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Found 16 with Last Name = 'tibasco' and Initial = 'j'
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50417543(CHEMBL1632210)
Affinity DataKi:  50.1nMAssay Description:Displacement of [3H]dofetilide from human ERG by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50417544(CHEMBL1632218)
Affinity DataKi:  316nMAssay Description:Displacement of [3H]dofetilide from human ERG by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50417549(CHEMBL1632223)
Affinity DataKi:  316nMAssay Description:Displacement of [3H]dofetilide from human ERG by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50417545(CHEMBL1631535)
Affinity DataKi:  501nMAssay Description:Displacement of [3H]dofetilide from human ERG by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50417546(CHEMBL1632220)
Affinity DataKi:  631nMAssay Description:Displacement of [3H]dofetilide from human ERG by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50417548(CHEMBL1631542)
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of [3H]dofetilide from human ERG by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50417547(CHEMBL1632206)
Affinity DataKi:  3.98E+3nMAssay Description:Displacement of [3H]dofetilide from human ERG by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50333015(1-(3-{2-[4-(2-Methyl-5-quinolinyl)-1-piperazinyl]e...)
Affinity DataKi:  1.26E+4nMAssay Description:Displacement of [3H]dofetilide from human ERG by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50333015(1-(3-{2-[4-(2-Methyl-5-quinolinyl)-1-piperazinyl]e...)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using atorvastatin as probeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50333015(1-(3-{2-[4-(2-Methyl-5-quinolinyl)-1-piperazinyl]e...)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using midazolam as probeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50333015(1-(3-{2-[4-(2-Methyl-5-quinolinyl)-1-piperazinyl]e...)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using nifedipine as probeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50333015(1-(3-{2-[4-(2-Methyl-5-quinolinyl)-1-piperazinyl]e...)
Affinity DataIC50:  6.00E+4nMAssay Description:Inhibition of human recombinant CYP2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50333015(1-(3-{2-[4-(2-Methyl-5-quinolinyl)-1-piperazinyl]e...)
Affinity DataIC50:  6.70E+4nMAssay Description:Inhibition of human recombinant CYP3A4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50333015(1-(3-{2-[4-(2-Methyl-5-quinolinyl)-1-piperazinyl]e...)
Affinity DataIC50:  7.60E+4nMAssay Description:Inhibition of human recombinant CYP219More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50333015(1-(3-{2-[4-(2-Methyl-5-quinolinyl)-1-piperazinyl]e...)
Affinity DataIC50:  8.60E+4nMAssay Description:Inhibition of human recombinant CYP2D6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50333015(1-(3-{2-[4-(2-Methyl-5-quinolinyl)-1-piperazinyl]e...)
Affinity DataIC50:  9.60E+4nMAssay Description:Inhibition of human recombinant CYP1A2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed