TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Shizuoka
Curated by ChEMBL
University Of Shizuoka
Curated by ChEMBL
Affinity DataIC50: 0.150nMAssay Description:Antagonist activity at human brain TRPV1 expressed in HEK293T cells assessed as inhibition of CAP-induced intracellular Ca2+ influx by fluorescence-b...More data for this Ligand-Target Pair
Affinity DataIC50: 2.30nMAssay Description:Inhibition of thromboxane A2 synthetase from human platelets by 1 uM of the compoundMore data for this Ligand-Target Pair
TargetGrowth/differentiation factor 8(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of myostatin (unknown origin) expressed in HEK293 cells incubated for 4 hrs by dual luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Shizuoka
Curated by ChEMBL
University Of Shizuoka
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Antagonist activity at human brain TRPV1 expressed in HEK293T cells assessed as inhibition of CAP-induced intracellular Ca2+ influx by fluorescence-b...More data for this Ligand-Target Pair
TargetGrowth/differentiation factor 8(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Inhibition of myostatin (unknown origin) expressed in HEK293 cells transfected with Smad2/3 responsive reporter plasmid incubated for 4 hrs by dual l...More data for this Ligand-Target Pair
TargetGrowth/differentiation factor 8(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Affinity DataIC50: 260nMAssay Description:Inhibition of myostatin (unknown origin) expressed in HEK293 cells transfected with Smad2/3 responsive reporter plasmid incubated for 4 hrs by dual l...More data for this Ligand-Target Pair
TargetGrowth/differentiation factor 8(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of myostatin (unknown origin) expressed in HEK293 cells transfected with Smad2/3 responsive reporter plasmid incubated for 4 hrs by dual l...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Mus musculus)
University Of Shizuoka
Curated by ChEMBL
University Of Shizuoka
Curated by ChEMBL
Affinity DataIC50: 350nMAssay Description:Antagonist at TRPM8 isolated from mouse dorsal root ganglion cells expressed in HEK T-REx cells assessed as inhibition of menthol-induced intracellul...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Mus musculus)
University Of Shizuoka
Curated by ChEMBL
University Of Shizuoka
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Antagonist at TRPM8 isolated from mouse dorsal root ganglion cells expressed in HEK T-REx cells assessed as inhibition of icilin-induced intracellula...More data for this Ligand-Target Pair
TargetTransforming growth factor beta-1 proprotein(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of TGF beta 1 (unknown origin) expressed in HEK293 cells transfected with Smad2/3 responsive reporter plasmid incubated for 4 hrs by dual ...More data for this Ligand-Target Pair
TargetGrowth/differentiation factor 8(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Affinity DataIC50: 3.56E+3nMAssay Description:Inhibition of myostatin (unknown origin) expressed in HEK293 cells incubated for 4 hrs by dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of the expression of AP1-luciferase by TPA-stimulated NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of the expression of AP1-luciferase by TPA-stimulated NIH3T3 cellsMore data for this Ligand-Target Pair
TargetGrowth/differentiation factor 8(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of myostatin (unknown origin) expressed in HEK293 cells incubated for 4 hrs by dual luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetTransforming growth factor beta-1 proprotein(Homo sapiens (Human))
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Tokyo University Of Pharmacy And Life Sciences
Curated by ChEMBL
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of TGF beta 1 (unknown origin) expressed in HEK293 cells transfected with Smad2/3 responsive reporter plasmid incubated for 4 hrs by dual ...More data for this Ligand-Target Pair
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibitory activity against transcription activator protein-1 (AP-1)More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Mus musculus)
University Of Shizuoka
Curated by ChEMBL
University Of Shizuoka
Curated by ChEMBL
Affinity DataIC50: 9.00E+3nMAssay Description:Antagonist at TRPM8 isolated from mouse dorsal root ganglion cells expressed in HEK T-REx cells assessed as inhibition of menthol-induced intracellul...More data for this Ligand-Target Pair
Affinity DataIC50: 1.18E+4nMAssay Description:Inhibition of the expression of AP1-luciferase by TPA-stimulated NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.33E+4nMAssay Description:Inhibition of the expression of AP1-luciferase by TPA-stimulated NIH3T3 cellsMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Shizuoka
Curated by ChEMBL
University Of Shizuoka
Curated by ChEMBL
Affinity DataIC50: 2.40E+4nMAssay Description:Antagonist activity at human brain TRPV1 expressed in HEK293T cells assessed as inhibition of heat-induced intracellular Ca2+ influx measured for 42 ...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Mus musculus)
University Of Shizuoka
Curated by ChEMBL
University Of Shizuoka
Curated by ChEMBL
Affinity DataIC50: 2.80E+4nMAssay Description:Antagonist at TRPM8 isolated from mouse dorsal root ganglion cells expressed in HEK T-REx cells assessed as inhibition of menthol-induced intracellul...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Mus musculus)
University Of Shizuoka
Curated by ChEMBL
University Of Shizuoka
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Antagonist at TRPM8 isolated from mouse dorsal root ganglion cells expressed in HEK T-REx cells assessed as inhibition of menthol-induced intracellul...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Mus musculus)
University Of Shizuoka
Curated by ChEMBL
University Of Shizuoka
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Antagonist at TRPM8 isolated from mouse dorsal root ganglion cells expressed in HEK T-REx cells assessed as inhibition of icilin-induced intracellula...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
University Of Shizuoka
Curated by ChEMBL
University Of Shizuoka
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Antagonist activity at human brain TRPV1 expressed in HEK293T cells assessed as inhibition of CAP-induced intracellular Ca2+ influx by fluorescence-b...More data for this Ligand-Target Pair
Affinity DataIC50: 5.20E+4nMAssay Description:Inhibitory activity against transcription activator protein-1 (AP-1)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against transcription activator protein-1 (AP-1)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against transcription activator protein-1 (AP-1)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against transcription activator protein-1 (AP-1)More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Mus musculus)
University Of Shizuoka
Curated by ChEMBL
University Of Shizuoka
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist at TRPM8 isolated from mouse dorsal root ganglion cells expressed in HEK T-REx cells assessed as inhibition of menthol-induced intracellul...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against transcription activator protein-1 (AP-1)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against transcription activator protein-1 (AP-1)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against transcription activator protein-1 (AP-1)More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Mus musculus)
University Of Shizuoka
Curated by ChEMBL
University Of Shizuoka
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist at TRPM8 isolated from mouse dorsal root ganglion cells expressed in HEK T-REx cells assessed as inhibition of icilin-induced intracellula...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Mus musculus)
University Of Shizuoka
Curated by ChEMBL
University Of Shizuoka
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist at TRPM8 isolated from mouse dorsal root ganglion cells expressed in HEK T-REx cells assessed as inhibition of icilin-induced intracellula...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against transcription activator protein-1 (AP-1)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against transcription activator protein-1 (AP-1)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against transcription activator protein-1 (AP-1)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against transcription activator protein-1 (AP-1)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against transcription activator protein-1 (AP-1)More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibitory activity against transcription activator protein-1 (AP-1)More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibitory activity against transcription activator protein-1 (AP-1)More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibitory activity against transcription activator protein-1 (AP-1)More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibitory activity against transcription activator protein-1 (AP-1)More data for this Ligand-Target Pair
Affinity DataIC50: 4.20E+5nMAssay Description:Inhibitory activity on AP1 using ELISA based AP1 DNA bindingMore data for this Ligand-Target Pair
Affinity DataIC50: 4.60E+5nMAssay Description:Inhibitory activity on AP1 using ELISA based AP1 DNA bindingMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Mus musculus)
University Of Shizuoka
Curated by ChEMBL
University Of Shizuoka
Curated by ChEMBL
Affinity DataIC50: >5.00E+5nMAssay Description:Antagonist at TRPM8 isolated from mouse dorsal root ganglion cells expressed in HEK T-REx cells assessed as inhibition of icilin-induced intracellula...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Mus musculus)
University Of Shizuoka
Curated by ChEMBL
University Of Shizuoka
Curated by ChEMBL
Affinity DataIC50: >5.00E+5nMAssay Description:Antagonist at TRPM8 isolated from mouse dorsal root ganglion cells expressed in HEK T-REx cells assessed as inhibition of menthol-induced intracellul...More data for this Ligand-Target Pair
Affinity DataIC50: 6.00E+5nMAssay Description:Inhibitory activity on AP1 using ELISA based AP1 DNA bindingMore data for this Ligand-Target Pair
Affinity DataIC50: 6.10E+5nMAssay Description:Inhibitory activity on AP1 using ELISA based AP1 DNA bindingMore data for this Ligand-Target Pair
Affinity DataIC50: 6.50E+5nMAssay Description:Inhibitory activity on AP1 using ELISA based AP1 DNA bindingMore data for this Ligand-Target Pair