Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of TET2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of recombinant human N-terminal Flag-tagged TET1 (1418 to 2136 residues) expressed in Baculovirus infected Sf9 cells assessed as reduction...More data for this Ligand-Target Pair
Affinity DataIC50: 2.31E+3nMAssay Description:Inhibition of TET3 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 3.48E+3nMAssay Description:Inhibition of TET1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 8.80E+3nMAssay Description:Inhibition of recombinant human N-terminal Flag-tagged C-terminal His-tagged TET3 (824 to 1795 residues) expressed in Baculovirus infected Sf9 cells ...More data for this Ligand-Target Pair
Affinity DataIC50: 9.40E+3nMAssay Description:Inhibition of recombinant human GST-tagged TET2 (1099 to 1936 residues) expressed in Escherichia coli BL21 (DE3)pLysS assessed as reduction in 5hmc l...More data for this Ligand-Target Pair
Affinity DataIC50: 1.05E+4nMAssay Description:Inhibition of recombinant human GST-tagged TET2 (1099 to 1936 residues) expressed in Escherichia coli BL21 (DE3)pLysS assessed as reduction in 5hmc l...More data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of recombinant human GST-tagged TET2 (1099 to 1936 residues) expressed in Escherichia coli BL21 (DE3)pLysS assessed as reduction in 5hmc l...More data for this Ligand-Target Pair
Affinity DataIC50: 1.97E+4nMAssay Description:Inhibition of recombinant human GST-tagged TET2 (1099 to 1936 residues) expressed in Escherichia coli BL21 (DE3)pLysS assessed as reduction in 5hmc l...More data for this Ligand-Target Pair
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of TET1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 5.48E+4nMAssay Description:Inhibition of recombinant human GST-tagged TET2 (1099 to 1936 residues) expressed in Escherichia coli BL21 (DE3)pLysS assessed as reduction in 5hmc l...More data for this Ligand-Target Pair
Affinity DataIC50: 7.30E+4nMAssay Description:Inhibition of TET2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.07E+5nMAssay Description:Inhibition of recombinant human GST-tagged TET2 (1099 to 1936 residues) expressed in Escherichia coli BL21 (DE3)pLysS assessed as reduction in 5hmc l...More data for this Ligand-Target Pair
Affinity DataIC50: 1.08E+5nMAssay Description:Inhibition of recombinant human GST-tagged TET2 (1099 to 1936 residues) expressed in Escherichia coli BL21 (DE3)pLysS assessed as reduction in 5hmc l...More data for this Ligand-Target Pair
Affinity DataIC50: 2.62E+5nMAssay Description:Inhibition of recombinant human GST-tagged TET2 (1099 to 1936 residues) expressed in Escherichia coli BL21 (DE3)pLysS assessed as reduction in 5hmc l...More data for this Ligand-Target Pair
TargetBiotin--[biotin carboxyl-carrier protein] ligase(Mycobacterium tuberculosis (strain CDC 1551 / Oshk...)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKd: 0.0400nMAssay Description:Inhibition of biotin binding to Mycobacterium tuberculosis BirA by isothermal titration calorimetryMore data for this Ligand-Target Pair
TargetBiotin--[biotin carboxyl-carrier protein] ligase(Mycobacterium tuberculosis (strain CDC 1551 / Oshk...)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKd: 0.100nMAssay Description:Inhibition of biotin binding to Mycobacterium tuberculosis BirA by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 3.42E+3nMAssay Description:Binding affinity to human recombinant TET2 (1099 to 1936) catalytic domain assessed as dissociation constant by micro-scale thermophoresis analysisMore data for this Ligand-Target Pair
Affinity DataKd: 300nMAssay Description:Binding affinity to human recombinant TET2 (1099 to 1936) catalytic domain assessed as dissociation constant by micro-scale thermophoresis analysisMore data for this Ligand-Target Pair
Affinity DataKd: 610nMAssay Description:Binding affinity to human recombinant TET2 (1099 to 1936) catalytic domain assessed as dissociation constant by micro-scale thermophoresis analysisMore data for this Ligand-Target Pair
TargetBiotin--[biotin carboxyl-carrier protein] ligase(Mycobacterium tuberculosis (strain CDC 1551 / Oshk...)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKd: 0.230nMAssay Description:Inhibition of biotin binding to Mycobacterium tuberculosis BirA by isothermal titration calorimetryMore data for this Ligand-Target Pair
TargetBiotin--[biotin carboxyl-carrier protein] ligase(Mycobacterium tuberculosis (strain CDC 1551 / Oshk...)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKd: 11nMAssay Description:Inhibition of biotin binding to Mycobacterium tuberculosis BirA by isothermal titration calorimetryMore data for this Ligand-Target Pair
TargetBiotin--[biotin carboxyl-carrier protein] ligase(Mycobacterium tuberculosis (strain CDC 1551 / Oshk...)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKd: 0.315nMAssay Description:Binding affinity to Mycobacterium tuberculosis H37Rv Biotin protein ligase expressed in Escherichia coli by ITC analysisMore data for this Ligand-Target Pair
TargetBiotin--[biotin carboxyl-carrier protein] ligase(Mycobacterium tuberculosis (strain CDC 1551 / Oshk...)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKd: 0.592nMAssay Description:Binding affinity to Mycobacterium tuberculosis H37Rv Biotin protein ligase expressed in Escherichia coli by ITC analysisMore data for this Ligand-Target Pair
TargetBiotin--[biotin carboxyl-carrier protein] ligase(Mycobacterium tuberculosis (strain CDC 1551 / Oshk...)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKd: 0.865nMAssay Description:Binding affinity to Mycobacterium tuberculosis H37Rv Biotin protein ligase expressed in Escherichia coli by ITC analysisMore data for this Ligand-Target Pair
TargetBiotin--[biotin carboxyl-carrier protein] ligase(Mycobacterium tuberculosis (strain CDC 1551 / Oshk...)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKd: 0.753nMAssay Description:Binding affinity to Mycobacterium tuberculosis H37Rv Biotin protein ligase expressed in Escherichia coli by ITC analysisMore data for this Ligand-Target Pair
TargetBiotin--[biotin carboxyl-carrier protein] ligase(Mycobacterium tuberculosis (strain CDC 1551 / Oshk...)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKd: 2.10nMAssay Description:Binding affinity to Mycobacterium tuberculosis H37Rv Biotin protein ligase expressed in Escherichia coli by ITC analysisMore data for this Ligand-Target Pair
TargetBiotin--[biotin carboxyl-carrier protein] ligase(Mycobacterium tuberculosis (strain CDC 1551 / Oshk...)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKd: 0.540nMAssay Description:Binding affinity to Mycobacterium tuberculosis H37Rv Biotin protein ligase expressed in Escherichia coli by ITC analysisMore data for this Ligand-Target Pair
TargetBiotin--[biotin carboxyl-carrier protein] ligase(Mycobacterium tuberculosis (strain CDC 1551 / Oshk...)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKd: 0.933nMAssay Description:Binding affinity to Mycobacterium tuberculosis H37Rv Biotin protein ligase expressed in Escherichia coli by ITC analysisMore data for this Ligand-Target Pair
TargetBiotin--[biotin carboxyl-carrier protein] ligase(Mycobacterium tuberculosis (strain CDC 1551 / Oshk...)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKd: 0.627nMAssay Description:Binding affinity to Mycobacterium tuberculosis H37Rv Biotin protein ligase expressed in Escherichia coli by ITC analysisMore data for this Ligand-Target Pair
TargetBiotin--[biotin carboxyl-carrier protein] ligase(Mycobacterium tuberculosis (strain CDC 1551 / Oshk...)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKd: 0.0270nMAssay Description:Binding affinity to Mycobacterium tuberculosis H37Rv Biotin protein ligase expressed in Escherichia coli by ITC analysisMore data for this Ligand-Target Pair
TargetBiotin--[biotin carboxyl-carrier protein] ligase(Mycobacterium tuberculosis (strain CDC 1551 / Oshk...)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKd: 0.614nMAssay Description:Binding affinity to Mycobacterium tuberculosis H37Rv Biotin protein ligase expressed in Escherichia coli by ITC analysisMore data for this Ligand-Target Pair
TargetBiotin--[biotin carboxyl-carrier protein] ligase(Mycobacterium tuberculosis (strain CDC 1551 / Oshk...)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKd: 0.153nMAssay Description:Binding affinity to Mycobacterium tuberculosis H37Rv Biotin protein ligase expressed in Escherichia coli by ITC analysisMore data for this Ligand-Target Pair
Affinity DataKd: 2.05E+3nMAssay Description:Binding affinity to human recombinant TET2 (1099 to 1936) catalytic domain assessed as dissociation constant by micro-scale thermophoresis analysisMore data for this Ligand-Target Pair
TargetBiotin--[biotin carboxyl-carrier protein] ligase(Mycobacterium tuberculosis (strain CDC 1551 / Oshk...)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKd: 0.324nMAssay Description:Binding affinity to Mycobacterium tuberculosis H37Rv Biotin protein ligase expressed in Escherichia coli by ITC analysisMore data for this Ligand-Target Pair
TargetBiotin--[biotin carboxyl-carrier protein] ligase(Mycobacterium tuberculosis (strain CDC 1551 / Oshk...)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKd: 0.769nMAssay Description:Binding affinity to Mycobacterium tuberculosis H37Rv Biotin protein ligase expressed in Escherichia coli by ITC analysisMore data for this Ligand-Target Pair