
Affinity DataIC50:  2.60E+3nMAssay Description:Binding to mu opioid receptor by using [3H]-DAMGO as radioligand in guinea pig brain minus cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50283519(4-methyl-10-(3-thienyl)-(1S,5R,13R,14S,17R)-12-oxa...)
Affinity DataIC50:  3.30E+3nMAssay Description:Binding to mu opioid receptor by using [3H]-DAMGO as radioligand in guinea pig brain minus cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50283523(4,10-dimethyl-(1S,5R,13R,14S,17R)-12-oxa-4-azapent...)
Affinity DataIC50:  4.50E+3nMAssay Description:Binding to mu opioid receptor by using [3H]-DAMGO as radioligand in guinea pig brain minus cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50283516(1-[14-hydroxy-4-methyl-(1S,5R,13R,14S,17R)-12-oxa-...)
Affinity DataIC50:  5.10E+3nMAssay Description:Binding to kappa opioid receptor by using [3H]-U-69,593 as radioligand in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50283518(14-hydroxy-4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-a...)
Affinity DataIC50:  6.40E+3nMAssay Description:Binding to mu opioid receptor by using [3H]-DAMGO as radioligand in guinea pig brain minus cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283517(10-(3-furyl)-4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4...)
Affinity DataIC50:  7.40E+3nMAssay Description:Binding to delta opioid receptor by using [3H]-DPDPE as radioligand in guinea pig brain minus cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283516(1-[14-hydroxy-4-methyl-(1S,5R,13R,14S,17R)-12-oxa-...)
Affinity DataIC50:  7.90E+3nMAssay Description:Binding to delta opioid receptor by using [3H]-DPDPE as radioligand in guinea pig brain minus cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50283521(10-(2-furyl)-4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4...)
Affinity DataIC50:  9.50E+3nMAssay Description:Binding to kappa opioid receptor by using [3H]-U-69,593 as radioligand in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50283522(4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-azapentacycl...)
Affinity DataIC50:  1.10E+4nMAssay Description:Binding to kappa opioid receptor by using [3H]-U-69,593 as radioligand in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50283519(4-methyl-10-(3-thienyl)-(1S,5R,13R,14S,17R)-12-oxa...)
Affinity DataIC50:  1.50E+4nMAssay Description:Binding to kappa opioid receptor by using [3H]-U-69,593 as radioligand in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50283525(4-methyl-10-(2-thienyl)-(1S,5R,13R,14S,17R)-12-oxa...)
Affinity DataIC50:  2.50E+4nMAssay Description:Binding to kappa opioid receptor by using [3H]-U-69,593 as radioligand in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50283523(4,10-dimethyl-(1S,5R,13R,14S,17R)-12-oxa-4-azapent...)
Affinity DataIC50:  3.60E+4nMAssay Description:Binding to kappa opioid receptor by using [3H]-U-69,593 as radioligand in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50283524(4-methyl-10-phenyl-(1S,5R,13R,14S,17R)-12-oxa-4-az...)
Affinity DataIC50:  7.60E+4nMAssay Description:Binding to kappa opioid receptor by using [3H]-U-69,593 as radioligand in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50283518(14-hydroxy-4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-a...)
Affinity DataIC50:  1.11E+5nMAssay Description:Binding to kappa opioid receptor by using [3H]-U-69,593 as radioligand in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50283520(10-benzo[b]thiophen-2-yl-4-methyl-(1S,5R,13R,14S,1...)
Affinity DataIC50:  1.26E+5nMAssay Description:Binding to kappa opioid receptor by using [3H]-U-69,593 as radioligand in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails Article