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Found 88 with Last Name = 'tomassini' and Initial = 'je'
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Isis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50144942(2'-C-Me-guanosine | 2'-C-methyl-guanosine | 2'-C-m...)
Affinity DataIC50:  130nMAssay Description:Inhibition HCV NS5B-mediated RNA synthesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385528(CHEMBL2040586)
Affinity DataIC50:  180nMAssay Description:Inhibition of Influenza replicationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385503(CHEMBL2040554)
Affinity DataIC50:  320nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50125801(4-[1-Benzyl-4-(4-chloro-benzyl)-piperidin-4-yl]-2-...)
Affinity DataIC50:  350nMAssay Description:Inhibition of Influenza replicationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50125801(4-[1-Benzyl-4-(4-chloro-benzyl)-piperidin-4-yl]-2-...)
Affinity DataIC50:  430nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385528(CHEMBL2040586)
Affinity DataIC50:  540nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Isis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50144937(2-Amino-9-((2R,3R,5S)-3-hydroxy-5-hydroxymethyl-te...)
Affinity DataIC50:  600nMAssay Description:Inhibition HCV NS5B-mediated RNA synthesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385503(CHEMBL2040554)
Affinity DataIC50:  710nMAssay Description:Inhibition of Influenza replicationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385531(CHEMBL2040602)
Affinity DataIC50:  800nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50125833(3-(4-Fluoro-benzylidene)-1-hydroxy-5-isobutyl-3H-p...)
Affinity DataIC50:  900nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385529(CHEMBL2040587)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385532(CHEMBL2040603)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Isis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50144947(2-Amino-9-((2R,3R,4R,5R)-4-hydroxy-5-hydroxymethyl...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition HCV NS5B-mediated RNA synthesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385529(CHEMBL2040587)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of Influenza replicationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Isis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50144938(2-Amino-9-((2R,3S,4S,5R)-4-fluoro-3-hydroxy-5-hydr...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition HCV NS5B-mediated RNA synthesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Isis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50144948((2R,3R,4R,5R)-2-(6-amino-9H-purin-9-yl)-5-(hydroxy...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition HCV NS5B-mediated RNA synthesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Isis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50144949((2R,3R,4R,5R)-2-(2,6-diamino-9H-purin-9-yl)-5-(hyd...)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition HCV NS5B-mediated RNA synthesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385534(CHEMBL2040605)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385535(CHEMBL2040606)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Isis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50144934((2R,3R,4R,5R)-2-(6-hydroxy-9H-purin-9-yl)-5-(hydro...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition HCV NS5B-mediated RNA synthesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385530(CHEMBL2040601)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50125822(1-Hydroxy-5-isobutyl-3-isobutylidene-3H-pyrazine-2...)
Affinity DataIC50:  5.10E+3nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385536(CHEMBL2040608)
Affinity DataIC50:  6.50E+3nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385533(CHEMBL2040604)
Affinity DataIC50:  7.30E+3nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Isis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50409930(CHEMBL2021379)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition HCV NS5B-mediated RNA synthesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Isis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50144950(3'-deoxyadenosine | 9-(beta-D-3'-Deoxyribofuranosy...)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition HCV NS5B-mediated RNA synthesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Isis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50144933((2R,3S,4S,5R)-4-Fluoro-5-hydroxymethyl-2-(6-methyl...)
Affinity DataIC50:  2.80E+4nMAssay Description:Inhibition HCV NS5B-mediated RNA synthesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Isis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50144939((2R,3R,4R,5R)-2-(2-amino-9H-purin-9-yl)-5-(hydroxy...)
Affinity DataIC50:  4.60E+4nMAssay Description:Inhibition HCV NS5B-mediated RNA synthesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Isis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50144945((2R,3R,4R,5R)-2-Hydroxymethyl-4-methoxy-5-(6-methy...)
Affinity DataIC50:  4.70E+4nMAssay Description:Inhibition HCV NS5B-mediated RNA synthesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Isis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50422565(CHEMBL2311161)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition HCV NS5B-mediated RNA synthesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Isis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50408410(CHEMBL480143)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition HCV NS5B-mediated RNA synthesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Isis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50144932((2R,3R,4R,5R)-4-Fluoro-2-hydroxymethyl-5-(6-methyl...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition HCV NS5B-mediated RNA synthesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Isis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50144941((2R,3R,4R,5R)-5-(6-amino-9H-purin-9-yl)-2-(hydroxy...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition HCV NS5B-mediated RNA synthesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Isis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50144936(CHEMBL1090 | VIDARABINE | adenine arabinoside)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition HCV NS5B-mediated RNA synthesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Isis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50144940((2R,3S,4R,5R)-2-(6-amino-9H-purin-9-yl)-5-(hydroxy...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition HCV NS5B-mediated RNA synthesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRNA-directed RNA polymerase(Hepatitis C virus)
Isis Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50144935((2R,3R,4R,5R)-2-(6-amino-9H-purin-9-yl)-3-ethyl-5-...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition HCV NS5B-mediated RNA synthesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385561(CHEMBL2040639)
Affinity DataIC50:  8.50E+4nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385566(CHEMBL2040632)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385567(CHEMBL2040637)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385537(CHEMBL2040609)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385538(CHEMBL2040610)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385539(CHEMBL2040611)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385540(CHEMBL2040612)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385541(CHEMBL2040613)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385542(CHEMBL2040614)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385543(CHEMBL2040616)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385544(CHEMBL2040617)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385545(CHEMBL2040618)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385546(CHEMBL2040620)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase acidic protein(Hepatitis C virus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50385547(CHEMBL2040621)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of cap 1 ALMV primed Influenza transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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